Affinity DataKi: 0.00500nMAssay Description:Competitive reversible inhibition of human C-terminal His6-tagged CD73 expressed in HEK293 cells using AMP as substrate preincubated with substrate f...More data for this Ligand-Target Pair
Affinity DataKi: 0.0500nMAssay Description:Binding affinity for 5-hydroxytryptamine 2A receptor expressed in 3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.130nMAssay Description:Binding affinity for 5-hydroxytryptamine 2A receptor expressed in 3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.170nMAssay Description:Binding affinity for 5-hydroxytryptamine 2A receptor expressed in 3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.170nMAssay Description:Binding affinity for 5-hydroxytryptamine 2A receptor expressed in 3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.180nMAssay Description:Binding affinity for 5-hydroxytryptamine 2A receptor expressed in 3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.180nMAssay Description:Binding affinity for 5-hydroxytryptamine 2A receptor expressed in 3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.220nMAssay Description:Binding affinity for 5-hydroxytryptamine 2A receptor expressed in 3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.240nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human H3 receptor expressed in HEK-293 cell membrane after 90 mins by liquid scintillation counting ...More data for this Ligand-Target Pair
Affinity DataKi: 0.280nMAssay Description:Binding affinity for 5-hydroxytryptamine 2A receptor expressed in 3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.280nMAssay Description:Binding affinity for 5-hydroxytryptamine 2A receptor expressed in 3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.280nMAssay Description:Binding affinity for 5-hydroxytryptamine 2A receptor expressed in 3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.280nMAssay Description:Binding affinity for 5-hydroxytryptamine 2A receptor expressed in 3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.290nMAssay Description:Binding affinity for 5-hydroxytryptamine 2A receptor expressed in 3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Binding affinity for 5-hydroxytryptamine 2A receptor expressed in 3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.310nMAssay Description:Binding affinity for 5-hydroxytryptamine 2A receptor expressed in 3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.320nMAssay Description:Binding affinity for 5-hydroxytryptamine 2A receptor expressed in 3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.440nMAssay Description:Binding affinity for 5-hydroxytryptamine 2A receptor expressed in 3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.540nMAssay Description:Displacement of [125I](+/-)DOI from human 5-HT2B receptor trasfected in CHO cell membrane after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 0.590nMAssay Description:Binding affinity for 5-hydroxytryptamine 2A receptor expressed in 3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.610nMAssay Description:Binding affinity for 5-hydroxytryptamine 2A receptor expressed in 3T3 cellsMore data for this Ligand-Target Pair
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform(Homo sapiens (Human))
Arcus Biosciences
Curated by ChEMBL
Arcus Biosciences
Curated by ChEMBL
Affinity DataKi: 0.700nMAssay Description:Inhibition of PI3Kgamma (unknown origin) at 10 uM using PIP2 as substrate preincubated for 60 mins followed by substrate addition and measured after ...More data for this Ligand-Target Pair
Affinity DataKi: 0.75nMAssay Description:Binding affinity for 5-hydroxytryptamine 2A receptor expressed in 3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.933nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human H3 receptor expressed in HEK-293 cell membrane after 90 mins by liquid scintillation counting ...More data for this Ligand-Target Pair
Affinity DataKi: 0.970nMAssay Description:Displacement of [125I](+/-)DOI from human 5-HT2B receptor trasfected in CHO cell membrane after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Displacement of [125I](+/-)DOI from human 5-HT2B receptor trasfected in CHO cell membrane after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1.06nMAssay Description:Binding affinity for 5-hydroxytryptamine 2A receptor expressed in 3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.07nMAssay Description:Binding affinity for 5-hydroxytryptamine 2A receptor expressed in 3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.24nMAssay Description:Binding affinity for 5-hydroxytryptamine 2A receptor expressed in 3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Displacement of [125I](+/-)DOI from human 5-HT2B receptor trasfected in CHO cell membrane after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 2.15nMAssay Description:Binding affinity for 5-hydroxytryptamine 2A receptor expressed in 3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Displacement of [125I](+/-)DOI from human 5-HT2B receptor trasfected in CHO cell membrane after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 2.23nMAssay Description:Binding affinity for 5-hydroxytryptamine 2A receptor expressed in 3T3 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Displacement of [125I]Iodoproxyfan from human histamine H3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Displacement of [125I]iodoproxyfan human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Inhibition of monoamine reuptake at norepinephrine transporterMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Binding affinity to NETMore data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:Binding affinity to NETMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity against Dopamine receptor D2 expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Inhibition of monoamine reuptake at norepinephrine transporterMore data for this Ligand-Target Pair
Affinity DataKi: 5.20nMAssay Description:Binding affinity to NETMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Inhibition of monoamine reuptake at norepinephrine transporterMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Inhibition of monoamine reuptake at norepinephrine transporterMore data for this Ligand-Target Pair
Affinity DataKi: 7.10nMAssay Description:Displacement of [125I](+/-)DOI from human 5-HT2B receptor trasfected in CHO cell membrane after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 7.40nMAssay Description:Displacement of [125I]Iodoproxyfan from human histamine H3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.70nMAssay Description:Binding affinity to NETMore data for this Ligand-Target Pair
Affinity DataKi: 7.70nMAssay Description:Binding affinity to NETMore data for this Ligand-Target Pair
Affinity DataKi: 7.93nMAssay Description:Binding affinity at NETMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Inhibition of monoamine reuptake at norepinephrine transporterMore data for this Ligand-Target Pair