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Found 5 with Last Name = 'willoughby' and Initial = 'me'
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50260355(CHEMBL2063071)
Affinity DataIC50:  4.30E+3nMAssay Description:Inhibition of human ABCG2 expressed in Sf9 cell membranes assessed as reduction in [125I]-IAAP binding incubated for 20 mins under UV light irradiati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50260355(CHEMBL2063071)
Affinity DataIC50:  9.30E+3nMAssay Description:Inhibition of human MDR1 expressed in Sf9 cell membranes assessed as reduction in [125I]-IAAP binding incubated for 20 mins under UV light irradiatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50260355(CHEMBL2063071)
Affinity DataIC50:  1.15E+4nMAssay Description:Inhibition of ABCG2 in human MCF7/FLV1000 cells assessed as increase in calcein-AM accumulation incubated for 10 mins by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50260356(CHEMBL2063072)
Affinity DataIC50:  1.33E+4nMAssay Description:Inhibition of ABCG2 in human MCF7/FLV1000 cells assessed as increase in calcein-AM accumulation incubated for 10 mins by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50260357(CHEMBL2063070)
Affinity DataIC50:  2.82E+4nMAssay Description:Inhibition of ABCG2 in human MCF7/FLV1000 cells assessed as increase in calcein-AM accumulation incubated for 10 mins by flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed