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Found 153 with Last Name = 'wang' and Initial = 'qj'
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50366620(RESINIFERATOXIN)
Affinity DataKi:  0.0230nMAssay Description:In vitro binding affinity towards vanilloid receptor by [3H]RTX displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86434(12-Deoxyphorbol 13-phenylacetate | CAS_105100 | NS...)
Affinity DataKi:  0.140nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86429(CAS_6437389 | NSC_6437389 | Thymeleatoxin | Thymel...)
Affinity DataKi:  0.220nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86431(CAS_4179 | Mezerein | NSC_4179)
Affinity DataKi:  0.270nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86429(CAS_6437389 | NSC_6437389 | Thymeleatoxin | Thymel...)
Affinity DataKi:  0.290nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolycystin-1(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86434(12-Deoxyphorbol 13-phenylacetate | CAS_105100 | NS...)
Affinity DataKi:  0.350nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPolycystin-1(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86431(CAS_4179 | Mezerein | NSC_4179)
Affinity DataKi:  0.430nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolycystin-1(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86432((-)-Octylindolactam V | CAS_159320 | NSC_159320)
Affinity DataKi:  0.450nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86432((-)-Octylindolactam V | CAS_159320 | NSC_159320)
Affinity DataKi:  0.530nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86431(CAS_4179 | Mezerein | NSC_4179)
Affinity DataKi:  0.550nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86434(12-Deoxyphorbol 13-phenylacetate | CAS_105100 | NS...)
Affinity DataKi:  0.560nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86432((-)-Octylindolactam V | CAS_159320 | NSC_159320)
Affinity DataKi:  0.770nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86429(CAS_6437389 | NSC_6437389 | Thymeleatoxin | Thymel...)
Affinity DataKi:  1.31nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86435(B8-DL-B8 | B8-DL-B8 (low PS))
Affinity DataKi:  2.90nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolycystin-1(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86429(CAS_6437389 | NSC_6437389 | Thymeleatoxin | Thymel...)
Affinity DataKi:  3.20nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86435(B8-DL-B8 | B8-DL-B8 (low PS))
Affinity DataKi:  3.57nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolycystin-1(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86429(CAS_6437389 | NSC_6437389 | Thymeleatoxin | Thymel...)
Affinity DataKi:  3.85nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86433(CAS_454217 | NSC_454217 | Prostratin)
Affinity DataKi:  4.83nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86430((-)-Indolactam V | (-)-Indolactam V (low PS) | CAS...)
Affinity DataKi:  8.16nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86435(B8-DL-B8 | B8-DL-B8 (low PS))
Affinity DataKi:  10nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86429(CAS_6437389 | NSC_6437389 | Thymeleatoxin | Thymel...)
Affinity DataKi:  10.7nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolycystin-1(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86435(B8-DL-B8 | B8-DL-B8 (low PS))
Affinity DataKi:  10.8nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86435(B8-DL-B8 | B8-DL-B8 (low PS))
Affinity DataKi:  11.6nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86430((-)-Indolactam V | (-)-Indolactam V (low PS) | CAS...)
Affinity DataKi:  12.6nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolycystin-1(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86433(CAS_454217 | NSC_454217 | Prostratin)
Affinity DataKi:  12.9nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86433(CAS_454217 | NSC_454217 | Prostratin)
Affinity DataKi:  24.6nMMore data for this Ligand-Target Pair
TargetPolycystin-1(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86435(B8-DL-B8 | B8-DL-B8 (low PS))
Affinity DataKi:  26.1nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86436(3-hydroxy-2-[4-methyl-3-(methylethyl)pentanoyloxy]...)
Affinity DataKi:  28.6nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86436(3-hydroxy-2-[4-methyl-3-(methylethyl)pentanoyloxy]...)
Affinity DataKi:  30.9nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolycystin-1(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86430((-)-Indolactam V | (-)-Indolactam V (low PS) | CAS...)
Affinity DataKi:  38nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86430((-)-Indolactam V | (-)-Indolactam V (low PS) | CAS...)
Affinity DataKi:  43.1nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolycystin-1(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86430((-)-Indolactam V | (-)-Indolactam V (low PS) | CAS...)
Affinity DataKi:  48.1nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolycystin-1(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86436(3-hydroxy-2-[4-methyl-3-(methylethyl)pentanoyloxy]...)
Affinity DataKi:  90nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolycystin-1(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86440(CAS_104731 | NSC_104731 | OAG)
Affinity DataKi:  146nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86440(CAS_104731 | NSC_104731 | OAG)
Affinity DataKi:  224nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Pittsburgh

Curated by PDSP Ki Database
LigandPNGBDBM86440(CAS_104731 | NSC_104731 | OAG)
Affinity DataKi:  230nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50082250(2,2-Dimethyl-propionic acid 2-{[2-(4-hydroxy-3-met...)
Affinity DataKi:  295nMAssay Description:In vitro binding affinity towards vanilloid receptor by [3H]RTX displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50082239(2,2-Dimethyl-propionic acid 2-benzyl-3-[2-(4-hydro...)
Affinity DataKi:  404nMAssay Description:In vitro binding affinity towards vanilloid receptor by [3H]RTX displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50082243((E)-4-Benzyl-5-[2-(4-hydroxy-3-methoxy-phenyl)-ace...)
Affinity DataKi:  480nMAssay Description:In vitro binding affinity towards vanilloid receptor by [3H]RTX displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50082248(2,2-Dimethyl-propionic acid (E)-2-{[2-(4-hydroxy-3...)
Affinity DataKi:  1.22E+3nMAssay Description:In vitro binding affinity towards vanilloid receptor by [3H]RTX displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50082242(2-[4-(2-Amino-ethoxy)-3-methoxy-phenyl]-N-[3-(3,4-...)
Affinity DataKi:  1.40E+3nMAssay Description:In vitro binding affinity towards vanilloid receptor by [3H]RTX displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50082252(7-Methyl-oct-6-enoic acid 4-hydroxy-3-methoxy-benz...)
Affinity DataKi:  5.31E+3nMAssay Description:In vitro binding affinity towards vanilloid receptor by [3H]RTX displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50082240(Acetic acid (E)-2-{[2-(4-hydroxy-3-methoxy-phenyl)...)
Affinity DataKi:  1.29E+4nMAssay Description:In vitro binding affinity towards vanilloid receptor by [3H]RTX displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50082237((E)-4-Benzyl-5-[2-(4-hydroxy-3-methoxy-phenyl)-ace...)
Affinity DataKi:  1.35E+4nMAssay Description:In vitro binding affinity towards vanilloid receptor by [3H]RTX displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50082238(Acetic acid 2-benzyl-3-[2-(4-hydroxy-3-methoxy-phe...)
Affinity DataKi:  1.93E+4nMAssay Description:In vitro binding affinity towards vanilloid receptor by [3H]RTX displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50082236(Acetic acid (Z)-2-{[2-(4-hydroxy-3-methoxy-phenyl)...)
Affinity DataKi:  2.92E+4nMAssay Description:In vitro binding affinity towards vanilloid receptor by [3H]RTX displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50082245(Acetic acid 2-{[2-(4-hydroxy-3-methoxy-phenyl)-ace...)
Affinity DataKi:  4.52E+4nMAssay Description:In vitro binding affinity towards vanilloid receptor by [3H]RTX displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50082246(Acetic acid 2-benzyloxymethyl-3-[2-(4-hydroxy-3-me...)
Affinity DataKi:  7.80E+4nMAssay Description:In vitro binding affinity towards vanilloid receptor by [3H]RTX displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50082244((4-Hydroxy-3-methoxy-phenyl)-acetic acid (Z)-2-ace...)
Affinity DataKi: >1.00E+5nMAssay Description:In vitro binding affinity towards vanilloid receptor by [3H]RTX displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50082253((4-Hydroxy-3-methoxy-phenyl)-acetic acid 2-acetoxy...)
Affinity DataKi: >1.00E+5nMAssay Description:In vitro binding affinity towards vanilloid receptor by [3H]RTX displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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