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Found 46 with Last Name = 'woltering' and Initial = 'm'
TargetThyroid hormone receptor alpha/beta(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50163887(CHEMBL183565 | N-[4-(1H-Indol-5-yloxy)-3,5-bis-tri...)
Affinity DataEC50:  23nMAssay Description:Agonist activity towards thyroid hormone receptor expressed in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Bayer-Schering Pharma

Curated by ChEMBL
LigandPNGBDBM28799(2-{[4-(2-{[(2,4-difluorophenyl)carbamoyl](heptyl)a...)
Affinity DataEC50:  2.00E+3nMAssay Description:Agonist activity at Gal4-fused human PPARdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha/beta(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50163889(CHEMBL182430 | N-[3-Chloro-4-(3-isopropyl-1H-indol...)
Affinity DataEC50:  8nMAssay Description:Agonist activity towards thyroid hormone receptor expressed in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha/beta(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50163890(CHEMBL183050 | N-[4-(3-Isopropyl-1H-indol-5-yloxy)...)
Affinity DataEC50:  4nMAssay Description:Agonist activity towards thyroid hormone receptor expressed in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha/beta(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50163891(CHEMBL360774 | N-{4-[3-(4-Fluoro-phenyl)-1H-indol-...)
Affinity DataEC50:  115nMAssay Description:Agonist activity towards thyroid hormone receptor expressed in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha/beta(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50163892(CHEMBL183851 | N-[3,5-Dimethyl-4-(3-pentyl-1H-inda...)
Affinity DataEC50:  8nMAssay Description:Agonist activity towards thyroid hormone receptor expressed in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha/beta(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50163893(CHEMBL183057 | N-[3,5-Dimethyl-4-(3-methyl-1H-indo...)
Affinity DataEC50:  15nMAssay Description:Agonist activity towards thyroid hormone receptor expressed in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha/beta(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50163895((S)-2-Amino-3-[4-(4-hydroxy-3-iodo-phenoxy)-3-iodo...)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity towards thyroid hormone receptor expressed in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha/beta(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50163894(CHEMBL183863 | N-{4-[3-(4-Fluoro-benzyl)-1H-indol-...)
Affinity DataEC50:  11nMAssay Description:Agonist activity towards thyroid hormone receptor expressed in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha/beta(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50163896(CHEMBL183000 | N-[4-(3-Isopropyl-1H-indol-5-yloxy)...)
Affinity DataEC50:  7.80nMAssay Description:Agonist activity towards thyroid hormone receptor expressed in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha/beta(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50163898(CHEMBL359647 | N-[3-Chloro-4-(3-isopropyl-1H-indol...)
Affinity DataEC50:  4nMAssay Description:Agonist activity towards thyroid hormone receptor expressed in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha/beta(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50163897(3-[4-(3-Isopropyl-1H-indol-5-yloxy)-3,5-bis-triflu...)
Affinity DataEC50:  2.60nMAssay Description:Agonist activity towards thyroid hormone receptor expressed in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha/beta(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50163902(CHEMBL183727 | N-[3,5-Dichloro-4-(1H-indol-5-yloxy...)
Affinity DataEC50:  15nMAssay Description:Agonist activity towards thyroid hormone receptor expressed in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha/beta(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50163899(CHEMBL183122 | N-[3,5-Dichloro-4-(3-isopropyl-1H-i...)
Affinity DataEC50:  4nMAssay Description:Agonist activity towards thyroid hormone receptor expressed in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha/beta(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50163900((E)-3-[4-(3-Isopropyl-1H-indol-5-yloxy)-3,5-bis-tr...)
Affinity DataEC50:  3.20nMAssay Description:Agonist activity towards thyroid hormone receptor expressed in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha/beta(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50163901(CHEMBL360137 | N-[3,5-Dibromo-4-(3-isopropyl-1H-in...)
Affinity DataEC50:  1.20nMAssay Description:Agonist activity towards thyroid hormone receptor expressed in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha/beta(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50163904(CHEMBL180952 | N-[4-(3-Isopropyl-1H-indol-5-ylmeth...)
Affinity DataEC50:  18nMAssay Description:Agonist activity towards thyroid hormone receptor expressed in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha/beta(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50163905(CHEMBL183829 | N-[4-(1H-Indol-5-yloxy)-3,5-dimethy...)
Affinity DataEC50:  72nMAssay Description:Agonist activity towards thyroid hormone receptor expressed in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha/beta(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50163903(CHEMBL180819 | N-{4-[3-(4-Fluoro-phenoxy)-1H-indol...)
Affinity DataEC50:  495nMAssay Description:Agonist activity towards thyroid hormone receptor expressed in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha/beta(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50163906(CHEMBL361162 | [4-(3-Isopropyl-1H-indol-5-yloxy)-3...)
Affinity DataEC50:  0.5nMAssay Description:Agonist activity towards thyroid hormone receptor expressed in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Bayer-Schering Pharma

Curated by ChEMBL
LigandPNGBDBM50319262(2-(4-(((2-(2,4-dimethylphenylamino)-2-oxoethyl)(fu...)
Affinity DataEC50:  6.00E+3nMAssay Description:Agonist activity at Gal4-fused human PPARdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Mus musculus)
Bayer-Schering Pharma

Curated by ChEMBL
LigandPNGBDBM28799(2-{[4-(2-{[(2,4-difluorophenyl)carbamoyl](heptyl)a...)
Affinity DataEC50:  10nMAssay Description:Agonist activity at Gal4-fused mouse PPARalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Mus musculus)
Bayer-Schering Pharma

Curated by ChEMBL
LigandPNGBDBM50319262(2-(4-(((2-(2,4-dimethylphenylamino)-2-oxoethyl)(fu...)
Affinity DataEC50:  20nMAssay Description:Agonist activity at Gal4-fused mouse PPARalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Bayer-Schering Pharma

Curated by ChEMBL
LigandPNGBDBM28799(2-{[4-(2-{[(2,4-difluorophenyl)carbamoyl](heptyl)a...)
Affinity DataEC50:  2.50E+3nMAssay Description:Agonist activity at Gal4-fused mouse PPARgammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Bayer-Schering Pharma

Curated by ChEMBL
LigandPNGBDBM50319262(2-(4-(((2-(2,4-dimethylphenylamino)-2-oxoethyl)(fu...)
Affinity DataEC50:  300nMAssay Description:Agonist activity at Gal4-fused mouse PPARgammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Bayer-Schering Pharma

Curated by ChEMBL
LigandPNGBDBM28799(2-{[4-(2-{[(2,4-difluorophenyl)carbamoyl](heptyl)a...)
Affinity DataEC50:  2.00E+3nMAssay Description:Agonist activity at Gal4-fused mouse PPARdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Bayer-Schering Pharma

Curated by ChEMBL
LigandPNGBDBM50319262(2-(4-(((2-(2,4-dimethylphenylamino)-2-oxoethyl)(fu...)
Affinity DataEC50:  2.00E+3nMAssay Description:Agonist activity at Gal4-fused mouse PPARdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer-Schering Pharma

Curated by ChEMBL
LigandPNGBDBM50319262(2-(4-(((2-(2,4-dimethylphenylamino)-2-oxoethyl)(fu...)
Affinity DataEC50:  20nMAssay Description:Agonist activity at Gal4-fused human PPARalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer-Schering Pharma

Curated by ChEMBL
LigandPNGBDBM50319263(2-(4-((benzyl(2-(2,4-dimethylphenylamino)-2-oxoeth...)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at Gal4-fused human PPARalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer-Schering Pharma

Curated by ChEMBL
LigandPNGBDBM50319264(2-(4-(((2-(2,4-dimethylphenylamino)-2-oxoethyl)(th...)
Affinity DataEC50:  700nMAssay Description:Agonist activity at Gal4-fused human PPARalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer-Schering Pharma

Curated by ChEMBL
LigandPNGBDBM50319265(2-(4-(((2-(2,4-dimethylphenylamino)-2-oxoethyl)(4-...)
Affinity DataEC50:  900nMAssay Description:Agonist activity at Gal4-fused human PPARalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer-Schering Pharma

Curated by ChEMBL
LigandPNGBDBM50319266(2-(4-(((2-(2,4-dimethylphenylamino)-2-oxoethyl)(pr...)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at Gal4-fused human PPARalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer-Schering Pharma

Curated by ChEMBL
LigandPNGBDBM50319267(2-(4-((butyl(2-(2,4-dimethylphenylamino)-2-oxoethy...)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at Gal4-fused human PPARalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer-Schering Pharma

Curated by ChEMBL
LigandPNGBDBM50319268(2-(4-(((2-(2,4-dimethylphenylamino)-2-oxoethyl)(he...)
Affinity DataEC50: >2.50E+4nMAssay Description:Agonist activity at Gal4-fused human PPARalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer-Schering Pharma

Curated by ChEMBL
LigandPNGBDBM50319269(2-(4-(((furan-2-ylmethyl)(2-oxo-2-(o-tolylamino)et...)
Affinity DataEC50:  2.00E+3nMAssay Description:Agonist activity at Gal4-fused human PPARalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer-Schering Pharma

Curated by ChEMBL
LigandPNGBDBM50319270(2-(4-(((2-(2,5-dimethylphenylamino)-2-oxoethyl)(fu...)
Affinity DataEC50:  600nMAssay Description:Agonist activity at Gal4-fused human PPARalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer-Schering Pharma

Curated by ChEMBL
LigandPNGBDBM50319271(2-(4-(((2-(2,5-dimethoxyphenylamino)-2-oxoethyl)(f...)
Affinity DataEC50:  300nMAssay Description:Agonist activity at Gal4-fused human PPARalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer-Schering Pharma

Curated by ChEMBL
LigandPNGBDBM50319272(2-(4-(((furan-2-ylmethyl)(2-(3-methoxyphenylamino)...)
Affinity DataEC50:  3.00E+3nMAssay Description:Agonist activity at Gal4-fused human PPARalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer-Schering Pharma

Curated by ChEMBL
LigandPNGBDBM50319273(2-(4-(((2-(2,4-difluorophenylamino)-2-oxoethyl)(fu...)
Affinity DataEC50:  1.50E+3nMAssay Description:Agonist activity at Gal4-fused human PPARalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer-Schering Pharma

Curated by ChEMBL
LigandPNGBDBM50319274(2-(4-(((furan-2-ylmethyl)(2-oxo-2-(pyridin-2-ylami...)
Affinity DataEC50: >2.50E+4nMAssay Description:Agonist activity at Gal4-fused human PPARalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer-Schering Pharma

Curated by ChEMBL
LigandPNGBDBM50319275(2-(4-(((2-(benzylamino)-2-oxoethyl)(furan-2-ylmeth...)
Affinity DataEC50:  1.30E+4nMAssay Description:Agonist activity at Gal4-fused human PPARalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer-Schering Pharma

Curated by ChEMBL
LigandPNGBDBM50319276(2-(4-(((2-(2-chlorobenzylamino)-2-oxoethyl)(furan-...)
Affinity DataEC50:  7.00E+3nMAssay Description:Agonist activity at Gal4-fused human PPARalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Bayer-Schering Pharma

Curated by ChEMBL
LigandPNGBDBM28799(2-{[4-(2-{[(2,4-difluorophenyl)carbamoyl](heptyl)a...)
Affinity DataEC50:  100nMAssay Description:Agonist activity at Gal4-fused human PPARalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bayer-Schering Pharma

Curated by ChEMBL
LigandPNGBDBM28799(2-{[4-(2-{[(2,4-difluorophenyl)carbamoyl](heptyl)a...)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at Gal4-fused human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Bayer-Schering Pharma

Curated by ChEMBL
LigandPNGBDBM50319262(2-(4-(((2-(2,4-dimethylphenylamino)-2-oxoethyl)(fu...)
Affinity DataEC50:  800nMAssay Description:Agonist activity at Gal4-fused human PPARgammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha/beta(Homo sapiens (Human))
Bayer Healthcare

Curated by ChEMBL
LigandPNGBDBM50163888(CHEMBL183176 | N-[4-(3-Isopropyl-1H-indol-5-yloxy)...)
Affinity DataEC50:  3nMAssay Description:Agonist activity towards thyroid hormone receptor expressed in human HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed