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Found 163 with Last Name = 'wang' and Initial = 'ys'
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50163700((S)-2-[(S)-2-(15-{(S)-1-[(R)-1-(1-Carbamoyl-2-hydr...)
Affinity DataKi:  102nMAssay Description:Inhibitory concentration against human immunodeficiency virus -1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50163699((S)-2-[(S)-2-(15-{(S)-1-[(R)-1-(1-Carbamoyl-2-hydr...)
Affinity DataKi:  103nMAssay Description:Inhibitory concentration against human immunodeficiency virus -1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50163688((S)-2-[(S)-2-(15-{(S)-1-[(R)-1-(1-Carbamoyl-2-hydr...)
Affinity DataKi:  106nMAssay Description:Inhibitory concentration against human immunodeficiency virus -1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50163711((S)-2-[(R)-2-(4-Benzyloxy-phenyl)-2-(15-{(S)-1-[(R...)
Affinity DataKi:  110nMAssay Description:Inhibitory concentration against human immunodeficiency virus -1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50370636(CHEMBL1791327)
Affinity DataKi:  112nMAssay Description:Inhibitory concentration against human immunodeficiency virus -1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50370640(CHEMBL1791339)
Affinity DataKi:  127nMAssay Description:Inhibitory concentration against human immunodeficiency virus -1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50370653(CHEMBL1791328)
Affinity DataKi:  140nMAssay Description:Inhibitory concentration against human immunodeficiency virus -1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50370638(CHEMBL1791330)
Affinity DataKi:  160nMAssay Description:Inhibitory concentration against human immunodeficiency virus -1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50370648(CHEMBL1791340)
Affinity DataKi:  164nMAssay Description:Inhibitory concentration against human immunodeficiency virus -1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50370650(CHEMBL1791331)
Affinity DataKi:  202nMAssay Description:Inhibitory concentration against human immunodeficiency virus -1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50370413(CHEMBL1791290)
Affinity DataKi:  220nMAssay Description:Binding activity towards Human immunodeficiency virus-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50370413(CHEMBL1791290)
Affinity DataKi:  220nMAssay Description:Inhibitory concentration against human immunodeficiency virus-1 protease; (Dimerization inhibitor)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50163694((S)-3-(4-Benzoyl-phenyl)-2-((S)-3-carbamoyl-2-{15-...)
Affinity DataKi:  223nMAssay Description:Inhibitory concentration against human immunodeficiency virus -1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50163710(((S)-3-Carbamoyl-2-{15-[(S)-1-((R)-1-carbamoyl-2-p...)
Affinity DataKi:  254nMAssay Description:Inhibitory concentration against human immunodeficiency virus -1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50163717(2-((S)-3-Carbamoyl-2-{15-[(S)-1-((R)-1-carbamoyl-2...)
Affinity DataKi:  267nMAssay Description:Inhibitory concentration against human immunodeficiency virus -1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50163696((S)-2-((S)-3-Carbamoyl-2-{15-[(S)-1-((R)-1-carbamo...)
Affinity DataKi:  268nMAssay Description:Inhibitory concentration against human immunodeficiency virus -1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50370643(CHEMBL1791333)
Affinity DataKi:  273nMAssay Description:Inhibitory concentration against human immunodeficiency virus -1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50163707(2-((S)-3-Carbamoyl-2-{15-[(S)-1-((R)-1-carbamoyl-2...)
Affinity DataKi:  285nMAssay Description:Inhibitory concentration against human immunodeficiency virus -1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50370654(CHEMBL1791341)
Affinity DataKi:  314nMAssay Description:Inhibitory concentration against human immunodeficiency virus -1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50370645(CHEMBL1791342)
Affinity DataKi:  361nMAssay Description:Inhibitory concentration against human immunodeficiency virus -1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50163692((S)-2-((S)-3-Carbamoyl-2-{15-[(S)-1-((R)-1-carbamo...)
Affinity DataKi:  384nMAssay Description:Inhibitory concentration against human immunodeficiency virus -1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50370641(CHEMBL1791318)
Affinity DataKi:  414nMAssay Description:Inhibitory concentration against human immunodeficiency virus -1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin D(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50300228((2E,5R)-5-(2-cyclohexylethyl)-5-(cyclohexylmethyl)...)
Affinity DataKi:  740nMAssay Description:Inhibition of human cathepsin D preincubated for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50145828(2-(4-{3-[(S)-1-Carboxy-2-(4-hydroxy-3,5-diiodo-phe...)
Affinity DataKi:  800nMAssay Description:Inhibition constant for HCV NS3 protease substrate binding siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50145844(2-(4-{3-[(S)-1-tert-Butoxycarbonyl-2-(4-hydroxy-3,...)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition constant for HCV NS3 protease substrate binding siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50370412(CHEMBL449777)
Affinity DataKi:  3.00E+3nMAssay Description:Binding activity towards Human immunodeficiency virus-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50163697((S)-2-[(R)-3-Carbamoyl-3-(15-{(S)-1-[(S)-1-((S)-1-...)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibitory concentration against human immunodeficiency virus -1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50150552((E)-3-{(S)-1-[((S)-Carbamoyl-{11-[(S)-1-((S)-1-car...)
Affinity DataKi:  4.90E+3nMAssay Description:Binding activity towards Human immunodeficiency virus-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50145820(3-(4-Hydroxy-3,5-diiodo-phenyl)-propionic acid | C...)
Affinity DataKi:  8.00E+4nMAssay Description:Inhibition constant for HCV NS3 protease substrate binding siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50145823(3-(4-Hydroxy-3,5-diiodo-phenyl)-3-phenyl-propionic...)
Affinity DataKi:  1.00E+5nMAssay Description:Inhibition constant for HCV NS3 protease substrate binding siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50370639(CHEMBL1791329)
Affinity DataKi:  1.40E+5nMAssay Description:Inhibitory concentration against human immunodeficiency virus -1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50145804(3-(4-Hydroxy-3,5-diiodo-phenyl)-2-phenyl-propionic...)
Affinity DataKi:  1.40E+5nMAssay Description:Inhibition constant for HCV NS3 protease substrate binding siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50145815(4-(4-Hydroxy-3,5-diiodo-phenyl)-butyric acid | CHE...)
Affinity DataKi:  1.80E+5nMAssay Description:Inhibition constant for HCV NS3 protease substrate binding siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50150540((E)-3-{(S)-1-[(S)-1-{11-[(S)-1-((S)-1-Carbamoyl-2-...)
Affinity DataKi:  1.99E+5nMAssay Description:Binding activity towards Human immunodeficiency virus-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50150542((E)-3-{(S)-1-[(S)-1-{11-[(S)-1-((S)-1-Carbamoyl-2-...)
Affinity DataKi:  2.09E+5nMAssay Description:Binding activity towards Human immunodeficiency virus-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50145808((R)-2-Acetylamino-3-(4-hydroxy-3,5-diiodo-phenyl)-...)
Affinity DataKi:  2.10E+5nMAssay Description:Inhibition constant for HCV NS3 protease substrate binding siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50163691((S)-2-[(R)-3-Carbamoyl-3-(15-{(S)-1-[(R)-1-((S)-1-...)
Affinity DataKi:  2.10E+5nMAssay Description:Inhibitory concentration against human immunodeficiency virus -1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50150541((E)-3-{(S)-1-[(S)-1-(11-{(S)-1-[(S)-1-Carbamoyl-2-...)
Affinity DataKi:  2.22E+5nMAssay Description:Binding activity towards Human immunodeficiency virus-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50370646(CHEMBL1791332)
Affinity DataKi:  2.35E+5nMAssay Description:Inhibitory concentration against human immunodeficiency virus -1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50145825((R)-2-tert-Butoxycarbonylamino-3-(4-hydroxy-3,5-di...)
Affinity DataKi:  2.60E+5nMAssay Description:Inhibition constant for HCV NS3 protease substrate binding siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50145833((S)-2-tert-Butoxycarbonylamino-3-(4-hydroxy-3,5-di...)
Affinity DataKi:  3.10E+5nMAssay Description:Inhibition constant for HCV NS3 protease substrate binding siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50163701((S)-2-[(R)-3-Carbamoyl-3-(15-{1-[(R)-1-((S)-1-carb...)
Affinity DataKi:  5.02E+5nMAssay Description:Inhibitory concentration against human immunodeficiency virus -1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50145835(4-Hydroxy-3,5-diiodo-benzoic acid | CHEMBL83650)
Affinity DataKi:  6.00E+5nMAssay Description:Inhibition constant for HCV NS3 protease substrate binding siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50145827(CHEMBL311209 | N-[(4-methylbenzene)sulfonamido]ben...)
Affinity DataKi:  6.50E+5nMAssay Description:Inhibition constant for HCV NS3 protease substrate binding siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50163691((S)-2-[(R)-3-Carbamoyl-3-(15-{(S)-1-[(R)-1-((S)-1-...)
Affinity DataIC50:  1.10nMAssay Description:Inhibitory concentration against human immunodeficiency virus-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50163719((S)-2-{3-(4-Amino-phenyl)-2-[15-({(S)-1-[(R)-1-(1-...)
Affinity DataIC50:  1.20nMAssay Description:Inhibitory concentration against human immunodeficiency virus-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50163697((S)-2-[(R)-3-Carbamoyl-3-(15-{(S)-1-[(S)-1-((S)-1-...)
Affinity DataIC50:  5.40nMAssay Description:Inhibitory concentration against human immunodeficiency virus-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50322823((S)-N-(4-(3-chloro-4-fluorophenylamino)-7-(tetrahy...)
Affinity DataIC50:  15nMAssay Description:Inhibition of C-terminal His-tagged N-terminal GST-tagged human EGFR (668 to 1210 residues) expressed in baculovirus infected Sf9 cells after 30 mins...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Yunnan University

Curated by ChEMBL
LigandPNGBDBM15579(CHEMBL972 | DEPRENYL | L-Deprenyl | N-methyl-N-[(2...)
Affinity DataIC50:  20nMAssay Description:Inhibition of human recombinant MAOB assessed as reduction in H2O2 production from p-tyramine incubated for 15 mins by Amplex red reagent based fluor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Nanjing University

Curated by ChEMBL
LigandPNGBDBM50529211(CHEMBL4452957)
Affinity DataIC50:  23nMAssay Description:Inhibition of C-terminal His-tagged N-terminal GST-tagged human EGFR (668 to 1210 residues) expressed in baculovirus infected Sf9 cells after 30 mins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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