Affinity DataKi: 4.32E+3nMAssay Description:Reversible inhibition of human CES1 assessed as hydrolysis of 4NPA to 4NPMore data for this Ligand-Target Pair
Affinity DataKi: 2.48E+4nMAssay Description:Reversible inhibition of human CES1 assessed as hydrolysis of 4NPA to 4NPMore data for this Ligand-Target Pair
Affinity DataKi: 3.55E+5nMAssay Description:Reversible inhibition of human CES1 assessed as hydrolysis of 4NPA to 4NPMore data for this Ligand-Target Pair
Affinity DataKi: 3.63E+5nMAssay Description:Inhibition of human CES1More data for this Ligand-Target Pair
Affinity DataKi: 4.68E+5nMAssay Description:Reversible inhibition of human CES1 assessed as hydrolysis of 4NPA to 4NPMore data for this Ligand-Target Pair
Affinity DataKi: 7.07E+5nMAssay Description:Reversible inhibition of human CES1 assessed as hydrolysis of 4NPA to 4NPMore data for this Ligand-Target Pair
Affinity DataKi: 7.90E+6nMAssay Description:Inhibition of human CES2More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of recombinant human GIRK1/4 channelMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 9nMAssay Description:Inhibition of recombinant human GIRK1/4 channelMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of recombinant human GIRK1/4 channelMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 25nMAssay Description:Inhibition of recombinant human GIRK1/4 channelMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Inhibition of recombinant human GIRK1/4 channelMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 50nMAssay Description:Inhibition of recombinant human GIRK1/4 channelMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 80nMAssay Description:Inhibition of recombinant human GIRK1/4 channelMore data for this Ligand-Target Pair
Affinity DataIC50: 87nMAssay Description:Inhibition of recombinant human GIRK1/4 channelMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 100nMAssay Description:Inhibition of recombinant human GIRK1/4 channelMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 100nMAssay Description:Inhibition of GIRK1/2 (unknown origin) channelMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of recombinant human GIRK1/4 channelMore data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Inhibition of recombinant human GIRK1/4 channelMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 150nMAssay Description:Inhibition of recombinant human GIRK1/4 channelMore data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:Inhibition of recombinant human GIRK1/4 channelMore data for this Ligand-Target Pair
Affinity DataIC50: 190nMAssay Description:Inhibition of recombinant human GIRK1/4 channelMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 200nMAssay Description:Inhibition of recombinant human GIRK1/2 channelMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 220nMAssay Description:Inhibition of recombinant human GIRK1/4 channelMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 250nMAssay Description:Inhibition of recombinant human GIRK1/4 channelMore data for this Ligand-Target Pair
Affinity DataIC50: 290nMAssay Description:Inhibition of recombinant human GIRK1/4 channelMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.96E+3nMAssay Description:Time-dependent inhibition of human CES1 assessed as hydrolysis of 4NPA to 4NP preincubated for 30 mins followed by 4NPA additionMore data for this Ligand-Target Pair
Affinity DataIC50: 2.27E+3nMAssay Description:Time-dependent inhibition of human CES1 assessed as hydrolysis of 4NPA to 4NP preincubated for 60 mins followed by 4NPA additionMore data for this Ligand-Target Pair
Affinity DataIC50: 2.51E+3nMAssay Description:Time-dependent inhibition of human CES1 assessed as hydrolysis of 4NPA to 4NP preincubated for 10 mins followed by 4NPA additionMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of recombinant human GIRK1/4 channelMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.42E+4nMAssay Description:Inhibition of recombinant human Cav1.2More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of recombinant hERG in the presence of dofetilide by competitive binding assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of recombinant hERG in the presence of dofetilide by competitive binding assayMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of recombinant human KCNQ1More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant human KCNQ1More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant human KCNQ1More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant hERG in the presence of dofetilide by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant hERG in the presence of dofetilide by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant human KCNQ1More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant human Cav1.2More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant human Cav1.2More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant human Nav1.5More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant human Nav1.5More data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant human Nav1.5More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant human Nav1.5More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant human Cav1.2More data for this Ligand-Target Pair