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Found 149 with Last Name = 'wang' and Initial = 'sb'
TargetBeta-arrestin-1(RABBIT)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM82381(L-659,989, (-))
Affinity DataKi:  0.510nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-arrestin-1(RABBIT)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50002829((2S,5S)-2-(3-Methanesulfonyl-5-methoxy-4-propoxy-p...)
Affinity DataKi:  1.10nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM82381(L-659,989, (-))
Affinity DataKi:  5.48nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-arrestin-1(RABBIT)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50002829((2S,5S)-2-(3-Methanesulfonyl-5-methoxy-4-propoxy-p...)
Affinity DataKi:  12.2nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50002829((2S,5S)-2-(3-Methanesulfonyl-5-methoxy-4-propoxy-p...)
Affinity DataKi:  14.3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50000714(3-[4-(2-Chloro-phenyl)-9-methyl-6H-1-thia-5,7,8,9a...)
Affinity DataKi:  79.3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50002829((2S,5S)-2-(3-Methanesulfonyl-5-methoxy-4-propoxy-p...)
Affinity DataKi:  152nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-arrestin-1(RABBIT)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50002829((2S,5S)-2-(3-Methanesulfonyl-5-methoxy-4-propoxy-p...)
Affinity DataKi:  205nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50002829((2S,5S)-2-(3-Methanesulfonyl-5-methoxy-4-propoxy-p...)
Affinity DataKi:  1.11E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50021572((2S,3S)-2-(3,4-Dimethoxy-phenyl)-3-methyl-5-propyl...)
Affinity DataIC50:  0nMAssay Description:Inhibitor concentration required to block 50% of the specific [3H]PAF binding to rabbit platelet membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50408421(CHEMBL2113725)
Affinity DataIC50:  2nMAssay Description:Displacement of [3H]-PAF from PAF receptor of human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50002823(2-{3-Methoxy-2-propoxy-5-[(2S,5S)-5-(3,4,5-trimeth...)
Affinity DataIC50:  6nMAssay Description:Displacement of [3H]-PAF from PAF receptor of human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50286666(CHEMBL347382 | N-hydroxy-N'-[3-methoxy-5-(5-(3,4,5...)
Affinity DataIC50:  8nMAssay Description:In vitro affinity for human PAF receptor on platelet membranes using [3H]-PAF displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50286666(CHEMBL347382 | N-hydroxy-N'-[3-methoxy-5-(5-(3,4,5...)
Affinity DataIC50:  8nMAssay Description:In vitro inhibition of 5-lipoxygenase in RBL-2H3 (Rat basophilic leukaemia) cells.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50408414(CHEMBL2113720)
Affinity DataIC50:  10nMAssay Description:Displacement of [3H]-PAF from PAF receptor of human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50408417(CHEMBL2113724)
Affinity DataIC50:  17nMAssay Description:Inhibition of 5-lipoxygenase mediated conversion of [14C]-arachidonic acid to leukotrienes in RBL-2H3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50286665(CHEMBL160692 | N-hydroxy-N'-[3-methoxy-5-(5-(3,4,5...)
Affinity DataIC50:  17nMAssay Description:In vitro affinity for human PAF receptor on platelet membranes using [3H]-PAF displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50286665(CHEMBL160692 | N-hydroxy-N'-[3-methoxy-5-(5-(3,4,5...)
Affinity DataIC50:  17nMAssay Description:In vitro inhibition of 5-lipoxygenase in RBL-2H3 (Rat basophilic leukaemia) cells.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50286669(5-lipoxygenase inhibitor | CHEMBL348609)
Affinity DataIC50:  17nMAssay Description:In vitro affinity for human PAF receptor on platelet membranes using [3H]-PAF displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50408419(CHEMBL2113723)
Affinity DataIC50:  19nMAssay Description:Inhibition of 5-lipoxygenase mediated conversion of [14C]-arachidonic acid to leukotrienes in RBL-2H3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50408413(CHEMBL2113727)
Affinity DataIC50:  20nMAssay Description:Displacement of [3H]-PAF from PAF receptor of human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50002831((2R,5R)-2,5-Bis-(3,4,5-trimethoxy-phenyl)-tetrahyd...)
Affinity DataIC50:  20nMAssay Description:Inhibition of PAF receptor binding to rabbit platelet plasma membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50408419(CHEMBL2113723)
Affinity DataIC50:  21nMAssay Description:Displacement of [3H]-PAF from PAF receptor of human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50408418(CHEMBL2113722)
Affinity DataIC50:  22nMAssay Description:Displacement of [3H]-PAF from PAF receptor of human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50408422(CHEMBL2113721)
Affinity DataIC50:  23nMAssay Description:Displacement of [3H]-PAF from PAF receptor of human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50408424(CHEMBL2113733)
Affinity DataIC50:  25nMAssay Description:Displacement of [3H]-PAF from PAF receptor of human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50286661(CHEMBL160290 | N-hydroxy-N'-[3-methoxy-5-(5-(3,4,5...)
Affinity DataIC50:  25nMAssay Description:In vitro affinity for human PAF receptor on platelet membranes using [3H]-PAF displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50286661(CHEMBL160290 | N-hydroxy-N'-[3-methoxy-5-(5-(3,4,5...)
Affinity DataIC50:  25nMAssay Description:In vitro affinity for human PAF receptor on platelet membranes using [3H]-PAF displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50286667(CHEMBL155851 | N-hydroxy-N'-[3-methoxy-5-(5-(3,4,5...)
Affinity DataIC50:  26nMAssay Description:In vitro affinity for human PAF receptor on platelet membranes using [3H]-PAF displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50286667(CHEMBL155851 | N-hydroxy-N'-[3-methoxy-5-(5-(3,4,5...)
Affinity DataIC50:  26nMAssay Description:In vitro affinity for human PAF receptor on platelet membranes using [3H]-PAF displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50286668(CHEMBL160218 | N-hydroxy-N'-[3-methoxy-5-(5-(3,4,5...)
Affinity DataIC50:  30nMAssay Description:In vitro affinity for human PAF receptor on platelet membranes using [3H]-PAF displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50286668(CHEMBL160218 | N-hydroxy-N'-[3-methoxy-5-(5-(3,4,5...)
Affinity DataIC50:  30nMAssay Description:In vitro affinity for human PAF receptor on platelet membranes using [3H]-PAF displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50408422(CHEMBL2113721)
Affinity DataIC50:  33nMAssay Description:Inhibition of 5-lipoxygenase mediated conversion of [14C]-arachidonic acid to leukotrienes in RBL-2H3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50064506(1-Butyl-3-{3-methoxy-2-propoxy-5-[5-(3,4,5-trimeth...)
Affinity DataIC50:  33nMAssay Description:In vitro inhibition of 5-lipoxygenase in RBL-2H3 (Rat basophilic leukaemia) cells.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50064506(1-Butyl-3-{3-methoxy-2-propoxy-5-[5-(3,4,5-trimeth...)
Affinity DataIC50:  33nMAssay Description:In vitro affinity for human PAF receptor on platelet membranes using [3H]-PAF displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50064506(1-Butyl-3-{3-methoxy-2-propoxy-5-[5-(3,4,5-trimeth...)
Affinity DataIC50:  33nMAssay Description:Displacement of [3H]-PAF from PAF receptor of human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50408423(CHEMBL2113726)
Affinity DataIC50:  38nMAssay Description:Displacement of [3H]-PAF from PAF receptor of human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50408415(CHEMBL2113730)
Affinity DataIC50:  39nMAssay Description:Displacement of [3H]-PAF from PAF receptor of human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50408418(CHEMBL2113722)
Affinity DataIC50:  43nMAssay Description:Inhibition of 5-lipoxygenase mediated conversion of [14C]-arachidonic acid to leukotrienes in RBL-2H3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50408417(CHEMBL2113724)
Affinity DataIC50:  45nMAssay Description:Displacement of [3H]-PAF from PAF receptor of human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50286658(5-lipoxygenase inhibitor | CHEMBL155760)
Affinity DataIC50:  56nMAssay Description:In vitro affinity for human PAF receptor on platelet membranes using [3H]-PAF displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50408413(CHEMBL2113727)
Affinity DataIC50:  58nMAssay Description:5-lipoxygenase inhibitory activity determined by measuring the conversion of [14C]-arachidonic acid to leukotrienes in RBL-2H3 cell using thin-layer ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50286660(5-lipoxygenase inhibitor | CHEMBL160839)
Affinity DataIC50:  59nMAssay Description:In vitro affinity for human PAF receptor on platelet membranes using [3H]-PAF displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50286659(5-lipoxygenase inhibitor | CHEMBL434090)
Affinity DataIC50:  68nMAssay Description:In vitro affinity for human PAF receptor on platelet membranes using [3H]-PAF displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50405462(CHEMBL2115332)
Affinity DataIC50:  70nMAssay Description:Inhibitor concentration required to block 50 of the specific [3H]PAF binding to rabbit platelet membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50408415(CHEMBL2113730)
Affinity DataIC50:  71nMAssay Description:Inhibition of 5-lipoxygenase mediated conversion of [14C]-arachidonic acid to leukotrienes in RBL-2H3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
Beijing Institute Of Pharmacology & Toxicology

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  83nMAssay Description:Inhibition of MERTK (unknown origin) using EFPIYDFLPAKKK-CONH2 as substrate and ATP after 180 mins by microfluidic capillary electrophoresis methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50286656(5-lipoxygenase inhibitor | CHEMBL160571)
Affinity DataIC50:  91nMAssay Description:In vitro affinity for human PAF receptor on platelet membranes using [3H]-PAF displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50000714(3-[4-(2-Chloro-phenyl)-9-methyl-6H-1-thia-5,7,8,9a...)
Affinity DataIC50:  94nMAssay Description:Displacement of [3H]-PAF from PAF receptor of human platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
University Of Virginia

Curated by ChEMBL
LigandPNGBDBM50408414(CHEMBL2113720)
Affinity DataIC50:  100nMAssay Description:Inhibition of 5-lipoxygenase mediated conversion of [14C]-arachidonic acid to leukotrienes in RBL-2H3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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