TargetSolute carrier family 22 member 6(Rattus norvegicus)
University Of Rochester School Of Medicine And Dentistry
Curated by ChEMBL
University Of Rochester School Of Medicine And Dentistry
Curated by ChEMBL
Affinity DataKi: 400nMAssay Description:TP_TRANSPORTER: inhibition of PAH uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 6(Rattus norvegicus)
University Of Rochester School Of Medicine And Dentistry
Curated by ChEMBL
University Of Rochester School Of Medicine And Dentistry
Curated by ChEMBL
Affinity DataKi: 1.10E+3nMAssay Description:TP_TRANSPORTER: inhibition of PAH uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 6(Rattus norvegicus)
University Of Rochester School Of Medicine And Dentistry
Curated by ChEMBL
University Of Rochester School Of Medicine And Dentistry
Curated by ChEMBL
Affinity DataKi: 1.90E+3nMAssay Description:TP_TRANSPORTER: inhibition of PAH uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 6(Rattus norvegicus)
University Of Rochester School Of Medicine And Dentistry
Curated by ChEMBL
University Of Rochester School Of Medicine And Dentistry
Curated by ChEMBL
Affinity DataKi: 9.00E+3nMAssay Description:TP_TRANSPORTER: inhibition of PAH uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
Affinity DataKi: 3.00E+4nMAssay Description:TP_TRANSPORTER: inhibition of carnitine in Xenopus laevis oocytesMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
Affinity DataIC50: 26nMAssay Description:Inhibition of human URAT1 expressed in xenopus oocyte assessed as inhibition of [14C]-labelled urate uptake after 60 mins by liquid scintillation cou...More data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
Affinity DataIC50: 35nMAssay Description:Inhibition of human URAT1 expressed in human MDCK cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
Affinity DataIC50: 42nMAssay Description:Inhibition of human URAT1 expressed in xenopus oocyte assessed as inhibition of [14C]-labelled urate uptake after 60 mins by liquid scintillation cou...More data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
Affinity DataIC50: 83nMAssay Description:Inhibition of human URAT1 expressed in xenopus oocyte assessed as inhibition of [14C]-labelled urate uptake after 60 mins by liquid scintillation cou...More data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
Affinity DataIC50: 111nMAssay Description:Inhibition of human URAT1 expressed in xenopus oocyte assessed as inhibition of [14C]-labelled urate uptake after 60 mins by liquid scintillation cou...More data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
Affinity DataIC50: 138nMAssay Description:Inhibition of human URAT1 expressed in xenopus oocyte assessed as inhibition of [14C]-labelled urate uptake after 60 mins by liquid scintillation cou...More data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
Affinity DataIC50: 177nMAssay Description:Inhibition of human URAT1 expressed in xenopus oocyte assessed as inhibition of [14C]-labelled urate uptake after 60 mins by liquid scintillation cou...More data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
Affinity DataIC50: 189nMAssay Description:Inhibition of human URAT1 expressed in xenopus oocyte assessed as inhibition of [14C]-labelled urate uptake after 60 mins by liquid scintillation cou...More data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of human URAT1 expressed in human MDCK cellsMore data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
Affinity DataIC50: 287nMAssay Description:Inhibition of human URAT1 expressed in xenopus oocyte assessed as inhibition of [14C]-labelled urate uptake after 60 mins by liquid scintillation cou...More data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
Affinity DataIC50: 358nMAssay Description:Inhibition of human URAT1 expressed in xenopus oocyte assessed as inhibition of [14C]-labelled urate uptake after 60 mins by liquid scintillation cou...More data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
Affinity DataIC50: 667nMAssay Description:Inhibition of human URAT1 expressed in xenopus oocyte assessed as inhibition of [14C]-labelled urate uptake after 60 mins by liquid scintillation cou...More data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
Affinity DataIC50: 772nMAssay Description:Inhibition of human URAT1 expressed in xenopus oocyte assessed as inhibition of [14C]-labelled urate uptake after 60 mins by liquid scintillation cou...More data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
Affinity DataIC50: 1.13E+3nMAssay Description:Inhibition of human URAT1 expressed in xenopus oocyte assessed as inhibition of [14C]-labelled urate uptake after 60 mins by liquid scintillation cou...More data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
Affinity DataIC50: 1.44E+3nMAssay Description:Inhibition of human URAT1 expressed in xenopus oocyte assessed as inhibition of [14C]-labelled urate uptake after 60 mins by liquid scintillation cou...More data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
Affinity DataIC50: 1.65E+3nMAssay Description:Inhibition of human URAT1 expressed in xenopus oocyte assessed as inhibition of [14C]-labelled urate uptake after 60 mins by liquid scintillation cou...More data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
Affinity DataIC50: 2.46E+3nMAssay Description:Inhibition of human URAT1 expressed in xenopus oocyte assessed as inhibition of [14C]-labelled urate uptake after 60 mins by liquid scintillation cou...More data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
Affinity DataIC50: 2.49E+3nMAssay Description:Inhibition of human URAT1 expressed in xenopus oocyte assessed as inhibition of [14C]-labelled urate uptake after 60 mins by liquid scintillation cou...More data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of human URAT1 expressed in xenopus oocyte assessed as inhibition of [14C]-labelled urate uptake after 60 mins by liquid scintillation cou...More data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
Affinity DataIC50: 3.92E+3nMAssay Description:Inhibition of human URAT1 expressed in xenopus oocyte assessed as inhibition of [14C]-labelled urate uptake after 60 mins by liquid scintillation cou...More data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
Affinity DataIC50: 3.94E+3nMAssay Description:Inhibition of human URAT1 expressed in xenopus oocyte assessed as inhibition of [14C]-labelled urate uptake after 60 mins by liquid scintillation cou...More data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
Affinity DataIC50: 6.68E+3nMAssay Description:Inhibition of human URAT1 expressed in xenopus oocyte assessed as inhibition of [14C]-labelled urate uptake after 60 mins by liquid scintillation cou...More data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
Affinity DataIC50: 1.97E+4nMAssay Description:Inhibition of human URAT1 expressed in xenopus oocyte assessed as inhibition of [14C]-labelled urate uptake after 60 mins by liquid scintillation cou...More data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
Affinity DataIC50: 2.35E+4nMAssay Description:Inhibition of human URAT1 expressed in xenopus oocyte assessed as inhibition of [14C]-labelled urate uptake after 60 mins by liquid scintillation cou...More data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
Affinity DataIC50: 3.37E+4nMAssay Description:Inhibition of human URAT1 expressed in xenopus oocyte assessed as inhibition of [14C]-labelled urate uptake after 60 mins by liquid scintillation cou...More data for this Ligand-Target Pair
TargetSolute carrier family 22 member 12(Homo sapiens (Human))
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
University Of Colorado Anschutz Medical Campus
Curated by ChEMBL
Affinity DataIC50: 8.64E+4nMAssay Description:Inhibition of human URAT1 expressed in xenopus oocyte assessed as inhibition of [14C]-labelled urate uptake after 60 mins by liquid scintillation cou...More data for this Ligand-Target Pair