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Found 235 with Last Name = 'waki' and Initial = 'm'
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Fujisawa Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM84928(CAS_125368 | FK 1052 | NSC_125368)
Affinity DataKi:  0.0100nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Fujisawa Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM84928(CAS_125368 | FK 1052 | NSC_125368)
Affinity DataKi:  0.0100nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGastrin/cholecystokinin type B receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50084033(1H-Indole-2-carboxylic acid [(R)-1-(2-fluoro-pheny...)
Affinity DataKi:  0.0600nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM29568(CHEMBL2 | PRAZOSIN | PRAZOSIN HYDROCHLORIDE | [3H]...)
Affinity DataKi:  0.100nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha-1B receptor in rat liver membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM29568(CHEMBL2 | PRAZOSIN | PRAZOSIN HYDROCHLORIDE | [3H]...)
Affinity DataKi:  0.230nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha-1A receptor in rat submaxillary gland membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.230nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
Fujisawa Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50084033(1H-Indole-2-carboxylic acid [(R)-1-(2-fluoro-pheny...)
Affinity DataKi:  0.400nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50115122(CHEMBL3609360)
Affinity DataKi:  0.610nMAssay Description:Displacement of [3H]prazosin from alpha1B adrenoceptor in rat liver membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50187753(6-fluoro-3-(1-(3-(piperidin-1-yl)propyl)piperidin-...)
Affinity DataKi:  0.630nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha-1B receptor in rat liver membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(GUINEA PIG)
Fujisawa Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.670nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50187752(3-(1-(4-(piperidin-1-yl)butyl)piperidin-4-yl)-1H-i...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha-1B receptor in rat liver membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50187747(3-(1-(5-(piperidin-1-yl)pentyl)piperidin-4-yl)-1H-...)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha-1B receptor in rat liver membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50115121(CHEMBL3609359)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]prazosin from alpha1B adrenoceptor in rat liver membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50187749(3-(1-(3-(piperidin-1-yl)propyl)piperidin-4-yl)-1H-...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]prazosin from alpha1B adrenoceptor in rat liver membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50187749(3-(1-(3-(piperidin-1-yl)propyl)piperidin-4-yl)-1H-...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha-1B receptor in rat liver membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50115118(CHEMBL3609357)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]prazosin from alpha1B adrenoceptor in rat liver membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50115188(CHEMBL3609353)
Affinity DataKi:  4.80nMAssay Description:Displacement of [3H]prazosin from alpha1B adrenoceptor in rat liver membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50115120(CHEMBL3609358)
Affinity DataKi:  7.10nMAssay Description:Displacement of [3H]prazosin from alpha1B adrenoceptor in rat liver membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50115123(CHEMBL3609354)
Affinity DataKi:  7.20nMAssay Description:Displacement of [3H]prazosin from alpha1B adrenoceptor in rat liver membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50115114(CHEMBL3609356)
Affinity DataKi:  7.5nMAssay Description:Displacement of [3H]prazosin from alpha1B adrenoceptor in rat liver membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50187757(1-(3-(4-(benzofuran-3-yl)piperidin-1-yl)propyl)pip...)
Affinity DataKi:  7.70nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha-1B receptor in rat liver membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Eisai

Curated by ChEMBL
LigandPNGBDBM50422179(CHEMBL2093912)
Affinity DataKi:  9.5nMAssay Description:Inhibitory activity against AcetylcholinesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Eisai

Curated by ChEMBL
LigandPNGBDBM50422179(CHEMBL2093912)
Affinity DataKi:  9.5nMAssay Description:Inhibitory activity against AcetylcholinesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50115113(CHEMBL3609355)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]prazosin from alpha1B adrenoceptor in rat liver membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50115190(CHEMBL3609351)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]prazosin from alpha1B adrenoceptor in rat liver membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50187754(3-(1-(3-(piperidin-1-yl)propyl)piperidin-4-yl)benz...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha-1B receptor in rat liver membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50187748(5-fluoro-3-(1-(3-(piperidin-1-yl)propyl)piperidin-...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha-1B receptor in rat liver membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50115190(CHEMBL3609351)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]prazosin from alpha1A adrenoceptor in rat submaxillary gland membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50115122(CHEMBL3609360)
Affinity DataKi:  16nMAssay Description:Binding affinity to human recombinant alpha1D adrenoceptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Eisai

Curated by ChEMBL
LigandPNGBDBM50422179(CHEMBL2093912)
Affinity DataKi:  17.5nMAssay Description:Inhibitory activity was calculated for the model Acetylcholinesterase (Expt-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Eisai

Curated by ChEMBL
LigandPNGBDBM50422179(CHEMBL2093912)
Affinity DataKi:  18nMAssay Description:Inhibitory activity was calculated for the model Acetylcholinesterase (Expt-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Eisai

Curated by ChEMBL
LigandPNGBDBM50029941(2-[2-(1-Benzyl-piperidin-4-yl)-ethyl]-5,6-dimethox...)
Affinity DataKi:  19nMAssay Description:Inhibitory activity was calculated for the model Acetylcholinesterase (Expt-1)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50187753(6-fluoro-3-(1-(3-(piperidin-1-yl)propyl)piperidin-...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha-1A receptor in rat submaxillary gland membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50187753(6-fluoro-3-(1-(3-(piperidin-1-yl)propyl)piperidin-...)
Affinity DataKi:  22nMAssay Description:Binding affinity to human adrenergic Alpha-1D receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50115122(CHEMBL3609360)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]prazosin from alpha1A adrenoceptor in rat submaxillary gland membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Eisai

Curated by ChEMBL
LigandPNGBDBM50029941(2-[2-(1-Benzyl-piperidin-4-yl)-ethyl]-5,6-dimethox...)
Affinity DataKi:  27nMAssay Description:Inhibitory activity against AcetylcholinesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50187747(3-(1-(5-(piperidin-1-yl)pentyl)piperidin-4-yl)-1H-...)
Affinity DataKi:  37nMAssay Description:Binding affinity to human adrenergic Alpha-1D receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Eisai

Curated by ChEMBL
LigandPNGBDBM50422179(CHEMBL2093912)
Affinity DataKi:  37.6nMAssay Description:Inhibitory activity was calculated for the model Acetylcholinesterase (Expt-2)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Eisai

Curated by ChEMBL
LigandPNGBDBM50422179(CHEMBL2093912)
Affinity DataKi:  38nMAssay Description:Inhibitory activity was calculated for the model Acetylcholinesterase (Expt-2)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Eisai

Curated by ChEMBL
LigandPNGBDBM50029941(2-[2-(1-Benzyl-piperidin-4-yl)-ethyl]-5,6-dimethox...)
Affinity DataKi:  47nMAssay Description:Inhibitory activity was calculated for the model Acetylcholinesterase (Expt-2)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50115189(CHEMBL3609352)
Affinity DataKi:  47nMAssay Description:Displacement of [3H]prazosin from alpha1B adrenoceptor in rat liver membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50115118(CHEMBL3609357)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]prazosin from alpha1A adrenoceptor in rat submaxillary gland membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50115114(CHEMBL3609356)
Affinity DataKi:  51nMAssay Description:Displacement of [3H]prazosin from alpha1A adrenoceptor in rat submaxillary gland membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50115123(CHEMBL3609354)
Affinity DataKi:  53nMAssay Description:Displacement of [3H]prazosin from alpha1A adrenoceptor in rat submaxillary gland membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Eisai

Curated by ChEMBL
LigandPNGBDBM50029912(2-(1-Benzyl-piperidin-4-yl)-5,6-dimethoxy-indan-1-...)
Affinity DataKi:  54nMAssay Description:Inhibitory activity against AcetylcholinesteraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Eisai

Curated by ChEMBL
LigandPNGBDBM50029912(2-(1-Benzyl-piperidin-4-yl)-5,6-dimethoxy-indan-1-...)
Affinity DataKi:  54nMAssay Description:Inhibitory activity was calculated for the model Acetylcholinesterase (Expt-2)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50187752(3-(1-(4-(piperidin-1-yl)butyl)piperidin-4-yl)-1H-i...)
Affinity DataKi:  56nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha-1A receptor in rat submaxillary gland membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50187747(3-(1-(5-(piperidin-1-yl)pentyl)piperidin-4-yl)-1H-...)
Affinity DataKi:  57nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha-1A receptor in rat submaxillary gland membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50187754(3-(1-(3-(piperidin-1-yl)propyl)piperidin-4-yl)benz...)
Affinity DataKi:  57nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha-1A receptor in rat submaxillary gland membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50187757(1-(3-(4-(benzofuran-3-yl)piperidin-1-yl)propyl)pip...)
Affinity DataKi:  60nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha-1A receptor in rat submaxillary gland membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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