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Found 62 with Last Name = 'wilson' and Initial = 'wd'
TargetDNA topoisomerase 2-alpha/2-beta(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50470684(CHEMBL173975)
Affinity DataIC50:  500nMAssay Description:Inhibitory activity for 50% on topoisomerase II isolated from Giardia lambliaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha/2-beta(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50470690(CHEMBL367883)
Affinity DataIC50:  500nMAssay Description:Inhibitory activity for 50% on topoisomerase II isolated from Giardia lambliaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha/2-beta(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50470688(CHEMBL170751)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibitory activity for 50% on topoisomerase II isolated from Giardia lambliaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha/2-beta(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50470689(CHEMBL171287)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibitory activity for 50% on topoisomerase II isolated from Giardia lambliaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha/2-beta(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50470685(CHEMBL557158)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibitory activity for 50% on topoisomerase II isolated from Giardia lambliaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha/2-beta(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50470686(CHEMBL170447)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibitory activity for 50% on topoisomerase II isolated from Giardia lambliaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha/2-beta(Homo sapiens (Human))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50470687(CHEMBL171707)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibitory activity for 50% on topoisomerase II isolated from Giardia lambliaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
University Of London

Curated by ChEMBL
LigandPNGBDBM50134014(CHEMBL343041 | N,N'-(9-(2-hydroxyphenylamino)acrid...)
Affinity DataEC50:  1.03E+3nMAssay Description:Inhibitory activity against human telomeraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
University Of London

Curated by ChEMBL
LigandPNGBDBM50134018(CHEMBL335819 | N,N'-(9-(4-aminophenylamino)acridin...)
Affinity DataEC50:  74nMAssay Description:Inhibitory activity against human telomeraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
University Of London

Curated by ChEMBL
LigandPNGBDBM50133998(CHEMBL137809 | N,N'-(9-(2-(methylthio)phenylamino)...)
Affinity DataEC50:  30nMAssay Description:Inhibitory activity against human telomeraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
University Of London

Curated by ChEMBL
LigandPNGBDBM50134024(CHEMBL139500 | N,N'-(9-(3-aminophenylamino)acridin...)
Affinity DataEC50:  1.09E+3nMAssay Description:Inhibitory activity against human telomeraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
University Of London

Curated by ChEMBL
LigandPNGBDBM50080849(3,6-Bis(3-pyrrolidinopropionamido)acridine | 3-PYR...)
Affinity DataEC50:  5.20E+3nMAssay Description:Inhibitory activity against human telomeraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
University Of London

Curated by ChEMBL
LigandPNGBDBM50134025(CHEMBL343795 | N,N'-(9-(4-fluorophenylamino)acridi...)
Affinity DataEC50:  70nMAssay Description:Inhibitory activity against human telomeraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
University Of London

Curated by ChEMBL
LigandPNGBDBM50134021(CHEMBL138761 | N,N'-(9-(3-(methylthio)phenylamino)...)
Affinity DataEC50:  60nMAssay Description:Inhibitory activity against human telomeraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
University Of London

Curated by ChEMBL
LigandPNGBDBM50134029(CHEMBL138369 | N,N'-(9-(phenylamino)acridine-2,7-d...)
Affinity DataEC50:  1.29E+3nMAssay Description:Inhibitory activity against human telomeraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
University Of London

Curated by ChEMBL
LigandPNGBDBM50134016(CHEMBL342921 | N,N'-(9-(3-methoxyphenylamino)acrid...)
Affinity DataEC50:  2.73E+3nMAssay Description:Inhibitory activity against human telomeraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
University Of London

Curated by ChEMBL
LigandPNGBDBM50134002(CHEMBL141540 | N,N'-(9-(2-(piperidin-1-yl)ethylami...)
Affinity DataEC50:  500nMAssay Description:Inhibitory activity against human telomeraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
University Of London

Curated by ChEMBL
LigandPNGBDBM50134028(CHEMBL142036 | N,N'-(9-(4-aminophenylamino)acridin...)
Affinity DataEC50:  200nMAssay Description:Inhibitory activity against human telomeraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
University Of London

Curated by ChEMBL
LigandPNGBDBM50134019(CHEMBL336417 | N,N'-(9-(3-aminophenylamino)acridin...)
Affinity DataEC50:  60nMAssay Description:Inhibitory activity against human telomeraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
University Of London

Curated by ChEMBL
LigandPNGBDBM50134032(CHEMBL138811 | N,N'-(9-(cyclopropylamino)acridine-...)
Affinity DataEC50:  50nMAssay Description:Inhibitory activity against human telomeraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
University Of London

Curated by ChEMBL
LigandPNGBDBM50134030(9-[4-(N,N-dimethylamino)phenylamino]-3,6-bis(3-pyr...)
Affinity DataEC50:  115nMAssay Description:Inhibitory activity against human telomeraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
University Of London

Curated by ChEMBL
LigandPNGBDBM50134031(CHEMBL137973 | N,N'-(9-(cyclohexylamino)acridine-2...)
Affinity DataEC50:  210nMAssay Description:Inhibitory activity against human telomeraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
University Of London

Curated by ChEMBL
LigandPNGBDBM50134013(CHEMBL341985 | N,N'-(9-(4-(dimethylamino)phenylami...)
Affinity DataEC50:  500nMAssay Description:Inhibitory activity against human telomeraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
University Of London

Curated by ChEMBL
LigandPNGBDBM50134022(CHEMBL336444 | N,N'-(9-(4-acetylphenylamino)acridi...)
Affinity DataEC50:  40nMAssay Description:Inhibitory activity against human telomeraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
University Of London

Curated by ChEMBL
LigandPNGBDBM50134017(CHEMBL138357 | N,N'-(9-(4-(dimethylamino)phenylami...)
Affinity DataEC50:  170nMAssay Description:Inhibitory activity against human telomeraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
University Of London

Curated by ChEMBL
LigandPNGBDBM50134026(CHEMBL138487 | N,N'-(9-(3-(dimethylamino)phenylami...)
Affinity DataEC50:  100nMAssay Description:Inhibitory activity against human telomeraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
University Of London

Curated by ChEMBL
LigandPNGBDBM50134033(CHEMBL139443 | N,N'-(9-(3-(dimethylamino)phenylami...)
Affinity DataEC50:  600nMAssay Description:Inhibitory activity against human telomeraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
University Of London

Curated by ChEMBL
LigandPNGBDBM50134015(CHEMBL44130 | N-[9-[2-(2-Amino-ethyl)-pyrrolidin-1...)
Affinity DataEC50:  18nMAssay Description:Inhibitory activity against human telomeraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
University Of London

Curated by ChEMBL
LigandPNGBDBM50134008(CHEMBL138187 | N,N'-(9-(3-(dimethylamino)propylami...)
Affinity DataEC50:  80nMAssay Description:Inhibitory activity against human telomeraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
University Of London

Curated by ChEMBL
LigandPNGBDBM50134023(CHEMBL337762 | N,N'-(9-(4-aminophenylamino)acridin...)
Affinity DataEC50:  2nMAssay Description:Inhibitory activity against human telomeraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
University Of London

Curated by ChEMBL
LigandPNGBDBM50134006(CHEMBL335564 | N,N'-(9-(2-methoxyethylamino)acridi...)
Affinity DataEC50:  140nMAssay Description:Inhibitory activity against human telomeraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
University Of London

Curated by ChEMBL
LigandPNGBDBM50134027(CHEMBL140180 | N,N'-(9-(2-(dimethylamino)ethylamin...)
Affinity DataEC50:  18nMAssay Description:Inhibitory activity against human telomeraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
University Of London

Curated by ChEMBL
LigandPNGBDBM50134020(CHEMBL141661 | N,N'-(9-(3-acetamidophenylamino)acr...)
Affinity DataEC50:  100nMAssay Description:Inhibitory activity against human telomeraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
University Of London

Curated by ChEMBL
LigandPNGBDBM50134003(CHEMBL141740 | N,N'-(9-(4-methoxyphenylamino)acrid...)
Affinity DataEC50:  460nMAssay Description:Inhibitory activity against human telomeraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
University Of London

Curated by ChEMBL
LigandPNGBDBM50134005(CHEMBL137928 | N,N'-(9-(2-(dimethylamino)ethylamin...)
Affinity DataEC50:  570nMAssay Description:Inhibitory activity against human telomeraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
University Of London

Curated by ChEMBL
LigandPNGBDBM50134001(CHEMBL140084 | N,N'-(9-(2-(dimethylamino)ethylamin...)
Affinity DataEC50:  270nMAssay Description:Inhibitory activity against human telomeraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
University Of London

Curated by ChEMBL
LigandPNGBDBM50134034(CHEMBL139687 | N-[9-[(Pyridin-3-ylmethyl)-amino]-6...)
Affinity DataEC50:  660nMAssay Description:Inhibitory activity against human telomeraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
University Of London

Curated by ChEMBL
LigandPNGBDBM50180764(2-pyrrolidin-1-yl-N-[6-(2-pyrrolidin-1-yl-acetylam...)
Affinity DataEC50:  5.20E+3nMAssay Description:Inhibition of telomerase activity from human A2780 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
University Of London

Curated by ChEMBL
LigandPNGBDBM50180765(CHEMBL381966 | N-[4-(acridin-9-ylamino)-phenyl]-3-...)
Affinity DataEC50: >2.00E+4nMAssay Description:Inhibition of telomerase activity from human A2780 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
University Of London

Curated by ChEMBL
LigandPNGBDBM50180767(3,6-bis[3-(pyrrolidin-1-yl)propionamido]-9-{4'-[2'...)
Affinity DataEC50:  167nMAssay Description:Inhibition of telomerase activity from human A2780 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
University Of London

Curated by ChEMBL
LigandPNGBDBM50134030(9-[4-(N,N-dimethylamino)phenylamino]-3,6-bis(3-pyr...)
Affinity DataEC50:  113nMAssay Description:Inhibition of telomerase activity from human A2780 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
University Of London

Curated by ChEMBL
LigandPNGBDBM50180770(3,6-bis[3-(pyrrolidin-1-yl)propionamido]-9-{4'-[3'...)
Affinity DataEC50:  67nMAssay Description:Inhibition of telomerase activity from human A2780 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
University Of London

Curated by ChEMBL
LigandPNGBDBM50180763(3,6-bis[5-(pyrrolidin-1-yl)pentanamido]-9-{4'-[3''...)
Affinity DataEC50:  255nMAssay Description:Inhibition of telomerase activity from human A2780 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
University Of London

Curated by ChEMBL
LigandPNGBDBM50180766(3,6-bis[4-(pyrrolidin-1-yl)butanamido]-9-{4'-[3''-...)
Affinity DataEC50:  326nMAssay Description:Inhibition of telomerase activity from human A2780 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
University Of London

Curated by ChEMBL
LigandPNGBDBM50180771(3,6-bis[6-(pyrrolidin-1-yl)hexanamido]-9-[4'-(N,N-...)
Affinity DataEC50:  6.91E+3nMAssay Description:Inhibition of telomerase activity from human A2780 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
University Of London

Curated by ChEMBL
LigandPNGBDBM50180768(3,6-[4-(pyrrolidin-1-yl)butanamido]-9-[4'-(N,N-dim...)
Affinity DataEC50:  99nMAssay Description:Inhibition of telomerase activity from human A2780 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
University Of London

Curated by ChEMBL
LigandPNGBDBM50180769(3,6-bis[5-(pyrrolidin-1-yl)pentanamido]-9-[4'-(N,N...)
Affinity DataEC50:  1.93E+3nMAssay Description:Inhibition of telomerase activity from human A2780 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
University Of London

Curated by ChEMBL
LigandPNGBDBM50180772(3,6-bis[3-(pyrrolidin-1-yl)propionamido]-9-{4'-[3'...)
Affinity DataEC50:  117nMAssay Description:Inhibition of telomerase activity from human A2780 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
University Of London

Curated by ChEMBL
LigandPNGBDBM50180773(3,6-bis[6-(pyrrolidin-1-yl)hexanamido]-9-{4'-[3''-...)
Affinity DataEC50:  146nMAssay Description:Inhibition of telomerase activity from human A2780 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
University Of London

Curated by ChEMBL
LigandPNGBDBM50134030(9-[4-(N,N-dimethylamino)phenylamino]-3,6-bis(3-pyr...)
Affinity DataEC50:  6.30E+3nMAssay Description:Inhibition of telomerase (unknown origin) by TRAP-LIG assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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