TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Cambridge University Forvie Site
Curated by ChEMBL
Cambridge University Forvie Site
Curated by ChEMBL
Affinity DataKi: 0.0400nMAssay Description:In vitro binding affinity at Bombesin BB2 receptor in the presence of [125I]-[Tyr] bombesin.More data for this Ligand-Target Pair
Affinity DataKi: 0.0680nMAssay Description:Antagonism of recombinant human bombesin receptor (bb1) labeled with [125I]- [Tyr] bombesin stably expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.150nMAssay Description:Antagonism of recombinant human bombesin receptor (bb1) labeled with [125I]- [Tyr] bombesin stably expressed in CHO cellsMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Cambridge University Forvie Site
Curated by ChEMBL
Cambridge University Forvie Site
Curated by ChEMBL
Affinity DataKi: 0.150nMAssay Description:In vitro binding affinity at Bombesin BB2 receptor in the presence of [125I]-[Tyr] bombesin.More data for this Ligand-Target Pair
Affinity DataKi: 0.170nMAssay Description:Antagonism of recombinant human bombesin receptor (bb1) labeled with [125I]- [Tyr] bombesin stably expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Antagonism of recombinant human bombesin receptor (bb1) labeled with [125I]- [Tyr] bombesin stably expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.320nMAssay Description:Antagonism of recombinant human bombesin receptor (bb1) labeled with [125I]- [Tyr] bombesin stably expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.390nMAssay Description:Antagonism of recombinant human bombesin receptor (bb1) labeled with [125I]- [Tyr] bombesin stably expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.440nMAssay Description:Antagonism of recombinant human bombesin receptor (bb1) labeled with [125I]- [Tyr] bombesin stably expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.460nMAssay Description:Antagonism of recombinant human bombesin receptor (bb1) labeled with [125I]- [Tyr] bombesin stably expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.520nMAssay Description:Antagonism of recombinant human bombesin receptor (bb1) labeled with [125I]- [Tyr] bombesin stably expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.590nMAssay Description:Antagonism of recombinant human bombesin receptor (bb1) labeled with [125I]- [Tyr] bombesin stably expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.620nMAssay Description:Antagonism of recombinant human bombesin receptor (bb1) labeled with [125I]- [Tyr] bombesin stably expressed in CHO cellsMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Cambridge University Forvie Site
Curated by ChEMBL
Cambridge University Forvie Site
Curated by ChEMBL
Affinity DataKi: 0.700nMAssay Description:In vitro binding affinity at Bombesin BB2 receptor in the presence of [125I]-[Tyr] bombesin.More data for this Ligand-Target Pair
Affinity DataKi: 0.970nMAssay Description:Antagonism of recombinant human bombesin receptor (bb1) labeled with [125I]- [Tyr] bombesin stably expressed in CHO cellsMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Cambridge University Forvie Site
Curated by ChEMBL
Cambridge University Forvie Site
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Antagonistic activity against cloned human Bombesin receptor bb2 labeled with [125I]- [Tyr] bombesin stably expressed in CHO cells; 0.66-1.3More data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Antagonism of recombinant human bombesin receptor (bb1) labeled with [125I]- [Tyr] bombesin stably expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Antagonism of recombinant human bombesin receptor (bb1) labeled with [125I]- [Tyr] bombesin stably expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Antagonism of recombinant human bombesin receptor (bb1) labeled with [125I]- [Tyr] bombesin stably expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Antagonism of recombinant human bombesin receptor (bb1) labeled with [125I]- [Tyr] bombesin stably expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:Antagonism of recombinant human bombesin receptor (bb1) labeled with [125I]- [Tyr] bombesin stably expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Antagonism of recombinant human bombesin receptor (bb1) labeled with [125I]- [Tyr] bombesin stably expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Antagonist activity at human CXCR3 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Binding affinity to CXCR3 receptor expressed in CHO cells assessed as ITAC-induced [35]GTPgammaS bindingMore data for this Ligand-Target Pair
Affinity DataKi: 3.40nMAssay Description:Antagonism of recombinant human bombesin receptor (bb1) labeled with [125I]- [Tyr] bombesin stably expressed in CHO cellsMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Cambridge University Forvie Site
Curated by ChEMBL
Cambridge University Forvie Site
Curated by ChEMBL
Affinity DataKi: 3.70nMAssay Description:In vitro binding affinity at Bombesin BB2 receptor in the presence of [125I]-[Tyr] bombesin.More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity to CXCR3 receptor expressed in CHO cells assessed as ITAC-induced [35]GTPgammaS bindingMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Binding affinity to CXCR3 receptor expressed in CHO cells assessed as ITAC-induced [35]GTPgammaS bindingMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Cambridge University Forvie Site
Curated by ChEMBL
Cambridge University Forvie Site
Curated by ChEMBL
Affinity DataKi: 5.80nMAssay Description:In vitro binding affinity at Bombesin BB2 receptor in the presence of [125I]-[Tyr] bombesin.More data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Binding affinity to CXCR3 receptor expressed in CHO cells assessed as ITAC-induced [35]GTPgammaS bindingMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Binding affinity to CXCR3 receptor expressed in CHO cells assessed as ITAC-induced [35]GTPgammaS bindingMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Antagonist activity at mouse CXCR3More data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Antagonist activity at mouse CXCR3More data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Antagonism of recombinant human bombesin receptor (bb1) labeled with [125I]- [Tyr] bombesin stably expressed in CHO cellsMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Cambridge University Forvie Site
Curated by ChEMBL
Cambridge University Forvie Site
Curated by ChEMBL
Affinity DataKi: 6.40nMAssay Description:In vitro binding affinity at Bombesin BB2 receptor in the presence of [125I]-[Tyr] bombesin.More data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Binding affinity to CXCR3 receptor expressed in CHO cells assessed as ITAC-induced [35]GTPgammaS bindingMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Antagonist activity at human CXCR3 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Antagonist activity at human CXCR3 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Cambridge University Forvie Site
Curated by ChEMBL
Cambridge University Forvie Site
Curated by ChEMBL
Affinity DataKi: 9nMAssay Description:In vitro binding affinity at Bombesin BB2 receptor in the presence of [125I]-[Tyr] bombesin.More data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Binding affinity to CXCR3 receptor expressed in CHO cells assessed as ITAC-induced [35]GTPgammaS bindingMore data for this Ligand-Target Pair
Affinity DataKi: 9.10nMAssay Description:Antagonism of recombinant human bombesin receptor (bb1) labeled with [125I]- [Tyr] bombesin stably expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 9.40nMAssay Description:Antagonism of recombinant human bombesin receptor (bb1) labeled with [125I]- [Tyr] bombesin stably expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Antagonist activity at human CXCR3 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Antagonist activity at human CXCR3 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Binding affinity to CXCR3 receptor expressed in CHO cells assessed as ITAC-induced [35]GTPgammaS bindingMore data for this Ligand-Target Pair
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
Cambridge University Forvie Site
Curated by ChEMBL
Cambridge University Forvie Site
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:In vitro binding affinity at Bombesin BB2 receptor in the presence of [125I]-[Tyr] bombesin.More data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Antagonist activity at human CXCR3 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Binding affinity to CXCR3 receptor expressed in CHO cells assessed as ITAC-induced [35]GTPgammaS bindingMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Binding affinity to CXCR3 receptor expressed in CHO cells assessed as ITAC-induced [35]GTPgammaS bindingMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Antagonist activity at human CXCR3 by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair