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Found 93 with Last Name = 'watkins' and Initial = 'eb'
TargetNADPH oxidase 4(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50455025(CHEMBL4208156)
Affinity DataIC50:  500nMAssay Description:Inhibition of Nox4 in HASMCs assessed as reduction in TGFbeta-induced increase in smooth muscle alpha actin level pretreated for 30 mins followed by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNADPH oxidase 4(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50455023(CHEMBL4204145)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of Nox4 in HASMCs assessed as reduction in TGFbeta-induced increase in smooth muscle alpha actin level pretreated for 30 mins followed by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase(Plasmodium falciparum)
University of Mississippi

LigandPNGBDBM23223(7-[8-formyl-1,6,7-trihydroxy-3-methyl-5-(propan-2-...)
Affinity DataIC50:  3.97E+3nMAssay Description:Enzyme assay using recombinant pfLDH and mLDH (bovine heart).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine proteinase falcipain 2a(Plasmodium falciparum)
University, Mississippi

LigandPNGBDBM93124(Trisubsituted thiazole, 14)
Affinity DataIC50:  6.60E+3nMAssay Description:In vitro antimalarial assay, antimalarial activity of the compounds was determined in vitro on chloroquine sensitive and resistant strains of plasmod...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetL-lactate dehydrogenase(Bos taurus (Bovine))
University of Mississippi

LigandPNGBDBM23223(7-[8-formyl-1,6,7-trihydroxy-3-methyl-5-(propan-2-...)
Affinity DataIC50:  6.90E+3nMAssay Description:Enzyme assay using recombinant pfLDH and mLDH (bovine heart).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine proteinase falcipain 2a(Plasmodium falciparum)
University, Mississippi

LigandPNGBDBM93130(Trisubsituted thiazole, 29)
Affinity DataIC50: >1.25E+4nMAssay Description:In vitro antimalarial assay, antimalarial activity of the compounds was determined in vitro on chloroquine sensitive and resistant strains of plasmod...More data for this Ligand-Target Pair
In DepthDetails Article
TargetCysteine proteinase falcipain 2a(Plasmodium falciparum)
University, Mississippi

LigandPNGBDBM93125(Trisubsituted thiazole, 15)
Affinity DataIC50: >1.25E+4nMAssay Description:In vitro antimalarial assay, antimalarial activity of the compounds was determined in vitro on chloroquine sensitive and resistant strains of plasmod...More data for this Ligand-Target Pair
In DepthDetails Article
TargetL-lactate dehydrogenase(Plasmodium falciparum)
University of Mississippi

LigandPNGBDBM93303(Oxamic Acid/Ester, 21)
Affinity DataIC50:  1.40E+4nMAssay Description:Enzyme assay using recombinant pfLDH and mLDH (bovine heart).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine proteinase falcipain 2a(Plasmodium falciparum)
University, Mississippi

LigandPNGBDBM93129(Trisubsituted thiazole, 23)
Affinity DataIC50:  1.53E+4nMAssay Description:In vitro antimalarial assay, antimalarial activity of the compounds was determined in vitro on chloroquine sensitive and resistant strains of plasmod...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetL-lactate dehydrogenase(Bos taurus (Bovine))
University of Mississippi

LigandPNGBDBM93300(Oxamic Acid/Ester, 18)
Affinity DataIC50:  2.00E+4nMAssay Description:Enzyme assay using recombinant pfLDH and mLDH (bovine heart).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase(Bos taurus (Bovine))
University of Mississippi

LigandPNGBDBM93303(Oxamic Acid/Ester, 21)
Affinity DataIC50:  2.50E+4nMAssay Description:Enzyme assay using recombinant pfLDH and mLDH (bovine heart).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADPH oxidase 4(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50455024(CHEMBL4205860)
Affinity DataIC50:  2.70E+4nMAssay Description:Inhibition of Nox4 in HASMCs assessed as reduction in TGFbeta-induced increase in smooth muscle alpha actin level pretreated for 30 mins followed by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University, Mississippi

LigandPNGBDBM93124(Trisubsituted thiazole, 14)
Affinity DataIC50:  2.94E+4nMAssay Description:In vitro antimalarial assay, antimalarial activity of the compounds was determined in vitro on chloroquine sensitive and resistant strains of plasmod...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetL-lactate dehydrogenase(Bos taurus (Bovine))
University of Mississippi

LigandPNGBDBM93307(Oxamic Acid/Ester, 25)
Affinity DataIC50:  3.10E+4nMAssay Description:Enzyme assay using recombinant pfLDH and mLDH (bovine heart).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase(Bos taurus (Bovine))
University of Mississippi

LigandPNGBDBM93309(Oxamic Acid/Ester, 27)
Affinity DataIC50:  3.20E+4nMAssay Description:Enzyme assay using recombinant pfLDH and mLDH (bovine heart).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine proteinase falcipain 2a(Plasmodium falciparum)
University, Mississippi

LigandPNGBDBM93128(Trisubsituted thiazole, 20)
Affinity DataIC50: >3.30E+4nMAssay Description:In vitro antimalarial assay, antimalarial activity of the compounds was determined in vitro on chloroquine sensitive and resistant strains of plasmod...More data for this Ligand-Target Pair
In DepthDetails Article
TargetCysteine proteinase falcipain 2a(Plasmodium falciparum)
University, Mississippi

LigandPNGBDBM93131(Trisubsituted thiazole, 30)
Affinity DataIC50: >3.30E+4nMAssay Description:In vitro antimalarial assay, antimalarial activity of the compounds was determined in vitro on chloroquine sensitive and resistant strains of plasmod...More data for this Ligand-Target Pair
In DepthDetails Article
TargetCysteine proteinase falcipain 2a(Plasmodium falciparum)
University, Mississippi

LigandPNGBDBM93127(Trisubsituted thiazole, 17)
Affinity DataIC50: >3.30E+4nMAssay Description:In vitro antimalarial assay, antimalarial activity of the compounds was determined in vitro on chloroquine sensitive and resistant strains of plasmod...More data for this Ligand-Target Pair
In DepthDetails Article
TargetL-lactate dehydrogenase(Plasmodium falciparum)
University of Mississippi

LigandPNGBDBM93318(Oxamic Acid/Ester, 36)
Affinity DataIC50:  3.50E+4nMAssay Description:Enzyme assay using recombinant pfLDH and mLDH (bovine heart).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCysteine proteinase falcipain 2a(Plasmodium falciparum)
University, Mississippi

LigandPNGBDBM93126(Trisubsituted thiazole, 16)
Affinity DataIC50:  3.91E+4nMAssay Description:In vitro antimalarial assay, antimalarial activity of the compounds was determined in vitro on chloroquine sensitive and resistant strains of plasmod...More data for this Ligand-Target Pair
In DepthDetails Article
TargetL-lactate dehydrogenase(Plasmodium falciparum)
University of Mississippi

LigandPNGBDBM93323(Oxamic Acid/Ester, 41)
Affinity DataIC50:  4.10E+4nMAssay Description:Enzyme assay using recombinant pfLDH and mLDH (bovine heart).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase(Plasmodium falciparum)
University of Mississippi

LigandPNGBDBM93299(Oxamic Acid/Ester, 17)
Affinity DataIC50:  4.30E+4nMAssay Description:Enzyme assay using recombinant pfLDH and mLDH (bovine heart).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase(Plasmodium falciparum)
University of Mississippi

LigandPNGBDBM93307(Oxamic Acid/Ester, 25)
Affinity DataIC50:  4.30E+4nMAssay Description:Enzyme assay using recombinant pfLDH and mLDH (bovine heart).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase(Bos taurus (Bovine))
University of Mississippi

LigandPNGBDBM93315(Oxamic Acid/Ester, 33)
Affinity DataIC50:  4.30E+4nMAssay Description:Enzyme assay using recombinant pfLDH and mLDH (bovine heart).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase(Bos taurus (Bovine))
University of Mississippi

LigandPNGBDBM93301(Oxamic Acid/Ester, 19)
Affinity DataIC50:  4.60E+4nMAssay Description:Enzyme assay using recombinant pfLDH and mLDH (bovine heart).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase(Plasmodium falciparum)
University of Mississippi

LigandPNGBDBM93305(Oxamic Acid/Ester, 23)
Affinity DataIC50:  4.70E+4nMAssay Description:Enzyme assay using recombinant pfLDH and mLDH (bovine heart).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University, Mississippi

LigandPNGBDBM93130(Trisubsituted thiazole, 29)
Affinity DataIC50: >5.00E+4nMAssay Description:In vitro antimalarial assay, antimalarial activity of the compounds was determined in vitro on chloroquine sensitive and resistant strains of plasmod...More data for this Ligand-Target Pair
In DepthDetails Article
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University, Mississippi

LigandPNGBDBM93128(Trisubsituted thiazole, 20)
Affinity DataIC50: >5.00E+4nMAssay Description:In vitro antimalarial assay, antimalarial activity of the compounds was determined in vitro on chloroquine sensitive and resistant strains of plasmod...More data for this Ligand-Target Pair
In DepthDetails Article
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University, Mississippi

LigandPNGBDBM93127(Trisubsituted thiazole, 17)
Affinity DataIC50: >5.00E+4nMAssay Description:In vitro antimalarial assay, antimalarial activity of the compounds was determined in vitro on chloroquine sensitive and resistant strains of plasmod...More data for this Ligand-Target Pair
In DepthDetails Article
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University, Mississippi

LigandPNGBDBM93126(Trisubsituted thiazole, 16)
Affinity DataIC50: >5.00E+4nMAssay Description:In vitro antimalarial assay, antimalarial activity of the compounds was determined in vitro on chloroquine sensitive and resistant strains of plasmod...More data for this Ligand-Target Pair
In DepthDetails Article
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University, Mississippi

LigandPNGBDBM93125(Trisubsituted thiazole, 15)
Affinity DataIC50: >5.00E+4nMAssay Description:In vitro antimalarial assay, antimalarial activity of the compounds was determined in vitro on chloroquine sensitive and resistant strains of plasmod...More data for this Ligand-Target Pair
In DepthDetails Article
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University, Mississippi

LigandPNGBDBM93131(Trisubsituted thiazole, 30)
Affinity DataIC50: >5.00E+4nMAssay Description:In vitro antimalarial assay, antimalarial activity of the compounds was determined in vitro on chloroquine sensitive and resistant strains of plasmod...More data for this Ligand-Target Pair
In DepthDetails Article
TargetL-lactate dehydrogenase(Plasmodium falciparum)
University of Mississippi

LigandPNGBDBM93324(Oxamic Acid/Ester, 42)
Affinity DataIC50:  5.10E+4nMAssay Description:Enzyme assay using recombinant pfLDH and mLDH (bovine heart).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCysteine proteinase falcipain 3(Plasmodium falciparum)
University, Mississippi

LigandPNGBDBM93129(Trisubsituted thiazole, 23)
Affinity DataIC50:  5.52E+4nMAssay Description:In vitro antimalarial assay, antimalarial activity of the compounds was determined in vitro on chloroquine sensitive and resistant strains of plasmod...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetL-lactate dehydrogenase(Bos taurus (Bovine))
University of Mississippi

LigandPNGBDBM93302(Oxamic Acid/Ester, 20)
Affinity DataIC50:  5.90E+4nMAssay Description:Enzyme assay using recombinant pfLDH and mLDH (bovine heart).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase(Plasmodium falciparum)
University of Mississippi

LigandPNGBDBM93300(Oxamic Acid/Ester, 18)
Affinity DataIC50:  5.90E+4nMAssay Description:Enzyme assay using recombinant pfLDH and mLDH (bovine heart).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase(Plasmodium falciparum)
University of Mississippi

LigandPNGBDBM93308(Oxamic Acid/Ester, 26)
Affinity DataIC50:  8.80E+4nMAssay Description:Enzyme assay using recombinant pfLDH and mLDH (bovine heart).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase(Bos taurus (Bovine))
University of Mississippi

LigandPNGBDBM93323(Oxamic Acid/Ester, 41)
Affinity DataIC50:  8.80E+4nMAssay Description:Enzyme assay using recombinant pfLDH and mLDH (bovine heart).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase(Bos taurus (Bovine))
University of Mississippi

LigandPNGBDBM93318(Oxamic Acid/Ester, 36)
Affinity DataIC50:  9.00E+4nMAssay Description:Enzyme assay using recombinant pfLDH and mLDH (bovine heart).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase(Plasmodium falciparum)
University of Mississippi

LigandPNGBDBM23222(Oxalamic acid | Oxamate | Oxamate, 3 | Oxamidic Ac...)
Affinity DataIC50:  9.44E+4nMAssay Description:Enzyme assay using recombinant pfLDH and mLDH (bovine heart).More data for this Ligand-Target Pair
TargetL-lactate dehydrogenase(Plasmodium falciparum)
University of Mississippi

LigandPNGBDBM93291(Oxamic Acid/Ester, 7)
Affinity DataIC50:  9.79E+4nMAssay Description:Enzyme assay using recombinant pfLDH and mLDH (bovine heart).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase(Plasmodium falciparum)
University of Mississippi

LigandPNGBDBM93302(Oxamic Acid/Ester, 20)
Affinity DataIC50:  1.01E+5nMAssay Description:Enzyme assay using recombinant pfLDH and mLDH (bovine heart).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase(Bos taurus (Bovine))
University of Mississippi

LigandPNGBDBM93291(Oxamic Acid/Ester, 7)
Affinity DataIC50:  1.07E+5nMAssay Description:Enzyme assay using recombinant pfLDH and mLDH (bovine heart).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase(Bos taurus (Bovine))
University of Mississippi

LigandPNGBDBM23222(Oxalamic acid | Oxamate | Oxamate, 3 | Oxamidic Ac...)
Affinity DataIC50:  1.16E+5nMAssay Description:Enzyme assay using recombinant pfLDH and mLDH (bovine heart).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase(Bos taurus (Bovine))
University of Mississippi

LigandPNGBDBM93305(Oxamic Acid/Ester, 23)
Affinity DataIC50:  1.33E+5nMAssay Description:Enzyme assay using recombinant pfLDH and mLDH (bovine heart).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase(Plasmodium falciparum)
University of Mississippi

LigandPNGBDBM93320(Oxamic Acid/Ester, 38)
Affinity DataIC50:  1.46E+5nMAssay Description:Enzyme assay using recombinant pfLDH and mLDH (bovine heart).More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase(Bos taurus (Bovine))
University of Mississippi

LigandPNGBDBM93296(Oxamic Acid/Ester, 14)
Affinity DataIC50:  1.50E+5nMAssay Description:Enzyme assay using recombinant pfLDH and mLDH (bovine heart).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase(Plasmodium falciparum)
University of Mississippi

LigandPNGBDBM93316(Oxamic Acid/Ester, 34)
Affinity DataIC50:  1.57E+5nMAssay Description:Enzyme assay using recombinant pfLDH and mLDH (bovine heart).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase(Bos taurus (Bovine))
University of Mississippi

LigandPNGBDBM93292(Oxamic Acid/Ester, 8)
Affinity DataIC50:  1.58E+5nMAssay Description:Enzyme assay using recombinant pfLDH and mLDH (bovine heart).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase(Plasmodium falciparum)
University of Mississippi

LigandPNGBDBM93293(Oxamic Acid/Ester, 10)
Affinity DataIC50:  1.60E+5nMAssay Description:Enzyme assay using recombinant pfLDH and mLDH (bovine heart).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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