TargetReverse transcriptase(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of Human immunodeficiency virus 1 subtype B reverse transcriptase DNA-dependent DNA polymerase activity by gel-based primer extension assa...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of wild type HIV1 subtype B reverse transcriptase by filter-based filtration assayMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of wild type HIV1 subtype B reverse transcriptase by filter-based filtration assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Biochem Therapeutic
Curated by ChEMBL
Biochem Therapeutic
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Ability to inhibit the HIV-1 reverse transcriptase in cord blood mononuclear cells.More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: 36nMAssay Description:Inhibition of DNA-dependent DNA polymerase activity of wild-type Human immunodeficiency virus 1 subtype B reverse transcriptase Y181C mutant by filte...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: 57nMAssay Description:Inhibition of DNA-dependent DNA polymerase activity of wild type HIV1 subtype B reverse transcriptase by gel-based primer extension assayMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: 68nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of wild type HIV1 subtype B reverse transcriptase by filter-based filtration assayMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: 93nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of wild-type Human immunodeficiency virus 1 subtype B reverse transcriptase by filter-based filtr...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: 97nMAssay Description:Inhibition of Human immunodeficiency virus 1 subtype B reverse transcriptase DNA-dependent DNA polymerase activity by gel-based primer extension assa...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: 107nMAssay Description:Inhibition of DNA-dependent DNA polymerase activity of wild-type Human immunodeficiency virus 1 subtype B reverse transcriptase Y181C mutant by filte...More data for this Ligand-Target Pair
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: 112nMAssay Description:Inhibition of Human immunodeficiency virus 1 subtype B reverse transcriptase G190A mutant by filter-based filtration assayMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: 126nMAssay Description:Inhibition of DNA-dependent DNA polymerase activity of wild type HIV1 subtype B reverse transcriptase by gel-based primer extension assayMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: 126nMAssay Description:Inhibition of Human immunodeficiency virus 1 subtype B reverse transcriptase Y181C mutant by filter-based filtration assayMore data for this Ligand-Target Pair
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: 129nMAssay Description:Inhibition of DNA-dependent DNA polymerase activity of wild-type Human immunodeficiency virus 1 subtype B reverse transcriptase G190A mutant by filte...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: 131nMAssay Description:Inhibition of DNA-dependent DNA polymerase activity of wild type HIV1 subtype B reverse transcriptase by gel-based primer extension assayMore data for this Ligand-Target Pair
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: 172nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 subtype B reverse transcriptase M230L mutant by filter-based filtration assayMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: 175nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of wild-type Human immunodeficiency virus 1 subtype B reverse transcriptase by filter-based filtr...More data for this Ligand-Target Pair
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: 191nMAssay Description:Inhibition of Human immunodeficiency virus 1 subtype B reverse transcriptase G190A mutant by filter-based filtration assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Biochem Therapeutic
Curated by ChEMBL
Biochem Therapeutic
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Ability to inhibit the HIV-1 reverse transcriptase in cord blood mononuclear cells.More data for this Ligand-Target Pair
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: 216nMAssay Description:Inhibition of DNA-dependent DNA polymerase activity of wild-type Human immunodeficiency virus 1 subtype B reverse transcriptase G190A mutant by filte...More data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Biochem Therapeutic
Curated by ChEMBL
Biochem Therapeutic
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Ability to inhibit the HIV-1 reverse transcriptase in cord blood mononuclear cells.More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: 257nMAssay Description:Inhibition of Human immunodeficiency virus 1 subtype B reverse transcriptase Y181C mutant by filter-based filtration assayMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Biochem Therapeutic
Curated by ChEMBL
Biochem Therapeutic
Curated by ChEMBL
Affinity DataIC50: 287nMAssay Description:Ability to inhibit the HIV-1 reverse transcriptase in cord blood mononuclear cells.More data for this Ligand-Target Pair
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: 316nMAssay Description:Inhibition of DNA-dependent DNA polymerase activity of wild-type Human immunodeficiency virus 1 subtype B reverse transcriptase G190A mutant by filte...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: 322nMAssay Description:Inhibition of Human immunodeficiency virus 1 subtype B reverse transcriptase DNA-dependent DNA polymerase activity by gel-based primer extension assa...More data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Biochem Therapeutic
Curated by ChEMBL
Biochem Therapeutic
Curated by ChEMBL
Affinity DataIC50: 355nMAssay Description:Ability to inhibit the HIV-1 reverse transcriptase in cord blood mononuclear cells.More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: 370nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of wild-type Human immunodeficiency virus 1 subtype B reverse transcriptase by filter-based filtr...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: 430nMAssay Description:Inhibition of DNA-dependent DNA polymerase activity of wild-type Human immunodeficiency virus 1 subtype B reverse transcriptase Y181C mutant by filte...More data for this Ligand-Target Pair
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: 517nMAssay Description:Inhibition of Human immunodeficiency virus 1 subtype B reverse transcriptase G190A mutant by filter-based filtration assayMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: 570nMAssay Description:Inhibition of Human immunodeficiency virus 1 subtype B reverse transcriptase Y181C mutant by filter-based filtration assayMore data for this Ligand-Target Pair
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: 696nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 subtype B reverse transcriptase M230L mutant by filter-based filtration assayMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: 700nMAssay Description:Inhibition of Human immunodeficiency virus 1 subtype B reverse transcriptase DNA-dependent DNA polymerase activity by gel-based primer extension assa...More data for this Ligand-Target Pair
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: 740nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 subtype B reverse transcriptase M230L mutant by filter-based filtration assayMore data for this Ligand-Target Pair
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: 910nMAssay Description:Inhibition of DNA-dependent DNA polymerase activity of HIV1 subtype B reverse transcriptase M230L mutant by gel-based primer extension assayMore data for this Ligand-Target Pair
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: 1.29E+3nMAssay Description:Inhibition of DNA-dependent DNA polymerase activity of HIV1 subtype B reverse transcriptase M230L mutant by gel-based primer extension assayMore data for this Ligand-Target Pair
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: 1.32E+3nMAssay Description:Inhibition of DNA-dependent DNA polymerase activity of HIV1 subtype B reverse transcriptase M230L mutant by gel-based primer extension assayMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of DNA-dependent DNA polymerase activity of wild type HIV1 subtype B reverse transcriptase by gel-based primer extension assayMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of wild type HIV1 subtype B reverse transcriptase by filter-based filtration assayMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of wild-type Human immunodeficiency virus 1 subtype B reverse transcriptase by filter-based filtr...More data for this Ligand-Target Pair
Affinity DataIC50: 1.52E+4nMAssay Description:Inhibition of human cathepsin DMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human cathepsin DMore data for this Ligand-Target Pair
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: >6.70E+4nMAssay Description:Inhibition of DNA-dependent DNA polymerase activity of wild-type Human immunodeficiency virus 1 subtype B reverse transcriptase G190A mutant by filte...More data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: >6.70E+4nMAssay Description:Inhibition of DNA-dependent DNA polymerase activity of wild-type Human immunodeficiency virus 1 subtype B reverse transcriptase Y181C mutant by filte...More data for this Ligand-Target Pair
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: 1.56E+5nMAssay Description:Inhibition of DNA-dependent DNA polymerase activity of HIV1 subtype B reverse transcriptase M230L mutant by gel-based primer extension assayMore data for this Ligand-Target Pair
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: 1.85E+5nMAssay Description:Inhibition of RNA-dependent DNA polymerase activity of HIV1 subtype B reverse transcriptase M230L mutant by filter-based filtration assayMore data for this Ligand-Target Pair
TargetReverse transcriptase protein(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of Human immunodeficiency virus 1 subtype B reverse transcriptase G190A mutant by filter-based filtration assayMore data for this Ligand-Target Pair
TargetReverse transcriptase(Human immunodeficiency virus 1)
Mcgill University Aids Centre
Curated by ChEMBL
Mcgill University Aids Centre
Curated by ChEMBL
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of Human immunodeficiency virus 1 subtype B reverse transcriptase Y181C mutant by filter-based filtration assayMore data for this Ligand-Target Pair