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Found 81 with Last Name = 'wong' and Initial = 'ak'
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50086880(Proteolytic Enzyme inhibitor)
Affinity DataKi:  1nMAssay Description:binding affinity towards HIV-1 Protease enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50086884((R)-N*4*-Hydroxy-2-isobutyl-N*1*-((S)-9-oxo-1,8-di...)
Affinity DataKi:  1nMAssay Description:binding affinity towards HIV-1 Protease enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50369797(CHEMBL1794029)
Affinity DataKi:  3nMAssay Description:binding affinity towards HIV-1 Protease enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50369799(CHEMBL1794024)
Affinity DataKi:  4nMAssay Description:binding affinity towards HIV-1 Protease enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50086886(CHEMBL436149 | N-[14-Benzyl-18-(3-guanidino-propyl...)
Affinity DataKi:  10nMAssay Description:binding affinity towards HIV-1 Protease enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50086883(2-{2-[2-(8-Carbamoylmethyl-6,9-dioxo-2-oxa-7,10-di...)
Affinity DataKi:  12nMAssay Description:binding affinity towards HIV-1 Protease enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50369800(CHEMBL1232357)
Affinity DataKi:  800nMAssay Description:binding affinity towards HIV-1 Protease enzymeMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50369798(CHEMBL1794028)
Affinity DataKi:  6.00E+4nMAssay Description:binding affinity towards HIV-1 Protease enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50066481((S)-2-Acetylamino-N-[(5S,11R,14S,17R,19aS)-17-cycl...)
Affinity DataIC50:  12nMAssay Description:50% reduction in myeloperoxidase secretion from human PMNs mediated by 100 nM C5aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50077479((S)-2-Amino-N-[(5S,11S,14S,17R,19aS)-17-cyclohexyl...)
Affinity DataIC50: >56.2nMAssay Description:Inhibition of binding of [125I]C5a to human polymorphonuclear leukocyte C5a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50077479((S)-2-Amino-N-[(5S,11S,14S,17R,19aS)-17-cyclohexyl...)
Affinity DataIC50:  60nMAssay Description:Inhibition of binding of [125I]-C5a to human polymorphonuclear leukocyte C5a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50066483((S)-2-Acetylamino-N-[(5S,12S,15S,18R,20aS)-18-cycl...)
Affinity DataIC50:  90nMAssay Description:50% reduction in myeloperoxidase secretion from human PMNs mediated by 100 nM C5aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50077493(CHEMBL2373542 | H-Lys-Tyr-Lys-His-Ser-Val-Val-Lys-...)
Affinity DataIC50: >174nMAssay Description:Inhibition of binding of [125I]C5a to human polymorphonuclear leukocyte C5a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50077493(CHEMBL2373542 | H-Lys-Tyr-Lys-His-Ser-Val-Val-Lys-...)
Affinity DataIC50: >174nMAssay Description:Inhibition of binding of [125I]C5a to human polymorphonuclear leukocyte C5a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50077485((S)-2-Acetylamino-N-[(5S,11S,14S,17R,19aS)-17-cycl...)
Affinity DataIC50: >269nMAssay Description:Inhibition of binding of [125I]C5a to human polymorphonuclear leukocyte C5a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50077485((S)-2-Acetylamino-N-[(5S,11S,14S,17R,19aS)-17-cycl...)
Affinity DataIC50: >269nMAssay Description:Inhibition of binding of [125I]C5a to human polymorphonuclear leukocyte C5a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50066481((S)-2-Acetylamino-N-[(5S,11R,14S,17R,19aS)-17-cycl...)
Affinity DataIC50:  280nMAssay Description:50% reduction in binding of [125I]-C5a to human polymorphonuclear cells (PMNs)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50077499((S)-2-Amino-N-[(5S,12S,15S,18R,20aS)-18-cyclohexyl...)
Affinity DataIC50:  300nMAssay Description:Inhibition of binding of [125I]-C5a to human polymorphonuclear leukocyte C5a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50077487((S)-2-Amino-N-[(5S,10S,13S,16R,18aS)-16-cyclohexyl...)
Affinity DataIC50: >309nMAssay Description:Inhibition of binding of [125I]C5a to human polymorphonuclear leukocyte C5a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50077487((S)-2-Amino-N-[(5S,10S,13S,16R,18aS)-16-cyclohexyl...)
Affinity DataIC50: >309nMAssay Description:Inhibition of binding of [125I]C5a to human polymorphonuclear leukocyte C5a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50077499((S)-2-Amino-N-[(5S,12S,15S,18R,20aS)-18-cyclohexyl...)
Affinity DataIC50: >331nMAssay Description:Inhibition of binding of [125I]C5a to human polymorphonuclear leukocyte C5a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50066478((S)-1-[(S)-6-Amino-2-((S)-2-methylamino-3-phenyl-p...)
Affinity DataIC50:  500nMAssay Description:50% reduction in myeloperoxidase secretion from human PMNs mediated by 100 nM C5aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50066479((S)-2-[(S)-2-[(R)-2-({(S)-1-[(S)-6-Amino-2-((S)-2-...)
Affinity DataIC50:  700nMAssay Description:50% reduction in myeloperoxidase secretion from human PMNs mediated by 100 nM C5aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50077504((R)-2-[(S)-2-[(R)-2-({(R)-1-[(S)-2-((S)-2-Acetylam...)
Affinity DataIC50:  794nMAssay Description:Inhibition of binding of [125I]C5a to human polymorphonuclear leukocyte C5a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50077497((R)-2-[(S)-2-[(R)-2-({(R)-1-[(S)-2-((S)-2-Acetylam...)
Affinity DataIC50:  800nMAssay Description:Inhibition of binding of [125I]-C5a to human polymorphonuclear leukocyte C5a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50077502(CHEMBL2373550 | H-Lys-Tyr-Lys-His-Ser-Val-Val-Lys-...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of binding of [125I]-C5a to human polymorphonuclear leukocyte C5a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50077502(CHEMBL2373550 | H-Lys-Tyr-Lys-His-Ser-Val-Val-Lys-...)
Affinity DataIC50:  1.23E+3nMAssay Description:Inhibition of binding of [125I]C5a to human polymorphonuclear leukocyte C5a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50066482((S)-2-[(S)-2-[(S)-2-({(S)-1-[(S)-6-Amino-2-((S)-2-...)
Affinity DataIC50:  1.80E+3nMAssay Description:50% reduction in binding of [125I]-C5a to human polymorphonuclear cells (PMNs)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50077482((R)-2-[(S)-2-[(R)-2-({(R)-1-[(S)-6-Amino-2-((S)-2-...)
Affinity DataIC50:  1.95E+3nMAssay Description:Inhibition of binding of [125I]C5a to human polymorphonuclear leukocyte C5a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50077486((R)-2-[(S)-2-[(R)-2-({(R)-1-[(S)-6-Amino-2-((S)-2-...)
Affinity DataIC50:  1.95E+3nMAssay Description:Inhibition of binding of [125I]C5a to human polymorphonuclear leukocyte C5a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50077482((R)-2-[(S)-2-[(R)-2-({(R)-1-[(S)-6-Amino-2-((S)-2-...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of binding of [125I]C5a to human polymorphonuclear leukocyte C5a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50077486((R)-2-[(S)-2-[(R)-2-({(R)-1-[(S)-6-Amino-2-((S)-2-...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of binding of [125I]C5a to human polymorphonuclear leukocyte C5a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50077500((R)-2-[(S)-2-[(R)-2-({(R)-1-[(S)-2-((S)-2-Acetylam...)
Affinity DataIC50:  2.63E+3nMAssay Description:Inhibition of binding of [125I]C5a to human polymorphonuclear leukocyte C5a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50077483((R)-2-[(S)-2-{(R)-2-[((R)-1-{(S)-6-Amino-2-[(S)-2-...)
Affinity DataIC50:  2.63E+3nMAssay Description:Inhibition of binding of [125I]C5a to human polymorphonuclear leukocyte C5a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50077489(CHEMBL410692 | N-{3-[(5S,8S,11R,14S,17R,19aS)-8-Be...)
Affinity DataIC50:  2.95E+3nMAssay Description:Inhibition of binding of [125I]C5a to human polymorphonuclear leukocyte C5a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50077489(CHEMBL410692 | N-{3-[(5S,8S,11R,14S,17R,19aS)-8-Be...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of binding of [125I]-C5a to human polymorphonuclear leukocyte C5a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50077481((R)-2-[(S)-2-[(R)-2-({(R)-1-[(R)-2-((S)-2-Acetylam...)
Affinity DataIC50:  3.02E+3nMAssay Description:Inhibition of binding of [125I]C5a to human polymorphonuclear leukocyte C5a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50077481((R)-2-[(S)-2-[(R)-2-({(R)-1-[(R)-2-((S)-2-Acetylam...)
Affinity DataIC50:  3.02E+3nMAssay Description:Inhibition of binding of [125I]C5a to human polymorphonuclear leukocyte C5a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50077490((S)-2-Amino-N-[(5S,11R,14S,17R,19aS)-17-cyclohexyl...)
Affinity DataIC50:  3.09E+3nMAssay Description:Inhibition of binding of [125I]C5a to human polymorphonuclear leukocyte C5a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50077490((S)-2-Amino-N-[(5S,11R,14S,17R,19aS)-17-cyclohexyl...)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of binding of [125I]-C5a to human polymorphonuclear leukocyte C5a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50066483((S)-2-Acetylamino-N-[(5S,12S,15S,18R,20aS)-18-cycl...)
Affinity DataIC50:  3.20E+3nMAssay Description:50% reduction in binding of [125I]-C5a to human polymorphonuclear cells (PMNs)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50077480((S)-2-Acetylamino-N-[(5S,12R,15S,18R,20aS)-18-cycl...)
Affinity DataIC50:  3.24E+3nMAssay Description:Inhibition of binding of [125I]C5a to human polymorphonuclear leukocyte C5a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50077480((S)-2-Acetylamino-N-[(5S,12R,15S,18R,20aS)-18-cycl...)
Affinity DataIC50:  3.24E+3nMAssay Description:Inhibition of binding of [125I]C5a to human polymorphonuclear leukocyte C5a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50077497((R)-2-[(S)-2-[(R)-2-({(R)-1-[(S)-2-((S)-2-Acetylam...)
Affinity DataIC50:  3.55E+3nMAssay Description:Inhibition of binding of [125I]C5a to human polymorphonuclear leukocyte C5a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50077504((R)-2-[(S)-2-[(R)-2-({(R)-1-[(S)-2-((S)-2-Acetylam...)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of binding of [125I]-C5a to human polymorphonuclear leukocyte C5a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50077503((S)-2-Amino-N-[(5S,10R,13S,16R,18aS)-16-cyclohexyl...)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibition of binding of [125I]C5a to human polymorphonuclear leukocyte C5a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50077503((S)-2-Amino-N-[(5S,10R,13S,16R,18aS)-16-cyclohexyl...)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibition of binding of [125I]C5a to human polymorphonuclear leukocyte C5a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50077496(2-[2-(2-{[1-(6-Amino-2-{2-[6-amino-2-(2-amino-3-ph...)
Affinity DataIC50:  4.57E+3nMAssay Description:Inhibition of binding of [125I]C5a to human polymorphonuclear leukocyte C5a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50077495((R)-2-[(S)-2-[(R)-2-({(R)-1-[(S)-6-Amino-2-((S)-2-...)
Affinity DataIC50:  4.57E+3nMAssay Description:Inhibition of binding of [125I]C5a to human polymorphonuclear leukocyte C5a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Homo sapiens (Human))
University Of Queensland

Curated by ChEMBL
LigandPNGBDBM50077495((R)-2-[(S)-2-[(R)-2-({(R)-1-[(S)-6-Amino-2-((S)-2-...)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibition of binding of [125I]-C5a to human polymorphonuclear leukocyte C5a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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