Compile Data Set for Download or QSAR
maximum 50k data
Found 279 with Last Name = 'williams' and Initial = 'me'
TargetAdenosine receptor A2a(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50243660(2-Furan-2-yl-7-[2-(7-nitro-1,2,4,5-tetrahydro-benz...)
Affinity DataKi:  0.700nMAssay Description:Antagonist activity at human adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50243661(7-[2-(7-Bromo-1,2,4,5-tetrahydro-benzo[d]azepin-3-...)
Affinity DataKi:  1.10nMAssay Description:Antagonist activity at human adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169328(5-{4-[3-(5-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-...)
Affinity DataKi:  1.10nMAssay Description:In vitro ability to displace [3H]-SCH-58,261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169314(2-Furan-2-yl-7-pyridin-2-yl-[1,2,4]triazolo[1,5-c]...)
Affinity DataKi:  1.40nMAssay Description:In vitro ability to displace [3H]-SCH-58,261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50243027(2-Furan-2-yl-7-{2-[8-(2-methoxy-ethoxy)-3,4-dihydr...)
Affinity DataKi:  1.5nMAssay Description:Antagonist activity at human adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50242875(7-[2-(3-Bromo-7,8-dihydro-5H-[1,6]naphthyridin-6-y...)
Affinity DataKi:  1.60nMAssay Description:Antagonist activity at human adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169318(2-Furan-2-yl-7-pyridin-4-yl-[1,2,4]triazolo[1,5-c]...)
Affinity DataKi:  1.90nMAssay Description:In vitro ability to displace [3H]-SCH-58,261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50243696(2-Furan-2-yl-7-[2-(7-methoxy-1,2,4,5-tetrahydro-be...)
Affinity DataKi:  1.90nMAssay Description:Antagonist activity at human adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50243025(7-[2-(6,7-Dimethoxy-3-methyl-3,4-dihydro-1H-isoqui...)
Affinity DataKi:  1.90nMAssay Description:Antagonist activity at human adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50242874(7-[2-(3-Cyclopropyl-7,8-dihydro-5H-[1,6]naphthyrid...)
Affinity DataKi:  1.90nMAssay Description:Antagonist activity at human adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50243659(2-Furan-2-yl-7-[2-(1,2,4,5-tetrahydro-benzo[d]azep...)
Affinity DataKi:  2nMAssay Description:Antagonist activity at human adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50243697(2-Furan-2-yl-7-{2-[7-(2-methoxy-ethoxy)-1,2,4,5-te...)
Affinity DataKi:  2nMAssay Description:Antagonist activity at human adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50242873(2-Furan-2-yl-7-[2-(3-methyl-7,8-dihydro-5H-[1,6]na...)
Affinity DataKi:  2nMAssay Description:Antagonist activity at human adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50048466(2-(furan-2-yl)-7-phenethyl-7H-pyrazolo[4,3-e][1,2,...)
Affinity DataKi:  2nMAssay Description:Antagonist activity at human adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169326(7-(3-{4-[3,5-Difluoro-4-(2-methoxy-ethoxy)-phenyl]...)
Affinity DataKi:  2.20nMAssay Description:In vitro ability to displace [3H]-SCH-58,261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50243026(7-[2-(1-Benzyl-6,7-dimethoxy-3,4-dihydro-1H-isoqui...)
Affinity DataKi:  2.30nMAssay Description:Antagonist activity at human adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169313(2-Furan-2-yl-7-[3-(4-thiazol-2-yl-piperazin-1-ylme...)
Affinity DataKi:  2.40nMAssay Description:In vitro ability to displace [3H]-SCH-58,261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50243028(2-Furan-2-yl-7-[2-(6-methoxy-3,4-dihydro-1H-isoqui...)
Affinity DataKi:  2.5nMAssay Description:Antagonist activity at human adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169312(7-(3-{4-[2-Fluoro-4-(2-methoxy-ethoxy)-phenyl]-pip...)
Affinity DataKi:  2.70nMAssay Description:In vitro ability to displace [3H]-SCH-58,261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169331(2-Furan-2-yl-7-(3-{4-[4-(2-methoxy-ethoxy)-2-methy...)
Affinity DataKi:  2.70nMAssay Description:In vitro ability to displace [3H]-SCH-58,261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169323(2-Furan-2-yl-7-(3-{4-[4-(2-methoxy-ethoxy)-phenyl]...)
Affinity DataKi:  2.80nMAssay Description:In vitro ability to displace [3H]-SCH-58,261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169317(CHEMBL360446 | [3-(5-Amino-2-furan-2-yl-[1,2,4]tri...)
Affinity DataKi:  2.80nMAssay Description:In vitro ability to displace [3H]-SCH-58,261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169332(7-(3-{4-[2-Chloro-4-(2-methoxy-ethoxy)-phenyl]-pip...)
Affinity DataKi:  2.90nMAssay Description:In vitro ability to displace [3H]-SCH-58,261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169309(7-(2,4-Dimethoxy-phenyl)-2-furan-2-yl-[1,2,4]triaz...)
Affinity DataKi:  2.90nMAssay Description:In vitro ability to displace [3H]-SCH-58,261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50242876(2-Furan-2-yl-7-{2-[3-(2-methoxy-ethoxy)-7,8-dihydr...)
Affinity DataKi:  3.10nMAssay Description:Antagonist activity at human adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50243029(2-Furan-2-yl-7-[2-(7-methoxy-3,4-dihydro-1H-isoqui...)
Affinity DataKi:  3.20nMAssay Description:Antagonist activity at human adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50243695(7-[2-(7-Chloro-1,2,4,5-tetrahydro-benzo[d]azepin-3...)
Affinity DataKi:  3.30nMAssay Description:Antagonist activity at human adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169304(2-Furan-2-yl-7-(3-{4-[3-methoxy-4-(2-methoxy-ethox...)
Affinity DataKi:  3.30nMAssay Description:In vitro ability to displace [3H]-SCH-58,261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169339(2-Furan-2-yl-7-{3-[(methyl-phenethyl-amino)-methyl...)
Affinity DataKi:  3.60nMAssay Description:In vitro ability to displace [3H]-SCH-58,261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169306(2-{4-[3-(5-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-...)
Affinity DataKi:  3.60nMAssay Description:In vitro ability to displace [3H]-SCH-58,261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169322(2-Furan-2-yl-7-m-tolyl-[1,2,4]triazolo[1,5-c]pyrim...)
Affinity DataKi:  3.70nMAssay Description:In vitro ability to displace [3H]-SCH-58,261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169324(2-Furan-2-yl-7-(3-{4-[3-(2-methoxy-ethoxy)-phenyl]...)
Affinity DataKi:  4nMAssay Description:In vitro ability to displace [3H]-SCH-58,261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50242937(7-[2-(3,4-Dihydro-1H-isoquinolin-2-yl)-ethyl]-2-fu...)
Affinity DataKi:  4.10nMAssay Description:Antagonist activity at human adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169338(2-(furan-2-yl)-7-(2-methoxyphenyl)-[1,2,4]triazolo...)
Affinity DataKi:  4.30nMAssay Description:In vitro ability to displace [3H]-SCH-58,261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169315(2-Furan-2-yl-7-thiophen-2-yl-[1,2,4]triazolo[1,5-c...)
Affinity DataKi:  4.40nMAssay Description:In vitro ability to displace [3H]-SCH-58,261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169333(2-Furan-2-yl-7-(2,3,4-trimethoxy-phenyl)-[1,2,4]tr...)
Affinity DataKi:  4.5nMAssay Description:In vitro ability to displace [3H]-SCH-58,261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169330(2-Furan-2-yl-7-(3,4,5-trimethoxy-phenyl)-[1,2,4]tr...)
Affinity DataKi:  4.5nMAssay Description:In vitro ability to displace [3H]-SCH-58,261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169319(7-(2,5-Dimethoxy-phenyl)-2-furan-2-yl-[1,2,4]triaz...)
Affinity DataKi:  4.5nMAssay Description:In vitro ability to displace [3H]-SCH-58,261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169316(2-Furan-2-yl-7-[3-(4-phenyl-piperazin-1-ylmethyl)-...)
Affinity DataKi:  4.60nMAssay Description:In vitro ability to displace [3H]-SCH-58,261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169321(2-Furan-2-yl-7-[3-(4-phenyl-piperidin-1-ylmethyl)-...)
Affinity DataKi:  4.60nMAssay Description:In vitro ability to displace [3H]-SCH-58,261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169336(2-Furan-2-yl-7-(4-isopropyl-phenyl)-[1,2,4]triazol...)
Affinity DataKi:  4.70nMAssay Description:In vitro ability to displace [3H]-SCH-58,261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50243698(7-[2-(7,8-Dihydro-5H-[1,6]naphthyridin-6-yl)-ethyl...)
Affinity DataKi:  4.80nMAssay Description:Antagonist activity at human adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169334(2-Furan-2-yl-7-(3-methoxy-phenyl)-[1,2,4]triazolo[...)
Affinity DataKi:  5nMAssay Description:In vitro ability to displace [3H]-SCH-58,261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169301(7-(3-Amino-phenyl)-2-furan-2-yl-[1,2,4]triazolo[1,...)
Affinity DataKi:  5nMAssay Description:In vitro ability to displace [3H]-SCH-58,261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50242940(2-Furan-2-yl-7-[2-(2-trifluoromethyl-7,8-dihydro-5...)
Affinity DataKi:  5nMAssay Description:Antagonist activity at human adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50243658(2-Furan-2-yl-7-{2-[7-(2-methoxy-ethoxy)-3,4-dihydr...)
Affinity DataKi:  5.10nMAssay Description:Antagonist activity at human adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50242936(2-Furan-2-yl-7-[2-(5-methoxy-1,3-dihydro-isoindol-...)
Affinity DataKi:  5.40nMAssay Description:Antagonist activity at human adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169310(3-(5-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-c]pyri...)
Affinity DataKi:  5.40nMAssay Description:In vitro ability to displace [3H]-SCH-58,261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50169303(7-Biphenyl-3-yl-2-furan-2-yl-[1,2,4]triazolo[1,5-c...)
Affinity DataKi:  5.5nMAssay Description:In vitro ability to displace [3H]-SCH-58,261 from A2A adenosine receptor in RatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50243657(2-Furan-2-yl-7-[2-(4-methoxy-1,3-dihydro-isoindol-...)
Affinity DataKi:  6nMAssay Description:Antagonist activity at human adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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