TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataKi: 0.490nMAssay Description:Displacement of [3H]U-69593 from kappa opioid receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(GUINEA PIG)
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataKi: 0.680nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University M£Nster
Curated by ChEMBL
University M£Nster
Curated by ChEMBL
Affinity DataKi: 1.90nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University M£Nster
Curated by ChEMBL
University M£Nster
Curated by ChEMBL
Affinity DataKi: 2.20nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University M£Nster
Curated by ChEMBL
University M£Nster
Curated by ChEMBL
Affinity DataKi: 2.20nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataKi: 3.17nMAssay Description:Displacement of [3H]U-69593 from kappa opioid receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University M£Nster
Curated by ChEMBL
University M£Nster
Curated by ChEMBL
Affinity DataKi: 3.58nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University M£Nster
Curated by ChEMBL
University M£Nster
Curated by ChEMBL
Affinity DataKi: 6.5nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University M£Nster
Curated by ChEMBL
University M£Nster
Curated by ChEMBL
Affinity DataKi: 7.5nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University M£Nster
Curated by ChEMBL
University M£Nster
Curated by ChEMBL
Affinity DataKi: 13.2nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University M£Nster
Curated by ChEMBL
University M£Nster
Curated by ChEMBL
Affinity DataKi: 16.2nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University M£Nster
Curated by ChEMBL
University M£Nster
Curated by ChEMBL
Affinity DataKi: 23.4nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University M£Nster
Curated by ChEMBL
University M£Nster
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University M£Nster
Curated by ChEMBL
University M£Nster
Curated by ChEMBL
Affinity DataKi: 26nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University M£Nster
Curated by ChEMBL
University M£Nster
Curated by ChEMBL
Affinity DataKi: 29.5nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University M£Nster
Curated by ChEMBL
University M£Nster
Curated by ChEMBL
Affinity DataKi: 33.3nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University M£Nster
Curated by ChEMBL
University M£Nster
Curated by ChEMBL
Affinity DataKi: 39.5nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University M£Nster
Curated by ChEMBL
University M£Nster
Curated by ChEMBL
Affinity DataKi: 76nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University M£Nster
Curated by ChEMBL
University M£Nster
Curated by ChEMBL
Affinity DataKi: 118nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University M£Nster
Curated by ChEMBL
University M£Nster
Curated by ChEMBL
Affinity DataKi: 125nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University M£Nster
Curated by ChEMBL
University M£Nster
Curated by ChEMBL
Affinity DataKi: 126nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataKi: 157nMAssay Description:Displacement of [3H]U-69593 from kappa opioid receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University M£Nster
Curated by ChEMBL
University M£Nster
Curated by ChEMBL
Affinity DataKi: 164nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University M£Nster
Curated by ChEMBL
University M£Nster
Curated by ChEMBL
Affinity DataKi: 175nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University M£Nster
Curated by ChEMBL
University M£Nster
Curated by ChEMBL
Affinity DataKi: 177nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University M£Nster
Curated by ChEMBL
University M£Nster
Curated by ChEMBL
Affinity DataKi: 258nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataKi: 585nMAssay Description:Displacement of [3H]U-69593 from kappa opioid receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataKi: 1.11E+3nMAssay Description:Displacement of [3H]U-69593 from kappa opioid receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataKi: 1.29E+3nMAssay Description:Displacement of [3H]U-69593 from kappa opioid receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University M£Nster
Curated by ChEMBL
University M£Nster
Curated by ChEMBL
Affinity DataKi: 1.35E+3nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataKi: 1.60E+3nMAssay Description:Displacement of [3H]U-69593 from kappa opioid receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataKi: 2.23E+3nMAssay Description:Displacement of [3H]U-69593 from kappa opioid receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University M£Nster
Curated by ChEMBL
University M£Nster
Curated by ChEMBL
Affinity DataKi: 2.40E+3nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataKi: 2.46E+3nMAssay Description:Displacement of [3H]U-69593 from kappa opioid receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(GUINEA PIG)
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataKi: 3.32E+3nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University M£Nster
Curated by ChEMBL
University M£Nster
Curated by ChEMBL
Affinity DataKi: 3.50E+3nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataKi: 3.59E+3nMAssay Description:Displacement of [3H]U-69593 from kappa opioid receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(GUINEA PIG)
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataKi: 4.05E+3nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(GUINEA PIG)
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataKi: 4.96E+3nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University M£Nster
Curated by ChEMBL
University M£Nster
Curated by ChEMBL
Affinity DataKi: 4.97E+3nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataKi: 5.02E+3nMAssay Description:Displacement of [3H]U-69593 from kappa opioid receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Institut F£R Pharmazeutische Und Medizinische Chemie
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]U-69593 from kappa opioid receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Ariad Pharmaceuticals
Curated by ChEMBL
Ariad Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:In vitro inhibition of Src protein tryrosine kinase using the Scintillation proximity kinase assay.More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Ariad Pharmaceuticals
Curated by ChEMBL
Ariad Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:In vitro inhibition of Src protein tryrosine kinase using the Scintillation proximity kinase assay.More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Ariad Pharmaceuticals
Curated by ChEMBL
Ariad Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:In vitro inhibition of Src protein tryrosine kinase using the Scintillation proximity kinase assay.More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Ariad Pharmaceuticals
Curated by ChEMBL
Ariad Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:In vitro inhibition of Src protein tryrosine kinase using the Scintillation proximity kinase assay.More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Ariad Pharmaceuticals
Curated by ChEMBL
Ariad Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:In vitro inhibition of Src protein tryrosine kinase using the Scintillation proximity kinase assay.More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Ariad Pharmaceuticals
Curated by ChEMBL
Ariad Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:In vitro inhibition of Src protein tryrosine kinase using the Scintillation proximity kinase assay.More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Ariad Pharmaceuticals
Curated by ChEMBL
Ariad Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:In vitro inhibition of Src protein tryrosine kinase using the Scintillation proximity kinase assay.More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Ariad Pharmaceuticals
Curated by ChEMBL
Ariad Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:In vitro inhibition of Src protein tryrosine kinase using the Scintillation proximity kinase assay.More data for this Ligand-Target Pair