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Found 87 with Last Name = 'welton' and Initial = 'af'
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50013923(3-(1-Butyl-4-methoxy-naphthalen-2-yl)-N-(1-methyl-...)
Affinity DataIC50:  1nMAssay Description:Inhibition of [3H]-PAF binding to platelet activating factor receptor citrate-treated dog bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50013924(3-(1-Butyl-4,7-dimethoxy-naphthalen-2-yl)-N-(1-met...)
Affinity DataIC50:  3nMAssay Description:Inhibition of [3H]-PAF binding to platelet activating factor receptor citrate-treated dog bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50018341(2-Ethyl-3',4'-dimethoxy-biphenyl-4-carboxylic acid...)
Affinity DataIC50:  4nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50018316(2-Butyl-3',4'-dimethoxy-biphenyl-4-carboxylic acid...)
Affinity DataIC50:  4nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50018325(CHEMBL53584 | [1,1';2',1'']Terphenyl-4'-carboxylic...)
Affinity DataIC50:  5nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50018315(2-Ethynyl-3',4'-dimethoxy-biphenyl-4-carboxylic ac...)
Affinity DataIC50:  5nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50013921(3-(1-Butyl-5-methoxy-naphthalen-2-yl)-N-(1-methyl-...)
Affinity DataIC50:  6nMAssay Description:Inhibition of [3H]-PAF binding to platelet activating factor receptor citrate-treated dog bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50013925(3-(1-Butyl-6-methoxy-naphthalen-2-yl)-N-(1-methyl-...)
Affinity DataIC50:  7nMAssay Description:Inhibition of [3H]-PAF binding to platelet activating factor receptor citrate-treated dog bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50013922(3-(1-Butyl-7-methoxy-naphthalen-2-yl)-N-(1-methyl-...)
Affinity DataIC50:  15nMAssay Description:Inhibition of [3H]-PAF binding to platelet activating factor receptor citrate-treated dog bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50018321(3',4'-Dimethoxy-biphenyl-4-carboxylic acid (1-meth...)
Affinity DataIC50:  15nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50018338(2-Butyl-3',4'-dimethoxy-biphenyl-4-carboxylic acid...)
Affinity DataIC50:  18nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50018337(3'-Methoxy-biphenyl-4-carboxylic acid (1-methyl-4-...)
Affinity DataIC50:  20nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50019689(3-Chloro-11-oxo-11H-pyrido[2,1-b]quinazoline-8-car...)
Affinity DataIC50:  20nMAssay Description:Inhibition of human platelet thromboxane synthase (TXA2) was determined in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50019683(11-Oxo-11H-pyrido[2,1-b]quinazoline-8-carboxylic a...)
Affinity DataIC50:  20nMAssay Description:Inhibition of human platelet thromboxane synthase (TXA2) was determined in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50019678(3-Methoxy-11-oxo-11H-pyrido[2,1-b]quinazoline-8-ca...)
Affinity DataIC50:  20nMAssay Description:Inhibition of human platelet thromboxane synthase (TXA2) was determined in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50013929(3-(6-Methoxy-3-pentyl-benzo[b]thiophen-2-yl)-N-(1-...)
Affinity DataIC50:  24nMAssay Description:Inhibition of [3H]-PAF binding to platelet activating factor receptor citrate-treated dog bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50013926(CHEMBL319384 | N-(1-Ethyl-4-pyridin-3-yl-butyl)-3-...)
Affinity DataIC50:  26nMAssay Description:Inhibition of [3H]-PAF binding to platelet activating factor receptor citrate-treated dog bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50013933(3-[6-Methoxy-1-(4-methoxy-phenyl)-3,4-dihydro-naph...)
Affinity DataIC50:  30nMAssay Description:Inhibition of [3H]-PAF binding to platelet activating factor receptor citrate-treated dog bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50013930(3-(6-Methoxy-3-pentyl-1H-inden-2-yl)-N-(1-methyl-4...)
Affinity DataIC50:  33nMAssay Description:Inhibition of [3H]-PAF binding to platelet activating factor receptor citrate-treated dog bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1/2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50006812(7-[3-(4-Acetyl-3-hydroxy-2-propyl-phenoxy)-2-hydro...)
Affinity DataIC50:  35nMAssay Description:In vitro inhibition of SRS-A-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50013927(5-(4-Methoxy-phenyl)-deca-2,4-dienoic acid (1-meth...)
Affinity DataIC50:  40nMAssay Description:Inhibition of [3H]-PAF binding to platelet activating factor receptor citrate-treated dog bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50013928(3-(6-Methoxy-3-pentyl-benzofuran-2-yl)-N-(1-methyl...)
Affinity DataIC50:  40nMAssay Description:Inhibition of [3H]-PAF binding to platelet activating factor receptor citrate-treated dog bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50018320(3',4'-Dimethoxy-2-propyl-biphenyl-4-carboxylic aci...)
Affinity DataIC50:  50nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50018324(CHEMBL299760 | [1,1';2',1'']Terphenyl-4'-carboxyli...)
Affinity DataIC50:  50nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50367404(CHEMBL1202758)
Affinity DataIC50:  50nMAssay Description:Inhibition of human platelet thromboxane synthase (TXA2) was determined in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50013931(3-[6-Methoxy-1-(4-methoxy-phenyl)-naphthalen-2-yl]...)
Affinity DataIC50:  55nMAssay Description:Inhibition of [3H]-PAF binding to platelet activating factor receptor citrate-treated dog bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50018329(3',4'-Dimethoxy-biphenyl-4-carbothioic acid (1-met...)
Affinity DataIC50:  60nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50019671(2-Isopropoxy-11-oxo-11H-pyrido[2,1-b]quinazoline-8...)
Affinity DataIC50:  60nMAssay Description:Inhibition of human platelet thromboxane synthase (TXA2) was determined in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50019670(2-Hydroxy-11-oxo-11H-pyrido[2,1-b]quinazoline-8-ca...)
Affinity DataIC50:  60nMAssay Description:Inhibition of human platelet thromboxane synthase (TXA2) was determined in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50018326(2-Allyl-3',4'-dimethoxy-biphenyl-4-carboxylic acid...)
Affinity DataIC50:  80nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1/2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50225202(CHEMBL49572)
Affinity DataIC50:  80nMAssay Description:In vitro inhibition of SRS-A-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50013932(3-(1-Butyl-6-methoxy-3,4-dihydro-naphthalen-2-yl)-...)
Affinity DataIC50:  90nMAssay Description:Inhibition of [3H]-PAF binding to platelet activating factor receptor citrate-treated dog bloodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50019680(2-Isopropyl-11-oxo-11H-pyrido[2,1-b]quinazoline-8-...)
Affinity DataIC50:  100nMAssay Description:Inhibition of human platelet thromboxane synthase (TXA2) was determined in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50019668(2-Isopropyl-11-oxo-11H-pyrido[2,1-b]quinazoline-8-...)
Affinity DataIC50:  100nMAssay Description:Inhibition of human platelet thromboxane synthase (TXA2) was determined in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50019684(2-Isopropyl-11-oxo-11H-pyrido[2,1-b]quinazoline-8-...)
Affinity DataIC50:  100nMAssay Description:Inhibition of human platelet thromboxane synthase (TXA2) was determined in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50019688(2-Bromo-11-oxo-11H-pyrido[2,1-b]quinazoline-8-carb...)
Affinity DataIC50:  100nMAssay Description:Inhibition of human platelet thromboxane synthase (TXA2) was determined in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50019665(2,3-Dimethyl-11-oxo-11H-pyrido[2,1-b]quinazoline-8...)
Affinity DataIC50:  100nMAssay Description:Inhibition of human platelet thromboxane synthase (TXA2) was determined in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50019676(2-Methyl-11-oxo-11H-pyrido[2,1-b]quinazoline-8-car...)
Affinity DataIC50:  100nMAssay Description:Inhibition of human platelet thromboxane synthase (TXA2) was determined in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1/2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50225299(CHEMBL301537)
Affinity DataIC50:  100nMAssay Description:In vitro inhibition of SRS-A-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50019672(2-Isopropyl-11-oxo-11H-pyrido[2,1-b]quinazoline-8-...)
Affinity DataIC50:  100nMAssay Description:Inhibition of human platelet thromboxane synthase (TXA2) was determined in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1/2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50225201(CHEMBL51531)
Affinity DataIC50:  100nMAssay Description:In vitro inhibition of SRS-A-induced contractions in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50018322(4,4''-Dimethoxy-[1,1';2',1'']terphenyl-4'-carboxyl...)
Affinity DataIC50:  125nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50018336(3',4'-Dimethoxy-biphenyl-4-carbothioic acid (4-pyr...)
Affinity DataIC50:  140nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50018327(2-Bromo-3',4'-dimethoxy-biphenyl-4-carboxylic acid...)
Affinity DataIC50:  180nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50018319(3',4'-Dimethoxy-2-nitro-biphenyl-4-carboxylic acid...)
Affinity DataIC50:  200nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50018323(3,3''-Dimethoxy-[1,1';2',1'']terphenyl-4'-carboxyl...)
Affinity DataIC50:  200nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50018328(3',4'-Dimethyl-biphenyl-4-carboxylic acid (4-pyrid...)
Affinity DataIC50:  200nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50018331(3',4'-Dimethoxy-2-nitro-biphenyl-4-carboxylic acid...)
Affinity DataIC50:  200nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50019669(2-Isopropyl-11-oxo-11H-pyrido[2,1-b]quinazoline-8-...)
Affinity DataIC50:  200nMAssay Description:Inhibition of human platelet thromboxane synthase (TXA2) was determined in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50019673(2-Isopropyl-11-oxo-11H-pyrido[2,1-b]quinazoline-8-...)
Affinity DataIC50:  200nMAssay Description:Inhibition of human platelet thromboxane synthase (TXA2) was determined in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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