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Found 172 with Last Name = 'wilson' and Initial = 'fx'
TargetInterleukin-8(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291126(CHEMBL265735 | CHEMBL3856136 | Interleukin-8 inhib...)
Affinity DataKi:  2.30E+3nMAssay Description:Inhibition of Interleukin-8 (IL-8)More data for this Ligand-Target Pair
In DepthDetails Article
TargetInterleukin-8(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291119(CHEMBL267510 | CHEMBL3856125 | Interleukin-8 inhib...)
Affinity DataKi:  4.00E+3nMAssay Description:Inhibition of Interleukin-8 (IL-8)More data for this Ligand-Target Pair
In DepthDetails Article
TargetInterleukin-8(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291124(CHEMBL3856133 | CHEMBL411572 | Interleukin-8 inhib...)
Affinity DataKi:  4.00E+3nMAssay Description:Inhibition of Interleukin-8 (IL-8)More data for this Ligand-Target Pair
In DepthDetails Article
TargetInterleukin-8(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291118(CHEMBL3856131 | CHEMBL438589 | Interleukin-8 inhib...)
Affinity DataKi:  6.00E+3nMAssay Description:Inhibition of Interleukin-8 (IL-8)More data for this Ligand-Target Pair
In DepthDetails Article
TargetInterleukin-8(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291131(CHEMBL3856127 | CHEMBL413247 | Interleukin-8 inhib...)
Affinity DataKi:  7.00E+3nMAssay Description:Inhibition of Interleukin-8 (IL-8)More data for this Ligand-Target Pair
In DepthDetails Article
TargetInterleukin-8(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291125(CHEMBL3856135 | CHEMBL411548 | Interleukin-8 inhib...)
Affinity DataKi:  9.30E+3nMAssay Description:Inhibition of Interleukin-8 (IL-8)More data for this Ligand-Target Pair
In DepthDetails Article
TargetInterleukin-8(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291120(CHEMBL3856128 | CHEMBL410171 | Interleukin-8 inhib...)
Affinity DataKi:  1.00E+4nMAssay Description:Inhibition of Interleukin-8 (IL-8)More data for this Ligand-Target Pair
In DepthDetails Article
TargetInterleukin-8(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291122(CHEMBL3856126 | CHEMBL428324 | Interleukin-8 inhib...)
Affinity DataKi:  1.20E+4nMAssay Description:Inhibition of Interleukin-8 (IL-8)More data for this Ligand-Target Pair
In DepthDetails Article
TargetInterleukin-8(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291128(CHEMBL267749 | CHEMBL3856129 | Interleukin-8 inhib...)
Affinity DataKi:  1.30E+4nMAssay Description:Inhibition of Interleukin-8 (IL-8)More data for this Ligand-Target Pair
In DepthDetails Article
TargetInterleukin-8(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50213962(CHEMBL410765)
Affinity DataKi:  1.30E+4nMAssay Description:Inhibition of Interleukin-8 (IL-8)More data for this Ligand-Target Pair
In DepthDetails Article
TargetInterleukin-8(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291130(CHEMBL3856130 | CHEMBL405300 | Interleukin-8 inhib...)
Affinity DataKi:  1.40E+4nMAssay Description:Inhibition of Interleukin-8 (IL-8)More data for this Ligand-Target Pair
In DepthDetails Article
TargetInterleukin-8(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291123(CHEMBL3856132 | CHEMBL410211 | Interleukin-8 inhib...)
Affinity DataKi:  3.10E+4nMAssay Description:Inhibition of Interleukin-8 (IL-8)More data for this Ligand-Target Pair
In DepthDetails Article
TargetInterleukin-8(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291121(CHEMBL2370828 | CHEMBL3856124 | Interleukin-8 inhi...)
Affinity DataKi:  1.06E+5nMAssay Description:Inhibition of Interleukin-8 (IL-8)More data for this Ligand-Target Pair
In DepthDetails Article
TargetInterleukin-8(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291129(CHEMBL2370827 | CHEMBL3856134 | Interleukin-8 inhi...)
Affinity DataKi:  3.83E+5nMAssay Description:Inhibition of Interleukin-8 (IL-8)More data for this Ligand-Target Pair
In DepthDetails Article
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Roche Discover Welwyn

Curated by ChEMBL
LigandPNGBDBM50096730(4-[3-Carboxy-2-(3-carboxy-propionylamino)-propiony...)
Affinity DataIC50:  4nMAssay Description:Inhibitory activity against non-nucleoside reverse transcriptase inhibitors (NNRTI) -resistant HIV-1 strain A17 variant with Y181C plus K103N mutatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Roche Discover Welwyn

Curated by ChEMBL
LigandPNGBDBM50096734((S)-4-[(S)-3-Carboxy-2-(3-carboxy-propionylamino)-...)
Affinity DataIC50:  4nMAssay Description:Inhibitory activity against non-nucleoside reverse transcriptase inhibitors (NNRTI) -resistant HIV-1 strain A17 with a Y181C mutation in RT (reverse ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Roche Discover Welwyn

Curated by ChEMBL
LigandPNGBDBM50096729((S)-4-((S)-1-{(S)-1-[(S)-1-((R)-1-Benzylaminooxaly...)
Affinity DataIC50:  4nMAssay Description:Binding affinity towards 5-hydroxytryptamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Roche Discover Welwyn

Curated by ChEMBL
LigandPNGBDBM50096726(4-[3-Carboxy-2-(3-carboxy-propionylamino)-propiony...)
Affinity DataIC50:  4nMAssay Description:Binding affinity towards 5-hydroxytryptamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Roche Discover Welwyn

Curated by ChEMBL
LigandPNGBDBM50096727((S)-4-[(S)-3-Carboxy-2-(3-carboxy-propionylamino)-...)
Affinity DataIC50:  6nMAssay Description:Inhibitory activity against non-nucleoside reverse transcriptase inhibitors (NNRTI) -resistant HIV-1 strain A17 variant with Y181C plus K103N mutatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Roche Discover Welwyn

Curated by ChEMBL
LigandPNGBDBM50096725(4-[3-Carboxy-2-(3-carboxy-propionylamino)-propiony...)
Affinity DataIC50:  7nMAssay Description:Inhibitory activity against delta receptor of (endomorphin 2) in mouse vas deferens was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Roche Discover Welwyn

Curated by ChEMBL
LigandPNGBDBM50096733(4-[3-Carboxy-2-(3-carboxy-propionylamino)-propiony...)
Affinity DataIC50:  7nMAssay Description:Binding affinity towards 5-hydroxytryptamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Roche Discover Welwyn

Curated by ChEMBL
LigandPNGBDBM50096728((S)-4-((S)-1-{(S)-1-[(S)-1-((S)-1-Amino-2-carbamoy...)
Affinity DataIC50:  7nMAssay Description:Inhibitory activity against non-nucleoside reverse transcriptase inhibitors (NNRTI) -resistant HIV-1 strain A17 with a Y181C mutation in RT (reverse ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Roche Discover Welwyn

Curated by ChEMBL
LigandPNGBDBM50096732(4-[3-Carboxy-2-(3-carboxy-propionylamino)-propiony...)
Affinity DataIC50:  8nMAssay Description:Inhibitory activity against non-nucleoside reverse transcriptase inhibitors (NNRTI) -resistant HIV-1 strain A17 with a Y181C mutation in RT (reverse ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Roche Discover Welwyn

Curated by ChEMBL
LigandPNGBDBM50096724((S)-4-((S)-1-{(S)-1-[(S)-1-((R)-1-Aminooxalyl-pent...)
Affinity DataIC50:  11nMAssay Description:Inhibitory activity against non-nucleoside reverse transcriptase inhibitors (NNRTI) -resistant HIV-1 strain A17 variant with Y181C plus K103N mutatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-C(Homo sapiens (Human))
Roche Discover Welwyn

Curated by ChEMBL
LigandPNGBDBM50096724((S)-4-((S)-1-{(S)-1-[(S)-1-((R)-1-Aminooxalyl-pent...)
Affinity DataIC50:  300nMAssay Description:Compound was tested for inhibition of Serine protease chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)
University College London

Curated by ChEMBL
LigandPNGBDBM50134735(CHEMBL531018 | GNF-Pf-2870 | SJ000111341 | TCMDC-1...)
Affinity DataIC50:  300nMAssay Description:Inhibition of Staphylococcus aureus DNA gyrase assessed as reduction in enzyme-catalyzed supercoiling of relaxed circular pBR322 DNA incubated for 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein/Non-structural protein 4A(Hepatitis C virus)
Roche Discover Welwyn

Curated by ChEMBL
LigandPNGBDBM50096731(4-[3-Carboxy-2-(3-carboxy-propionylamino)-propiony...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibitory activity against non-nucleoside reverse transcriptase inhibitors (NNRTI) -resistant HIV-1 strain A17 variant with Y181C plus K103N mutatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50519637(CHEMBL4550375)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of monoamino oxidase B (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50519636(BMN 195 | BMN-195 | Ezutromid | SMT-C1100 | SMTC-1...)
Affinity DataIC50:  5.40E+3nMAssay Description:Inhibition of CYP1A2 in human liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)
University College London

Curated by ChEMBL
LigandPNGBDBM50134758(CHEMBL3753934)
Affinity DataIC50:  5.60E+3nMAssay Description:Inhibition of Staphylococcus aureus DNA gyrase assessed as reduction in enzyme-catalyzed supercoiling of relaxed circular pBR322 DNA incubated for 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)
University College London

Curated by ChEMBL
LigandPNGBDBM50134757(CHEMBL3752020)
Affinity DataIC50:  8.80E+3nMAssay Description:Inhibition of Staphylococcus aureus DNA gyrase assessed as reduction in enzyme-catalyzed supercoiling of relaxed circular pBR322 DNA incubated for 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMultidrug and toxin extrusion protein 1(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50519637(CHEMBL4550375)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of MATE1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Roche Discover Welwyn

Curated by ChEMBL
LigandPNGBDBM50096724((S)-4-((S)-1-{(S)-1-[(S)-1-((R)-1-Aminooxalyl-pent...)
Affinity DataIC50:  1.20E+4nMAssay Description:Compound was tested for inhibition of ElastaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50121975((6-Methoxy-quinolin-4-yl)-(5-vinyl-1-aza-bicyclo[2...)
Affinity DataIC50:  2.80E+4nMAssay Description:Inhibition of human CYP3A4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetDNA gyrase subunit A/B(Staphylococcus aureus)
University College London

Curated by ChEMBL
LigandPNGBDBM50134759(CHEMBL3753858)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Staphylococcus aureus DNA gyrase assessed as reduction in enzyme-catalyzed supercoiling of relaxed circular pBR322 DNA incubated for 30...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
Roche Discover Welwyn

Curated by ChEMBL
LigandPNGBDBM50096724((S)-4-((S)-1-{(S)-1-[(S)-1-((R)-1-Aminooxalyl-pent...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibitory activity against Opioid receptor mu 1 of (endomorphin 2) in guinea pig ileum was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUtrophin(Homo sapiens)
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50519636(BMN 195 | BMN-195 | Ezutromid | SMT-C1100 | SMTC-1...)
Affinity DataEC50:  110nMAssay Description:Activation of human utrophin-1 in mouse mdx myoblasts by H2K-mdx utrnA-luc assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUtrophin(Homo sapiens)
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50519637(CHEMBL4550375)
Affinity DataEC50:  370nMAssay Description:Activation of human utrophin-1 in mouse mdx myoblasts by H2K-mdx utrnA-luc assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUtrophin(Homo sapiens)
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50519637(CHEMBL4550375)
Affinity DataEC50: >1.00E+4nMAssay Description:Activation of human utrophin-1 in iDMD cells by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUtrophin(Homo sapiens)
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50519638(CHEMBL4442951)
Affinity DataEC50:  8.35E+3nMAssay Description:Activation of human utrophin-1 in iDMD cells by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUtrophin(Homo sapiens)
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50519636(BMN 195 | BMN-195 | Ezutromid | SMT-C1100 | SMTC-1...)
Affinity DataEC50:  1.28E+3nMAssay Description:Activation of human utrophin-1 in iDMD cells by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUtrophin(Homo sapiens)
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50519638(CHEMBL4442951)
Affinity DataEC50:  120nMAssay Description:Activation of human utrophin-1 in mouse mdx myoblasts by H2K-mdx utrnA-luc assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUtrophin(Homo sapiens)
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50519636(BMN 195 | BMN-195 | Ezutromid | SMT-C1100 | SMTC-1...)
Affinity DataEC50:  187nMAssay Description:Modulation of human utrophinA expressed in mouse H2K cells assessed as upregulation of utrophin production after 24 hrs by luciferase reporter gene a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUtrophin(Homo sapiens)
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50542742(CHEMBL4639832)
Affinity DataEC50:  10nMAssay Description:Modulation of human utrophinA expressed in mouse H2K cells assessed as upregulation of utrophin production after 24 hrs by luciferase reporter gene a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUtrophin(Homo sapiens)
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50542743(CHEMBL4637833)
Affinity DataEC50:  38nMAssay Description:Modulation of human utrophinA expressed in mouse H2K cells assessed as upregulation of utrophin production after 24 hrs by luciferase reporter gene a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUtrophin(Homo sapiens)
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50542744(CHEMBL4636035)
Affinity DataEC50:  110nMAssay Description:Modulation of human utrophinA expressed in mouse H2K cells assessed as upregulation of utrophin production after 24 hrs by luciferase reporter gene a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUtrophin(Homo sapiens)
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50542745(CHEMBL4644129)
Affinity DataEC50:  146nMAssay Description:Modulation of human utrophinA expressed in mouse H2K cells assessed as upregulation of utrophin production after 24 hrs by luciferase reporter gene a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUtrophin(Homo sapiens)
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50542746(CHEMBL4639067)
Affinity DataEC50:  4nMAssay Description:Modulation of human utrophinA expressed in mouse H2K cells assessed as upregulation of utrophin production after 24 hrs by luciferase reporter gene a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUtrophin(Homo sapiens)
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50542747(CHEMBL4638445)
Affinity DataEC50:  71nMAssay Description:Modulation of human utrophinA expressed in mouse H2K cells assessed as upregulation of utrophin production after 24 hrs by luciferase reporter gene a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUtrophin(Homo sapiens)
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50542748(CHEMBL4641041)
Affinity DataEC50:  26nMAssay Description:Modulation of human utrophinA expressed in mouse H2K cells assessed as upregulation of utrophin production after 24 hrs by luciferase reporter gene a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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