Affinity DataKi: 0.200nMAssay Description:Antagonist activity at human adenosine A1 receptor expressed in HEK293 cells assessed as reduction in CPA-mediated inhibition of forskolin-stimulated...More data for this Ligand-Target Pair
Affinity DataKi: 0.280nMAssay Description:Antagonist activity at human adenosine A1 receptor expressed in HEK293 cells assessed as reduction in CPA-mediated inhibition of forskolin-stimulated...More data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Antagonist activity at human adenosine receptor A2b expressed in HEK293 cells assessed as inhibition of NECA-induced cAMP level preincubated for 15 m...More data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Displacement of [3H]-MRS-1754 from human adenosine receptor A2b expressed in HEK293 cell membranes after 90 mins by liquid scintillation counting met...More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Displacement of [3H]-MRS-1754 from human adenosine receptor A2b expressed in HEK293 cell membranes after 90 mins by liquid scintillation counting met...More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Displacement of [3H]-MRS-1754 from human adenosine receptor A2b expressed in HEK293 cell membranes after 90 mins by liquid scintillation counting met...More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in HEK293 cell membranes after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]-MRS-1754 from human adenosine receptor A2b expressed in HEK293 cell membranes after 90 mins by liquid scintillation counting met...More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Displacement of [3H]-MRS-1754 from human adenosine A2B receptor expressed in HEK293 cell membranes after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]-MRS-1754 from human adenosine A2B receptor expressed in HEK293 cell membranes after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]-MRS-1754 from human adenosine receptor A2b expressed in HEK293 cell membranes after 90 mins by liquid scintillation counting met...More data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]-MRS-1754 from human adenosine A2B receptor expressed in HEK293 cell membranes after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]-MRS-1754 from human adenosine A2B receptor expressed in HEK293 cell membranes after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in HEK293 cells assessed as inhibition of NECA-induced increase in cAMP accumulation in...More data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Displacement of [3H]-MRS-1754 from human adenosine receptor A2b expressed in HEK293 cell membranes after 90 mins by liquid scintillation counting met...More data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Displacement of [125I]ABOPX from human adenosine receptor A2b expressed in HEK293 cell membranes after 3 hrs by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Antagonist activity at human adenosine A1 receptor expressed in HEK293 cells assessed as reduction in CPA-mediated inhibition of forskolin-stimulated...More data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Displacement of [3H]-MRS-1754 from human adenosine A2B receptor expressed in HEK293 cell membranes after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Antagonist activity at human adenosine A1 receptor expressed in HEK293 cells assessed as reduction in CPA-mediated inhibition of forskolin-stimulated...More data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Displacement of [3H]-MRS-1754 from human adenosine receptor A2b expressed in HEK293 cell membranes after 90 mins by liquid scintillation counting met...More data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:Displacement of [3H]-MRS-1754 from human adenosine A2B receptor expressed in HEK293 cell membranes after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Inhibition of bovine adenosine deaminase pre-incubated for 5 mins before adenosine additionMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Displacement of [3H]-MRS-1754 from human adenosine receptor A2b expressed in HEK293 cell membranes after 90 mins by liquid scintillation counting met...More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Displacement of [3H]-MRS-1754 from human adenosine A2B receptor expressed in HEK293 cell membranes after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:Displacement of [3H]-MRS-1754 from human adenosine A2B receptor expressed in HEK293 cell membranes after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Displacement of [3H]-MRS-1754 from human adenosine receptor A2b expressed in HEK293 cell membranes after 90 mins by liquid scintillation counting met...More data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in HEK293 cell membranes after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Displacement of [3H]-MRS-1754 from human adenosine A2B receptor expressed in HEK293 cell membranes after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:Displacement of [3H]-MRS-1754 from human adenosine A2B receptor expressed in HEK293 cell membranes after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Displacement of [3H]-MRS-1754 from human adenosine receptor A2b expressed in HEK293 cell membranes after 90 mins by liquid scintillation counting met...More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Displacement of [3H]-MRS-1754 from human adenosine receptor A2b expressed in HEK293 cell membranes after 90 mins by liquid scintillation counting met...More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Antagonist activity at human adenosine receptor A2b expressed in HEK293 cells assessed as inhibition of NECA-induced cAMP level preincubated for 15 m...More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Displacement of [3H]-MRS-1754 from human adenosine receptor A2b expressed in HEK293 cell membranes after 90 mins by liquid scintillation counting met...More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Antagonist activity at human adenosine receptor A2b expressed in HEK293 cells assessed as inhibition of NECA-induced cAMP level preincubated for 15 m...More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Displacement of [3H]-MRS-1754 from human adenosine receptor A2b expressed in HEK293 cell membranes after 90 mins by liquid scintillation counting met...More data for this Ligand-Target Pair
Affinity DataKi: 4.5nMAssay Description:Displacement of [3H]-MRS-1754 from human adenosine receptor A2b expressed in HEK293 cell membranes after 90 mins by liquid scintillation counting met...More data for this Ligand-Target Pair