Affinity DataKi: 1.40nMAssay Description:Inhibition of human full-length recombinant PARP-1More data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Inhibition of PARP-1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Henan University
Curated by ChEMBL
Henan University
Curated by ChEMBL
Affinity DataKi: 386nMAssay Description:Mixed-type inhibition of electric eel AChE using acetylthiocholine chloride as substrate incubated for 15 mins prior to substrate addition by Linewea...More data for this Ligand-Target Pair
Affinity DataIC50: 0.110nMAssay Description:Inhibition of PARP-2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 0.570nMAssay Description:Inhibition of human recombinant PARP-1 (662 to 1011 residues)More data for this Ligand-Target Pair
Affinity DataIC50: 0.830nMAssay Description:Inhibition of PARP-1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of human recombinant PARP-1More data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Inhibition of mouse recombinant PARP-2More data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:Inhibition of human PARP-2 using histone as substrate incubated for 16 hrs by ELISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:Inhibition of human PARP-1 using histone as substrate incubated for 16 hrs by ELISA assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 4.20nMAssay Description:Displacement of 5-FITC labelled (+)-JQ1 from His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3) )-codon plus-RIL cells incu...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 4.20nMAssay Description:Displacement of 5-FITC labelled (+)-JQ1 from His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3) )-codon plus-RIL cells incu...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 4.5nMAssay Description:Displacement of 5-FITC labelled (+)-JQ1 from His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3) )-codon plus-RIL cells incu...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 4.5nMAssay Description:Displacement of 5-FITC labelled (+)-JQ1 from His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3) )-codon plus-RIL cells incu...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 4.60nMAssay Description:Displacement of 5-FITC labelled (+)-JQ1 from His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3) )-codon plus-RIL cells incu...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 4.60nMAssay Description:Displacement of 5-FITC labelled (+)-JQ1 from His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3) )-codon plus-RIL cells incu...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 4.60nMAssay Description:Displacement of 5-FITC labelled (+)-JQ1 from His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3) )-codon plus-RIL cells incu...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 4.60nMAssay Description:Displacement of 5-FITC labelled (+)-JQ1 from His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3) )-codon plus-RIL cells incu...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 4.80nMAssay Description:Displacement of 5-FITC labelled (+)-JQ1 from His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3) )-codon plus-RIL cells incu...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 4.80nMAssay Description:Displacement of 5-FITC labelled (+)-JQ1 from His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3) )-codon plus-RIL cells incu...More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of PARP-1 (unknown origin)More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 5.20nMAssay Description:Displacement of 5-FITC labelled (+)-JQ1 from His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3) )-codon plus-RIL cells incu...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 5.20nMAssay Description:Displacement of 5-FITC labelled (+)-JQ1 from His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3) )-codon plus-RIL cells incu...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 5.30nMAssay Description:Displacement of 5-FITC labelled (+)-JQ1 from His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3) )-codon plus-RIL cells incu...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 5.30nMAssay Description:Displacement of 5-FITC labelled (+)-JQ1 from His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3) )-codon plus-RIL cells incu...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 5.40nMAssay Description:Displacement of 5-FITC labelled (+)-JQ1 from His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3) )-codon plus-RIL cells incu...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 5.40nMAssay Description:Displacement of 5-FITC labelled (+)-JQ1 from His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3) )-codon plus-RIL cells incu...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 5.70nMAssay Description:Displacement of 5-FITC labelled (+)-JQ1 from His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3) )-codon plus-RIL cells incu...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 5.70nMAssay Description:Displacement of 5-FITC labelled (+)-JQ1 from His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3) )-codon plus-RIL cells incu...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 5.80nMAssay Description:Displacement of 5-FITC labelled (+)-JQ1 from His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3) )-codon plus-RIL cells incu...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 5.80nMAssay Description:Displacement of 5-FITC labelled (+)-JQ1 from His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3) )-codon plus-RIL cells incu...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 5.90nMAssay Description:Displacement of 5-FITC labelled (+)-JQ1 from His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3) )-codon plus-RIL cells incu...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 5.90nMAssay Description:Displacement of 5-FITC labelled (+)-JQ1 from His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3) )-codon plus-RIL cells incu...More data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of PARP-2 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 6.10nMAssay Description:Displacement of 5-FITC labelled (+)-JQ1 from His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3) )-codon plus-RIL cells incu...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 6.10nMAssay Description:Displacement of 5-FITC labelled (+)-JQ1 from His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3) )-codon plus-RIL cells incu...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 6.60nMAssay Description:Displacement of 5-FITC labelled (+)-JQ1 from His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3) )-codon plus-RIL cells incu...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 6.60nMAssay Description:Displacement of 5-FITC labelled (+)-JQ1 from His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3) )-codon plus-RIL cells incu...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 6.80nMAssay Description:Displacement of 5-FITC labelled (+)-JQ1 from His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3) )-codon plus-RIL cells incu...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 6.80nMAssay Description:Displacement of 5-FITC labelled (+)-JQ1 from His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3) )-codon plus-RIL cells incu...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Displacement of 5-FITC labelled (+)-JQ1 from His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3) )-codon plus-RIL cells incu...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Displacement of 5-FITC labelled (+)-JQ1 from His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3) )-codon plus-RIL cells incu...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 7.10nMAssay Description:Displacement of 5-FITC labelled (+)-JQ1 from His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3) )-codon plus-RIL cells incu...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 7.10nMAssay Description:Displacement of 5-FITC labelled (+)-JQ1 from His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3) )-codon plus-RIL cells incu...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 7.90nMAssay Description:Displacement of 5-FITC labelled (+)-JQ1 from His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3) )-codon plus-RIL cells incu...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 7.90nMAssay Description:Displacement of 5-FITC labelled (+)-JQ1 from His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3) )-codon plus-RIL cells incu...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 8.60nMAssay Description:Displacement of 5-FITC labelled (+)-JQ1 from His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3) )-codon plus-RIL cells incu...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 8.60nMAssay Description:Displacement of 5-FITC labelled (+)-JQ1 from His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3) )-codon plus-RIL cells incu...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 8.70nMAssay Description:Displacement of 5-FITC labelled (+)-JQ1 from His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3) )-codon plus-RIL cells incu...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
University Of Chinese Academy Of Sciences
Curated by ChEMBL
University Of Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 8.70nMAssay Description:Displacement of 5-FITC labelled (+)-JQ1 from His6-tagged human BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3) )-codon plus-RIL cells incu...More data for this Ligand-Target Pair