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Found 56 with Last Name = 'wannamaker' and Initial = 'm'
TargetLanosterol synthase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50003025(1-((4aS,5S,6S,8aS)-6-Hydroxy-5,8a-dimethyl-octahyd...)
Affinity DataKi:  28nMAssay Description:Inhibitory concentration of the compound against purified rat liver Oxidosqualene cyclase (OSC)More data for this Ligand-Target Pair
In DepthDetails Article
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050712(CHEMBL3318007)
Affinity DataKi:  1.60E+3nMAssay Description:Inhibition of GSK3beta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50003025(1-((4aS,5S,6S,8aS)-6-Hydroxy-5,8a-dimethyl-octahyd...)
Affinity DataIC50:  100nMAssay Description:Inhibitory concentration against purified rat liver Oxidosqualene cyclase (OSC)More data for this Ligand-Target Pair
In DepthDetails Article
TargetLanosterol synthase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50003025(1-((4aS,5S,6S,8aS)-6-Hydroxy-5,8a-dimethyl-octahyd...)
Affinity DataIC50:  110nMAssay Description:Inhibitory activity against Oxidosqualene-lanosterol cyclase enzyme obtained from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50003026(1-(6-Hydroxy-5,8a-dimethyl-octahydro-isoquinolin-2...)
Affinity DataIC50:  210nMAssay Description:Inhibitory activity against Oxidosqualene-lanosterol cyclase enzyme obtained from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50281884(2-(1-Dodecyl-piperidin-4-yl)-propan-1-ol | CHEMBL1...)
Affinity DataIC50:  420nMAssay Description:Inhibitory concentration against purified rat liver Oxidosqualene cyclase (OSC)More data for this Ligand-Target Pair
In DepthDetails Article
TargetLanosterol synthase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50003032((4aS,5S,6S,8aS)-2-Dodecyl-5,8a-dimethyl-decahydro-...)
Affinity DataIC50:  550nMAssay Description:Inhibitory concentration against purified rat liver Oxidosqualene cyclase (OSC)More data for this Ligand-Target Pair
In DepthDetails Article
TargetLanosterol synthase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50003032((4aS,5S,6S,8aS)-2-Dodecyl-5,8a-dimethyl-decahydro-...)
Affinity DataIC50:  550nMAssay Description:Inhibitory activity against Oxidosqualene-lanosterol cyclase enzyme obtained from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50281889(1-(1,5,9-Trimethyl-decyl)-piperidine | CHEMBL41817...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibitory concentration against purified rat liver Oxidosqualene cyclase (OSC)More data for this Ligand-Target Pair
In DepthDetails Article
TargetLanosterol synthase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50281895(1-(1,5,9-Trimethyl-decyl)-piperidin-4-ol | CHEMBL1...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibitory concentration against purified rat liver Oxidosqualene cyclase (OSC)More data for this Ligand-Target Pair
In DepthDetails Article
TargetLanosterol synthase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50281888(2-[1-(1,5,9-Trimethyl-decyl)-piperidin-4-yl]-propa...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibitory concentration against purified rat liver Oxidosqualene cyclase (OSC)More data for this Ligand-Target Pair
In DepthDetails Article
TargetLanosterol synthase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50003027((4aS,5S,6S,8aS)-5,8a-Dimethyl-2-(1,5,9-trimethyl-d...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibitory activity against Oxidosqualene-lanosterol cyclase enzyme obtained from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50003027((4aS,5S,6S,8aS)-5,8a-Dimethyl-2-(1,5,9-trimethyl-d...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibitory concentration against purified rat liver Oxidosqualene cyclase (OSC)More data for this Ligand-Target Pair
In DepthDetails Article
TargetLanosterol synthase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50281893((4aS,5S,6S,8aS)-5,8a-Dimethyl-2-((E)-1,5,9-trimeth...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibitory concentration against purified rat liver Oxidosqualene cyclase (OSC)More data for this Ligand-Target Pair
In DepthDetails Article
TargetLanosterol synthase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50281886(1-(1,5,9-Trimethyl-decyl)-piperidin-3-ol | CHEMBL1...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibitory concentration against purified rat liver Oxidosqualene cyclase (OSC)More data for this Ligand-Target Pair
In DepthDetails Article
TargetLanosterol synthase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50281885(1-Dodecyl-piperidin-3-ol | CHEMBL17348)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibitory concentration against purified rat liver Oxidosqualene cyclase (OSC)More data for this Ligand-Target Pair
In DepthDetails Article
TargetLanosterol synthase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50003030((2S,4aS,8aR)-1,1,4a-Trimethyl-decahydro-naphthalen...)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibitory activity against Oxidosqualene-lanosterol cyclase enzyme obtained from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50281891(1-Dodecyl-piperidin-4-ol | CHEMBL17729)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibitory concentration against purified rat liver Oxidosqualene cyclase (OSC)More data for this Ligand-Target Pair
In DepthDetails Article
TargetLanosterol synthase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50281887(1-((E)-1,5,9-Trimethyl-deca-4,8-dienyl)-piperidin-...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory concentration against purified rat liver Oxidosqualene cyclase (OSC)More data for this Ligand-Target Pair
In DepthDetails Article
TargetLanosterol synthase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50281890(1-[4-(2-Hydroxy-1-methyl-ethyl)-piperidin-1-yl]-tr...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory concentration against purified rat liver Oxidosqualene cyclase (OSC)More data for this Ligand-Target Pair
In DepthDetails Article
TargetLanosterol synthase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50003028(2-(Dodecane-1-sulfinyl)-5,8a-dimethyl-decahydro-is...)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibitory activity against Oxidosqualene-lanosterol cyclase enzyme obtained from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50281896(1-((E)-1,5,9-Trimethyl-deca-4,8-dienyl)-piperidin-...)
Affinity DataIC50:  4.00E+4nMAssay Description:Inhibitory concentration against purified rat liver Oxidosqualene cyclase (OSC)More data for this Ligand-Target Pair
In DepthDetails Article
TargetLanosterol synthase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50281892(1-((E)-1,5,9-Trimethyl-deca-4,8-dienyl)-piperidine...)
Affinity DataIC50:  4.00E+4nMAssay Description:Inhibitory concentration against purified rat liver Oxidosqualene cyclase (OSC)More data for this Ligand-Target Pair
In DepthDetails Article
TargetLanosterol synthase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50003031(1-(6-Hydroxy-5,8a-dimethyl-octahydro-isoquinolin-2...)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibitory activity against Oxidosqualene-lanosterol cyclase enzyme obtained from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50281894(2-(1-Benzyl-piperidin-4-yl)-propan-1-ol | CHEMBL28...)
Affinity DataIC50:  5.70E+4nMAssay Description:Inhibitory concentration against purified rat liver Oxidosqualene cyclase (OSC)More data for this Ligand-Target Pair
In DepthDetails Article
TargetLanosterol synthase(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50003029(2-(Dodecane-1-sulfonyl)-5,8a-dimethyl-decahydro-is...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against Oxidosqualene-lanosterol cyclase enzyme obtained from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050716(CHEMBL3317990)
Affinity DataKd:  20nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050717(CHEMBL3317991)
Affinity DataKd:  90nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050718(CHEMBL3317969)
Affinity DataKd:  100nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050719(CHEMBL3317970)
Affinity DataKd:  300nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050720(CHEMBL3317972)
Affinity DataKd:  700nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050721(CHEMBL3317973)
Affinity DataKd:  300nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050722(CHEMBL3317974)
Affinity DataKd:  100nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050750(CHEMBL3317975)
Affinity DataKd:  100nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050754(CHEMBL3317976)
Affinity DataKd:  400nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050756(CHEMBL3317977)
Affinity DataKd:  80nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050757(CHEMBL3317978)
Affinity DataKd:  90nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050758(CHEMBL3317979)
Affinity DataKd:  4.90E+3nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050759(CHEMBL3317980)
Affinity DataKd:  100nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050760(CHEMBL3317981)
Affinity DataKd:  70nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050708(CHEMBL3318004)
Affinity DataKd: <2nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050707(CHEMBL3318003)
Affinity DataKd:  9nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050706(CHEMBL3318002)
Affinity DataKd: <2nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050705(CHEMBL3318001)
Affinity DataKd: <2nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050703(CHEMBL3318000)
Affinity DataKd: <2nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050702(CHEMBL3317999)
Affinity DataKd:  30nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050701(CHEMBL3317986)
Affinity DataKd:  400nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050700(CHEMBL3317985)
Affinity DataKd:  200nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050699(CHEMBL3317984)
Affinity DataKd:  400nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolymerase basic protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Vertex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50050698(CHEMBL3317983)
Affinity DataKd:  200nMAssay Description:Binding affinity to influenza A virus (A/Puerto Rico/8/1934(H1N1)) PB2 by competition binding fluorescence polarization (FP) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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