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Found 76 with Last Name = 'werbovetz' and Initial = 'k'
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50369323(MECAMYLAMINE)
Affinity DataIC50:  600nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK-tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium leve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
The Ohio State University

LigandPNGBDBM50035218(CHEMBL61 | PODOFILOX | Podophyllinic acid lactone ...)
Affinity DataIC50:  1.40E+3nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50035218(CHEMBL61 | PODOFILOX | Podophyllinic acid lactone ...)
Affinity DataIC50:  1.56E+3nMAssay Description:Inhibition of porcine brain tubulin polymerization by GTP-induced assemblyMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50475544(CHEMBL372120)
Affinity DataIC50:  4.50E+3nMAssay Description:Inhibition of porcine brain tubulin polymerization by GTP-induced assemblyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
The Ohio State University

LigandPNGBDBM81747(Chembridge No 9067250, Class 1, 8)
Affinity DataIC50:  5.20E+3nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50437522(CHEMBL2407120)
Affinity DataIC50:  6.00E+3nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK-tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium leve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University

LigandPNGBDBM81744(Oryzalin Analogue, 3)
Affinity DataIC50:  6.40E+3nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University

LigandPNGBDBM81745(Oryzalin Analogue, 4)
Affinity DataIC50:  6.60E+3nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50437521(CHEMBL2407121)
Affinity DataIC50:  7.50E+3nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK-tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium leve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50475546(CHEMBL382519)
Affinity DataIC50:  9.10E+3nMAssay Description:Inhibition of porcine brain tubulin polymerization by GTP-induced assemblyMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50366799(TUBOCURARINE | TUBOCURARINE CHLORIDE)
Affinity DataIC50:  9.20E+3nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK-tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium leve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University

LigandPNGBDBM81746(Chembridge No 7992831, 5)
Affinity DataIC50:  1.30E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50437513(CHEMBL2407128)
Affinity DataIC50:  1.48E+4nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK-tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium leve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50437534(CHEMBL2407134)
Affinity DataIC50:  1.54E+4nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK-tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium leve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50437518(CHEMBL152025)
Affinity DataIC50:  1.71E+4nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK-tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium leve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50475541(CHEMBL196754)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of porcine brain tubulin polymerization by GTP-induced assemblyMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50437517(CHEMBL2407124)
Affinity DataIC50:  1.93E+4nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK-tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium leve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50437519(CHEMBL2407123)
Affinity DataIC50:  1.94E+4nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK-tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium leve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50437520(CHEMBL2407122)
Affinity DataIC50:  1.96E+4nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK-tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium leve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50437514(CHEMBL2407127)
Affinity DataIC50:  2.05E+4nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK-tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium leve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50437512(CHEMBL2407129)
Affinity DataIC50:  2.24E+4nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK-tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium leve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50437536(CHEMBL2407132)
Affinity DataIC50:  2.32E+4nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK-tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium leve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50437535(CHEMBL2407133)
Affinity DataIC50:  3.76E+4nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK-tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium leve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
The Ohio State University

LigandPNGBDBM81746(Chembridge No 7992831, 5)
Affinity DataIC50:  3.80E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University

LigandPNGBDBM81743(Oryzalin, 1)
Affinity DataIC50: >4.00E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
The Ohio State University

LigandPNGBDBM81743(Oryzalin, 1)
Affinity DataIC50: >4.00E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
The Ohio State University

LigandPNGBDBM81744(Oryzalin Analogue, 3)
Affinity DataIC50: >4.00E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50476974(CHEMBL55225 | sulfamidas35)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of porcine tubulin assemblyMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50475542(CHEMBL378162)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of porcine brain tubulin polymerization by GTP-induced assemblyMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM4810((3Z)-3-[(3,5-dimethyl-1H-pyrrol-2-yl)methylidene]-...)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of porcine brain tubulin polymerization by GTP-induced assemblyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50475543(CHEMBL382323)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of porcine brain tubulin polymerization by GTP-induced assemblyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50131995((E)-3-(4-hydroxybenzylidene)indolin-2-one | 3-(4-H...)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of porcine brain tubulin polymerization by GTP-induced assemblyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50475545(CHEMBL381416)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of porcine brain tubulin polymerization by GTP-induced assemblyMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50476973(CHEMBL393580)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of porcine tubulin assemblyMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50476972(CHEMBL393396)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of porcine tubulin assemblyMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50476975(CHEMBL236160)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of porcine tubulin assemblyMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
The Ohio State University

LigandPNGBDBM81745(Oryzalin Analogue, 4)
Affinity DataIC50: >5.00E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
The Ohio State University

Curated by ChEMBL
LigandPNGBDBM50437533(CHEMBL2407135)
Affinity DataIC50:  5.41E+4nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK-tsA201 cells assessed as inhibition of epibatidine-induced intracellular calcium leve...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University

LigandPNGBDBM81747(Chembridge No 9067250, Class 1, 8)
Affinity DataIC50:  5.50E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University

LigandPNGBDBM81748(Chembridge No 7946770, Class 1, 9)
Affinity DataIC50:  5.80E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University

LigandPNGBDBM81753(Chembridge No 9035165, Class 2, 13)
Affinity DataIC50:  6.00E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
The Ohio State University

LigandPNGBDBM81752(Chembridge No 9035650, Class 2, 12)
Affinity DataIC50:  6.10E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
The Ohio State University

LigandPNGBDBM81753(Chembridge No 9035165, Class 2, 13)
Affinity DataIC50:  6.30E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
The Ohio State University

LigandPNGBDBM81751(Chembridge No 9041709, Class 2, 11)
Affinity DataIC50:  6.30E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University

LigandPNGBDBM81749(Chembridge No 7960631, Class 1, 10)
Affinity DataIC50:  6.40E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University

LigandPNGBDBM81752(Chembridge No 9035650, Class 2, 12)
Affinity DataIC50:  6.60E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
The Ohio State University

LigandPNGBDBM81748(Chembridge No 7946770, Class 1, 9)
Affinity DataIC50:  6.70E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha chain(Leishmania tarentolae (Sauroleishmania tarentolae))
The Ohio State University

LigandPNGBDBM81751(Chembridge No 9041709, Class 2, 11)
Affinity DataIC50:  6.80E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
The Ohio State University

LigandPNGBDBM81749(Chembridge No 7960631, Class 1, 10)
Affinity DataIC50:  6.80E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
The Ohio State University

LigandPNGBDBM81750(Chembridge No 9063043, Class 1, 17)
Affinity DataIC50:  7.00E+4nMAssay Description:In vitro activity assay using leishmania tarentolae and porcine brain tubulin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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