Compile Data Set for Download or QSAR
maximum 50k data
Found 66 with Last Name = 'wirtz' and Initial = 's'
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208974(CHEMBL390543 | N-cyclohexyl-2-(2,4-dichlorophenyl)...)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208948(2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-cyclohexyl...)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208975(1-(4-bromophenyl)-2-(2-chlorophenyl)-5-ethyl-N-((1...)
Affinity DataKi:  3.70nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50140237(1-(4-Chloro-phenyl)-2-(2,4-dichloro-phenyl)-1H-imi...)
Affinity DataKi:  3.90nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208955(2-(2-chlorophenyl)-N-cyclohexyl-1-p-tolyl-1H-imida...)
Affinity DataKi:  4.60nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208951(CHEMBL229583 | N-cyclohexyl-2-(2,4-dichlorophenyl)...)
Affinity DataKi:  4.90nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208968(2-(2-chlorophenyl)-1-(4-chlorophenyl)-5-ethyl-N-((...)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208972(2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2...)
Affinity DataKi:  5.70nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208969(2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2R)-2...)
Affinity DataKi:  6.30nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208978(2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2...)
Affinity DataKi:  6.90nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208973(1-(4-chlorophenyl)-N-cyclohexyl-2-(2,4-dimethylphe...)
Affinity DataKi:  7.20nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50123692(5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-1H-pyr...)
Affinity DataKi:  7.80nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208956(CHEMBL229584 | N-cyclohexyl-2-(2,4-dichlorophenyl)...)
Affinity DataKi:  8.20nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50107330(3-[Bis-(4-fluoro-phenyl)-methoxy]-8-(4-phenyl-buty...)
Affinity DataKi:  8.51nMAssay Description:Displacement of [3H]WIN-35 428 binding at dopamine transporter (DAT) in rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208982(2-(2-chlorophenyl)-N-cyclohexyl-1-(4-methoxyphenyl...)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208971(5-butyl-2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50107328(3-(4-Chloro-phenyl)-8-methyl-8-aza-bicyclo[3.2.1]o...)
Affinity DataKi:  14.5nMAssay Description:Displacement of [3H]WIN-35 428 binding at dopamine transporter (DAT) in rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208970(2-(2-chlorophenyl)-N-cyclohexyl-1-(4-methylcyclohe...)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208976(CHEMBL395322 | rac-2-(2-chlorophenyl)-1-(4-chlorop...)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208949(2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208979(2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1R,2S)-2...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208964(5-bromo-2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((...)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208967(2-(2-chlorophenyl)-N-cyclohexyl-1-(4-fluorophenyl)...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50107329(3-[Bis-(4-fluoro-phenyl)-methoxy]-8-[4-(4-nitro-ph...)
Affinity DataKi:  20.2nMAssay Description:Displacement of [3H]WIN-35 428 binding at dopamine transporter (DAT) in rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208961(1-(4-chlorophenyl)-N-cyclohexyl-2-o-tolyl-1H-imida...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208965(CHEMBL389198 | rac-1-(4-chlorophenyl)-2-(2,4-dichl...)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208966(CHEMBL390545 | rac-2-(2-chlorophenyl)-1-(4-chlorop...)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208954(1-(4-chlorophenyl)-N-cyclohexyl-2-(2,5-dichlorophe...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208952(2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2...)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208977(2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1S,2S)-2...)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50107327(4-(4-{3-[Bis-(4-fluoro-phenyl)-methoxy]-8-aza-bicy...)
Affinity DataKi:  29.7nMAssay Description:Displacement of [3H]WIN-35 428 binding at dopamine transporter (DAT) in rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50107325(3-(4-Chloro-phenyl)-8-[4-(4-isothiocyanato-phenyl)...)
Affinity DataKi:  31.5nMAssay Description:Displacement of [3H]WIN-35 428 binding at dopamine transporter (DAT) in rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50107334(8-[4-(4-Azido-3-iodo-phenyl)-butyl]-3-(4-chloro-ph...)
Affinity DataKi:  33nMAssay Description:Displacement of [3H]WIN-35 428 binding at dopamine transporter (DAT) in rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208947(2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-cyclohexyl...)
Affinity DataKi:  34nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208958(1-(4-chlorophenyl)-N-cyclohexyl-2-(2,4-difluorophe...)
Affinity DataKi:  36nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208960(1-(4-chlorophenyl)-N-cyclohexyl-2-(2-ethylphenyl)-...)
Affinity DataKi:  39nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208959(CHEMBL230583 | rac-2-(2-chlorophenyl)-1-(4-chlorop...)
Affinity DataKi:  41nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208984(2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1R,2R)-2...)
Affinity DataKi:  75nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208980(1-(4-chlorophenyl)-N-cyclohexyl-2-(2-methoxyphenyl...)
Affinity DataKi:  95nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208963(2-(2-chlorophenyl)-1-(4-chlorophenyl)-N-((1R,2R)-2...)
Affinity DataKi:  97nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208950(1-(4-chlorophenyl)-N-cyclohexyl-2-phenyl-1H-imidaz...)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50107332(8-[4-(4-Azido-3-iodo-phenyl)-butyl]-3-[bis-(4-fluo...)
Affinity DataKi:  159nMAssay Description:Displacement of [3H]WIN-35 428 binding at dopamine transporter (DAT) in rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50140237(1-(4-Chloro-phenyl)-2-(2,4-dichloro-phenyl)-1H-imi...)
Affinity DataKi:  240nMAssay Description:Displacement of [3H]CP559440 from human CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208953(CHEMBL229858 | N-((1S,2S)-2-aminocyclohexyl)-1-(4-...)
Affinity DataKi:  270nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50107331(8-[3-(4-Azido-3-iodo-phenyl)-propyl]-3-[bis-(4-flu...)
Affinity DataKi:  284nMAssay Description:Displacement of [3H]WIN-35 428 binding at dopamine transporter (DAT) in rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50107326(3-[Bis-(4-fluoro-phenyl)-methoxy]-8-[4-(4-isothioc...)
Affinity DataKi:  420nMAssay Description:Displacement of [3H]WIN-35 428 binding at dopamine transporter (DAT) in rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50107333(3-[Bis-(4-fluoro-phenyl)-methoxy]-8-[3-(4-isothioc...)
Affinity DataKi:  611nMAssay Description:Displacement of [3H]WIN-35 428 binding at dopamine transporter (DAT) in rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208957(1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-N-((1S,2...)
Affinity DataKi:  620nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50208962(1-(4-chlorophenyl)-2-(2,4-dichlorophenyl)-N-((1R,2...)
Affinity DataKi:  920nMAssay Description:Displacement of [3H]CP559440 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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