TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of human ABCG2 expressed in Sf9 cell membranes assessed as reduction in [125I]-IAAP binding incubated for 20 mins under UV light irradiati...More data for this Ligand-Target Pair
Affinity DataIC50: 9.30E+3nMAssay Description:Inhibition of human MDR1 expressed in Sf9 cell membranes assessed as reduction in [125I]-IAAP binding incubated for 20 mins under UV light irradiatio...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataIC50: 1.15E+4nMAssay Description:Inhibition of ABCG2 in human MCF7/FLV1000 cells assessed as increase in calcein-AM accumulation incubated for 10 mins by flow cytometryMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataIC50: 1.33E+4nMAssay Description:Inhibition of ABCG2 in human MCF7/FLV1000 cells assessed as increase in calcein-AM accumulation incubated for 10 mins by flow cytometryMore data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Purdue University
Curated by ChEMBL
Purdue University
Curated by ChEMBL
Affinity DataIC50: 2.82E+4nMAssay Description:Inhibition of ABCG2 in human MCF7/FLV1000 cells assessed as increase in calcein-AM accumulation incubated for 10 mins by flow cytometryMore data for this Ligand-Target Pair