TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 102nMAssay Description:Inhibitory concentration against human immunodeficiency virus -1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 103nMAssay Description:Inhibitory concentration against human immunodeficiency virus -1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 106nMAssay Description:Inhibitory concentration against human immunodeficiency virus -1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 110nMAssay Description:Inhibitory concentration against human immunodeficiency virus -1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 112nMAssay Description:Inhibitory concentration against human immunodeficiency virus -1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 127nMAssay Description:Inhibitory concentration against human immunodeficiency virus -1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 140nMAssay Description:Inhibitory concentration against human immunodeficiency virus -1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 160nMAssay Description:Inhibitory concentration against human immunodeficiency virus -1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 164nMAssay Description:Inhibitory concentration against human immunodeficiency virus -1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 202nMAssay Description:Inhibitory concentration against human immunodeficiency virus -1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 220nMAssay Description:Binding activity towards Human immunodeficiency virus-1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 220nMAssay Description:Inhibitory concentration against human immunodeficiency virus-1 protease; (Dimerization inhibitor)More data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 223nMAssay Description:Inhibitory concentration against human immunodeficiency virus -1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 254nMAssay Description:Inhibitory concentration against human immunodeficiency virus -1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 267nMAssay Description:Inhibitory concentration against human immunodeficiency virus -1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 268nMAssay Description:Inhibitory concentration against human immunodeficiency virus -1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 273nMAssay Description:Inhibitory concentration against human immunodeficiency virus -1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 285nMAssay Description:Inhibitory concentration against human immunodeficiency virus -1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 314nMAssay Description:Inhibitory concentration against human immunodeficiency virus -1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 361nMAssay Description:Inhibitory concentration against human immunodeficiency virus -1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 384nMAssay Description:Inhibitory concentration against human immunodeficiency virus -1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 414nMAssay Description:Inhibitory concentration against human immunodeficiency virus -1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 740nMAssay Description:Inhibition of human cathepsin D preincubated for 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 800nMAssay Description:Inhibition constant for HCV NS3 protease substrate binding siteMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:Inhibition constant for HCV NS3 protease substrate binding siteMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 3.00E+3nMAssay Description:Binding activity towards Human immunodeficiency virus-1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 3.00E+3nMAssay Description:Inhibitory concentration against human immunodeficiency virus -1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 4.90E+3nMAssay Description:Binding activity towards Human immunodeficiency virus-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 8.00E+4nMAssay Description:Inhibition constant for HCV NS3 protease substrate binding siteMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+5nMAssay Description:Inhibition constant for HCV NS3 protease substrate binding siteMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 1.40E+5nMAssay Description:Inhibitory concentration against human immunodeficiency virus -1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 1.40E+5nMAssay Description:Inhibition constant for HCV NS3 protease substrate binding siteMore data for this Ligand-Target Pair
Affinity DataKi: 1.80E+5nMAssay Description:Inhibition constant for HCV NS3 protease substrate binding siteMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 1.99E+5nMAssay Description:Binding activity towards Human immunodeficiency virus-1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 2.09E+5nMAssay Description:Binding activity towards Human immunodeficiency virus-1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 2.10E+5nMAssay Description:Inhibition constant for HCV NS3 protease substrate binding siteMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 2.10E+5nMAssay Description:Inhibitory concentration against human immunodeficiency virus -1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 2.22E+5nMAssay Description:Binding activity towards Human immunodeficiency virus-1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 2.35E+5nMAssay Description:Inhibitory concentration against human immunodeficiency virus -1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 2.60E+5nMAssay Description:Inhibition constant for HCV NS3 protease substrate binding siteMore data for this Ligand-Target Pair
Affinity DataKi: 3.10E+5nMAssay Description:Inhibition constant for HCV NS3 protease substrate binding siteMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataKi: 5.02E+5nMAssay Description:Inhibitory concentration against human immunodeficiency virus -1 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 6.00E+5nMAssay Description:Inhibition constant for HCV NS3 protease substrate binding siteMore data for this Ligand-Target Pair
Affinity DataKi: 6.50E+5nMAssay Description:Inhibition constant for HCV NS3 protease substrate binding siteMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataIC50: 1.10nMAssay Description:Inhibitory concentration against human immunodeficiency virus-1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataIC50: 1.20nMAssay Description:Inhibitory concentration against human immunodeficiency virus-1 proteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataIC50: 5.40nMAssay Description:Inhibitory concentration against human immunodeficiency virus-1 proteaseMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Inhibition of C-terminal His-tagged N-terminal GST-tagged human EGFR (668 to 1210 residues) expressed in baculovirus infected Sf9 cells after 30 mins...More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of human recombinant MAOB assessed as reduction in H2O2 production from p-tyramine incubated for 15 mins by Amplex red reagent based fluor...More data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Inhibition of C-terminal His-tagged N-terminal GST-tagged human EGFR (668 to 1210 residues) expressed in baculovirus infected Sf9 cells after 30 mins...More data for this Ligand-Target Pair