Affinity DataIC50: 200nMAssay Description:Inverse agonist activity at SF-1More data for this Ligand-Target Pair
Affinity DataIC50: 7.30E+3nMAssay Description:Inverse agonist activity at SF-1More data for this Ligand-Target Pair
Affinity DataEC50: 430nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
Affinity DataEC50: 90nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
Affinity DataEC50: 22nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
Affinity DataEC50: 12nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
Affinity DataEC50: 160nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
Affinity DataEC50: 100nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
Affinity DataEC50: 60nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
Affinity DataEC50: 1.40E+3nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
Affinity DataEC50: 70nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
Affinity DataEC50: 320nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
Affinity DataEC50: 2.10E+3nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
Affinity DataEC50: 34nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
Affinity DataEC50: 230nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
Affinity DataEC50: 150nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
Affinity DataEC50: 330nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+3nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
Affinity DataEC50: 30nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
Affinity DataEC50: 1.20E+3nMpH: 7.5 T: 2°CAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human LRH1 and a TIF2-deriv...More data for this Ligand-Target Pair
Affinity DataEC50: 54nMAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human SF1 and a peptide der...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human SF1 and a peptide der...More data for this Ligand-Target Pair
Affinity DataEC50: 30nMAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human SF1 and a peptide der...More data for this Ligand-Target Pair
Affinity DataEC50: 10nMAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human SF1 and a peptide der...More data for this Ligand-Target Pair
Affinity DataEC50: 170nMAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human SF1 and a peptide der...More data for this Ligand-Target Pair
Affinity DataEC50: 140nMAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human SF1 and a peptide der...More data for this Ligand-Target Pair
Affinity DataEC50: 130nMAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human SF1 and a peptide der...More data for this Ligand-Target Pair
Affinity DataEC50: 800nMAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human SF1 and a peptide der...More data for this Ligand-Target Pair
Affinity DataEC50: 14nMAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human SF1 and a peptide der...More data for this Ligand-Target Pair
Affinity DataEC50: 130nMAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human SF1 and a peptide der...More data for this Ligand-Target Pair
Affinity DataEC50: 130nMAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human SF1 and a peptide der...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human SF1 and a peptide der...More data for this Ligand-Target Pair
Affinity DataEC50: 43nMAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human SF1 and a peptide der...More data for this Ligand-Target Pair
Affinity DataEC50: 180nMAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human SF1 and a peptide der...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human SF1 and a peptide der...More data for this Ligand-Target Pair
Affinity DataEC50: 120nMAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human SF1 and a peptide der...More data for this Ligand-Target Pair
Affinity DataEC50: 560nMAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human SF1 and a peptide der...More data for this Ligand-Target Pair
Affinity DataEC50: 700nMAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human SF1 and a peptide der...More data for this Ligand-Target Pair
Affinity DataEC50: 11nMAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human SF1 and a peptide der...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human SF1 and a peptide der...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human SF1 and a peptide der...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human SF1 and a peptide der...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:The screen utilizes a ligand mediated co-factor interaction between purified bacterial expressed ligand binding domain of human SF1 and a peptide der...More data for this Ligand-Target Pair
Affinity DataEC50: 2.51E+3nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair
Affinity DataEC50: 3.16E+3nMAssay Description:Agonist activity at human LRH-1 receptor assessed as TIF2 737-757 peptide recruitment by TR-FRET assay relative to controlMore data for this Ligand-Target Pair