TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
TargetGastrin/cholecystokinin type B receptor(GUINEA PIG)
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Affinity DataKi: 0.100nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha-1B receptor in rat liver membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.230nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha-1A receptor in rat submaxillary gland membranesMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(GUINEA PIG)
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
TargetGastrin/cholecystokinin type B receptor(RAT)
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Affinity DataKi: 0.610nMAssay Description:Displacement of [3H]prazosin from alpha1B adrenoceptor in rat liver membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.630nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha-1B receptor in rat liver membranesMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(GUINEA PIG)
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Fujisawa Pharmaceutical
Curated by PDSP Ki Database
Affinity DataKi: 1.10nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha-1B receptor in rat liver membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha-1B receptor in rat liver membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Displacement of [3H]prazosin from alpha1B adrenoceptor in rat liver membranesMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Displacement of [3H]prazosin from alpha1B adrenoceptor in rat liver membranesMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha-1B receptor in rat liver membranesMore data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Displacement of [3H]prazosin from alpha1B adrenoceptor in rat liver membranesMore data for this Ligand-Target Pair
Affinity DataKi: 4.80nMAssay Description:Displacement of [3H]prazosin from alpha1B adrenoceptor in rat liver membranesMore data for this Ligand-Target Pair
Affinity DataKi: 7.10nMAssay Description:Displacement of [3H]prazosin from alpha1B adrenoceptor in rat liver membranesMore data for this Ligand-Target Pair
Affinity DataKi: 7.20nMAssay Description:Displacement of [3H]prazosin from alpha1B adrenoceptor in rat liver membranesMore data for this Ligand-Target Pair
Affinity DataKi: 7.5nMAssay Description:Displacement of [3H]prazosin from alpha1B adrenoceptor in rat liver membranesMore data for this Ligand-Target Pair
Affinity DataKi: 7.70nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha-1B receptor in rat liver membranesMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Eisai
Curated by ChEMBL
Eisai
Curated by ChEMBL
Affinity DataKi: 9.5nMAssay Description:Inhibitory activity against AcetylcholinesteraseMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Eisai
Curated by ChEMBL
Eisai
Curated by ChEMBL
Affinity DataKi: 9.5nMAssay Description:Inhibitory activity against AcetylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Displacement of [3H]prazosin from alpha1B adrenoceptor in rat liver membranesMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Displacement of [3H]prazosin from alpha1B adrenoceptor in rat liver membranesMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha-1B receptor in rat liver membranesMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha-1B receptor in rat liver membranesMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Displacement of [3H]prazosin from alpha1A adrenoceptor in rat submaxillary gland membraneMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Binding affinity to human recombinant alpha1D adrenoceptorMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Eisai
Curated by ChEMBL
Eisai
Curated by ChEMBL
Affinity DataKi: 17.5nMAssay Description:Inhibitory activity was calculated for the model Acetylcholinesterase (Expt-1)More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Eisai
Curated by ChEMBL
Eisai
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Inhibitory activity was calculated for the model Acetylcholinesterase (Expt-1)More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Eisai
Curated by ChEMBL
Eisai
Curated by ChEMBL
Affinity DataKi: 19nMAssay Description:Inhibitory activity was calculated for the model Acetylcholinesterase (Expt-1)More data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha-1A receptor in rat submaxillary gland membranesMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Binding affinity to human adrenergic Alpha-1D receptorMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Displacement of [3H]prazosin from alpha1A adrenoceptor in rat submaxillary gland membraneMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Eisai
Curated by ChEMBL
Eisai
Curated by ChEMBL
Affinity DataKi: 27nMAssay Description:Inhibitory activity against AcetylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:Binding affinity to human adrenergic Alpha-1D receptorMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Eisai
Curated by ChEMBL
Eisai
Curated by ChEMBL
Affinity DataKi: 37.6nMAssay Description:Inhibitory activity was calculated for the model Acetylcholinesterase (Expt-2)More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Eisai
Curated by ChEMBL
Eisai
Curated by ChEMBL
Affinity DataKi: 38nMAssay Description:Inhibitory activity was calculated for the model Acetylcholinesterase (Expt-2)More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Eisai
Curated by ChEMBL
Eisai
Curated by ChEMBL
Affinity DataKi: 47nMAssay Description:Inhibitory activity was calculated for the model Acetylcholinesterase (Expt-2)More data for this Ligand-Target Pair
Affinity DataKi: 47nMAssay Description:Displacement of [3H]prazosin from alpha1B adrenoceptor in rat liver membranesMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Displacement of [3H]prazosin from alpha1A adrenoceptor in rat submaxillary gland membraneMore data for this Ligand-Target Pair
Affinity DataKi: 51nMAssay Description:Displacement of [3H]prazosin from alpha1A adrenoceptor in rat submaxillary gland membraneMore data for this Ligand-Target Pair
Affinity DataKi: 53nMAssay Description:Displacement of [3H]prazosin from alpha1A adrenoceptor in rat submaxillary gland membraneMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Eisai
Curated by ChEMBL
Eisai
Curated by ChEMBL
Affinity DataKi: 54nMAssay Description:Inhibitory activity against AcetylcholinesteraseMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Eisai
Curated by ChEMBL
Eisai
Curated by ChEMBL
Affinity DataKi: 54nMAssay Description:Inhibitory activity was calculated for the model Acetylcholinesterase (Expt-2)More data for this Ligand-Target Pair
Affinity DataKi: 56nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha-1A receptor in rat submaxillary gland membranesMore data for this Ligand-Target Pair
Affinity DataKi: 57nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha-1A receptor in rat submaxillary gland membranesMore data for this Ligand-Target Pair
Affinity DataKi: 57nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha-1A receptor in rat submaxillary gland membranesMore data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha-1A receptor in rat submaxillary gland membranesMore data for this Ligand-Target Pair