Affinity DataKi: 0.360nMAssay Description:Inhibition of human active TRKA assessed as decrease in substrate phosphorylation incubated for 2 hrs using CSKtide as substrate in presence of ATP m...More data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Inhibition of human TRKA at active state by kinetic based analysisMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Antagonism of Cysteinyl leukotriene receptor 1 from guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Antagonism of Cysteinyl leukotriene receptor 1 from guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of human TRKA at inactive state by kinetic based analysisMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 4(Homo sapiens (Human))
University of Berne
Curated by PDSP Ki Database
University of Berne
Curated by PDSP Ki Database
Affinity DataKi: 1.40nMAssay Description:Inhibition of recombinant matrix metalloprotease-3 (MMP-3)More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Antagonism of Cysteinyl leukotriene receptor 1 from guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Antagonism of Cysteinyl leukotriene receptor 1 from guinea pig lung membranesMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 4(Homo sapiens (Human))
University of Berne
Curated by PDSP Ki Database
University of Berne
Curated by PDSP Ki Database
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University of Berne
Curated by PDSP Ki Database
University of Berne
Curated by PDSP Ki Database
Affinity DataKi: 3.70nMAssay Description:Inhibition of human inactive TRKA assessed as decrease in substrate phosphorylation incubated for 2 hrs using CSKtide as substrate in presence of ATP...More data for this Ligand-Target Pair
TargetSomatostatin receptor type 4(Homo sapiens (Human))
University of Berne
Curated by PDSP Ki Database
University of Berne
Curated by PDSP Ki Database
TargetSomatostatin receptor type 1(Homo sapiens (Human))
University of Berne
Curated by PDSP Ki Database
University of Berne
Curated by PDSP Ki Database
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University of Berne
Curated by PDSP Ki Database
University of Berne
Curated by PDSP Ki Database
TargetSomatostatin receptor type 1(Homo sapiens (Human))
University of Berne
Curated by PDSP Ki Database
University of Berne
Curated by PDSP Ki Database
Affinity DataKi: 4nMAssay Description:Antagonism of Cysteinyl leukotriene receptor 1 from guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Antagonism of Cysteinyl leukotriene receptor 1 from guinea pig lung membranesMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University of Berne
Curated by PDSP Ki Database
University of Berne
Curated by PDSP Ki Database
Affinity DataKi: 5nMAssay Description:Antagonism of Cysteinyl leukotriene receptor 1 from guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 6.10nMAssay Description:Inhibition of recombinant matrix metalloprotease-2 (MMP-2)More data for this Ligand-Target Pair
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University of Berne
Curated by PDSP Ki Database
University of Berne
Curated by PDSP Ki Database
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University of Berne
Curated by PDSP Ki Database
University of Berne
Curated by PDSP Ki Database
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University of Berne
Curated by PDSP Ki Database
University of Berne
Curated by PDSP Ki Database
Affinity DataKi: 7nMAssay Description:Antagonism of Cysteinyl leukotriene receptor 1 from guinea pig lung membranesMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University of Berne
Curated by PDSP Ki Database
University of Berne
Curated by PDSP Ki Database
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University of Berne
Curated by PDSP Ki Database
University of Berne
Curated by PDSP Ki Database
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University of Berne
Curated by PDSP Ki Database
University of Berne
Curated by PDSP Ki Database
Affinity DataKi: 14nMAssay Description:Antagonism of Cysteinyl leukotriene receptor 1 from guinea pig lung membranesMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Inhibition of recombinant matrix metalloprotease-2 (MMP-2)More data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Inhibition of human inactive TRKA assessed as decrease in substrate phosphorylation incubated for 2 hrs using CSKtide as substrate in presence of ATP...More data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Binding affinity against human opioid receptor like 1 (hORL) was determined using [leucyl-3H]nociceptin in vitro in CHO cellsMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Affinity DataKi: 28nMAssay Description:Binding affinity of the compound to human Tachykinin receptor 1More data for this Ligand-Target Pair
TargetSomatostatin receptor type 1(Homo sapiens (Human))
University of Berne
Curated by PDSP Ki Database
University of Berne
Curated by PDSP Ki Database
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University of Berne
Curated by PDSP Ki Database
University of Berne
Curated by PDSP Ki Database
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University of Berne
Curated by PDSP Ki Database
University of Berne
Curated by PDSP Ki Database
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University of Berne
Curated by PDSP Ki Database
University of Berne
Curated by PDSP Ki Database
Affinity DataKi: 45nMAssay Description:Binding affinity against human opioid receptor like 1 (hORL) was determined using [leucyl-3H]nociceptin in vitro in CHO cellsMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University of Berne
Curated by PDSP Ki Database
University of Berne
Curated by PDSP Ki Database
Affinity DataKi: 45nMAssay Description:Inhibition of Hepatitis C virus genotype 1a NS3/4A protease A156T mutant expressed in Escherichia coli BL21 (DE3) cells assessed as substrate cleavag...More data for this Ligand-Target Pair
TargetSomatostatin receptor type 4(Homo sapiens (Human))
University of Berne
Curated by PDSP Ki Database
University of Berne
Curated by PDSP Ki Database
Affinity DataKi: 62nMAssay Description:Inhibition of recombinant matrix metalloprotease-3 (MMP-3)More data for this Ligand-Target Pair
Affinity DataKi: 66nMAssay Description:Inhibition of human TRKA at inactive state by kinetic based analysisMore data for this Ligand-Target Pair
Affinity DataKi: 67nMAssay Description:Inhibition of human active TRKA assessed as decrease in substrate phosphorylation incubated for 2 hrs using CSKtide as substrate in presence of ATP m...More data for this Ligand-Target Pair
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University of Berne
Curated by PDSP Ki Database
University of Berne
Curated by PDSP Ki Database
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University of Berne
Curated by PDSP Ki Database
University of Berne
Curated by PDSP Ki Database
Affinity DataKi: 72nMAssay Description:Binding affinity against human opioid receptor like 1 (hORL) was determined using [leucyl-3H]nociceptin in vitro in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 78nMAssay Description:Binding affinity against human Opioid receptor mu 1 (hMOR) was determined using [3H]diprenorphine in vitro transfected to COS-1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 78nMAssay Description:Binding affinity against human Opioid receptor kappa 1 (hKOR) was determined using [3H]diprenorphine in vitro in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 78nMAssay Description:Binding affinity against human opioid receptor like 1 (hORL) was determined using [leucyl-3H]nociceptin in vitro in CHO cellsMore data for this Ligand-Target Pair