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Found 6 with Last Name = 'whitworth' and Initial = 'g'
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Simon Fraser University

Curated by ChEMBL
LigandPNGBDBM50323697((3AR,5R,6S,7R,7AR)-2-(ETHYLAMINO)-5-(HYDROXYMETHYL...)
Affinity DataKi:  21nMAssay Description:Inhibition of human O-GlcNAcaseMore data for this Ligand-Target Pair
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Simon Fraser University

Curated by ChEMBL
LigandPNGBDBM50323695(2-((5R,6R,7R,8S)-8-acetamido-6,7-dihydroxy-5-(hydr...)
Affinity DataKi:  420nMAssay Description:Inhibition of human O-GlcNAcaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Simon Fraser University

Curated by ChEMBL
LigandPNGBDBM50323696((3AR,5R,6S,7R,7AR)-5-(HYDROXYMETHYL)-2-PROPYL-5,6,...)
Affinity DataKi:  600nMAssay Description:Inhibition of human O-GlcNAcaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Simon Fraser University

Curated by ChEMBL
LigandPNGBDBM149230(US8962664, 6)
Affinity DataKi:  5.60E+3nM ΔG°:  -31.2kJ/molepH: 7.4 T: 2°CAssay Description:Experimental Procedure for Kinetic Analyses: Enzymatic reactions were carried out in PBS buffer (pH 7.4) using pNP-GlcNAc as a substrate (0.5 mM) and...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Simon Fraser University

Curated by ChEMBL
LigandPNGBDBM149229(US8962664, 4)
Affinity DataKi:  7.70E+3nM ΔG°:  -30.4kJ/molepH: 7.4 T: 2°CAssay Description:Experimental Procedure for Kinetic Analyses: Enzymatic reactions were carried out in PBS buffer (pH 7.4) using pNP-GlcNAc as a substrate (0.5 mM) and...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProtein O-GlcNAcase(Homo sapiens (Human))
Simon Fraser University

Curated by ChEMBL
LigandPNGBDBM149228(US8962664, 2)
Affinity DataKi:  1.00E+4nM ΔG°:  -29.7kJ/molepH: 7.4 T: 2°CAssay Description:Experimental Procedure for Kinetic Analyses: Enzymatic reactions were carried out in PBS buffer (pH 7.4) using pNP-GlcNAc as a substrate (0.5 mM) and...More data for this Ligand-Target Pair
In DepthDetails US Patent