Compile Data Set for Download or QSAR
maximum 50k data
Found 187 with Last Name = 'wong' and Initial = 'sc'
TargetDisintegrin and metalloproteinase domain-containing protein 17 [215-477,S266A,N452Q](Homo sapiens (Human))
Schering-Plough Research Institute

LigandPNGBDBM26526((2R)-N-hydroxy-2-[(3S)-3-methyl-3-{4-[(2-methylqui...)
Affinity DataKi:  0.0600nM ΔG°:  -57.8kJ/molepH: 7.3 T: 2°CAssay Description:Enzyme activity was determined by a kinetic assay measuring the rate of increase in fluorescent intensity generated by the cleavage of an internally ...More data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17 [215-477,S266A,N452Q](Homo sapiens (Human))
Schering-Plough Research Institute

LigandPNGBDBM26524((1R,2S)-1-({3-fluoro-4-[(2-phenylquinolin-4-yl)met...)
Affinity DataKi:  0.140nM ΔG°:  -55.7kJ/molepH: 7.3 T: 2°CAssay Description:Enzyme activity was determined by a kinetic assay measuring the rate of increase in fluorescent intensity generated by the cleavage of an internally ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17 [215-477,S266A,N452Q](Homo sapiens (Human))
Schering-Plough Research Institute

LigandPNGBDBM26525((1S,2R)-1-N-hydroxy-2-({4-[(2-phenylquinolin-4-yl)...)
Affinity DataKi:  0.180nM ΔG°:  -55.1kJ/molepH: 7.3 T: 2°CAssay Description:Enzyme activity was determined by a kinetic assay measuring the rate of increase in fluorescent intensity generated by the cleavage of an internally ...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211619((S)-N-(1-(4-(4-ethoxy-2-(2-fluorophenylsulfonyl)ph...)
Affinity DataKi:  0.900nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50108281(CHEMBL32197 | N-{3-(3,4-Dichloro-phenyl)-5-(4-hydr...)
Affinity DataKi:  1nMAssay Description:Tested for binding affinity against neurokinin 1 (NK1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50108271(CHEMBL32124 | N-{3-(3,4-Dichloro-phenyl)-5-(4-hydr...)
Affinity DataKi:  1nMAssay Description:Binding affinity test against Neurokinin 2 (NK2) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50108260(1-(5-tert-Butyl-[1,2,4]oxadiazol-3-ylmethoxy)-3-(3...)
Affinity DataKi:  1nMAssay Description:Binding affinity test against Neurokinin 2 (NK2) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211617((S)-trifluoro-N-(1-(4-(2-(2-fluorophenylsulfonyl)-...)
Affinity DataKi:  1.10nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50172158((S)-N-(1-(4-(4-chloro-2-(2-fluorophenylsulfonyl)ph...)
Affinity DataKi:  1.30nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211632((S)-trifluoro-N-(1-(4-(2-(2-fluorophenylsulfonyl)-...)
Affinity DataKi:  1.30nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211636((S)-N-(1-(4-(4-cyclopropyl-2-(2-fluorophenylsulfon...)
Affinity DataKi:  1.40nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50108242(CHEMBL286646 | N-{3-(3,4-Dichloro-phenyl)-5-(4-hyd...)
Affinity DataKi:  2nMAssay Description:Tested for binding affinity against neurokinin 1 (NK1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50108271(CHEMBL32124 | N-{3-(3,4-Dichloro-phenyl)-5-(4-hydr...)
Affinity DataKi:  2nMAssay Description:Tested for binding affinity against neurokinin 1 (NK1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50108272(CHEMBL33249 | N-{3-(3,4-Dichloro-phenyl)-5-(4-hydr...)
Affinity DataKi:  2nMAssay Description:Binding affinity test against Neurokinin 2 (NK2) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50108267(CHEMBL32537 | N-{3-(3,4-Dichloro-phenyl)-5-(4-hydr...)
Affinity DataKi:  2nMAssay Description:Binding affinity test against Neurokinin 2 (NK2) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50108281(CHEMBL32197 | N-{3-(3,4-Dichloro-phenyl)-5-(4-hydr...)
Affinity DataKi:  2nMAssay Description:Binding affinity test against Neurokinin 2 (NK2) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50108272(CHEMBL33249 | N-{3-(3,4-Dichloro-phenyl)-5-(4-hydr...)
Affinity DataKi:  2nMAssay Description:Tested for binding affinity against neurokinin 1 (NK1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50108256(CHEMBL33243 | N-{3-(3,4-Dichloro-phenyl)-5-(4-hydr...)
Affinity DataKi:  2nMAssay Description:Tested for binding affinity against neurokinin 1 (NK1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50108238(3,5-Dichloro-N-{3-(3,4-dichloro-phenyl)-5-(4-hydro...)
Affinity DataKi:  2nMAssay Description:Tested for binding affinity against neurokinin 1 (NK1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50108240(5-Methyl-thiophene-2-carboxylic acid {3-(3,4-dichl...)
Affinity DataKi:  2nMAssay Description:Binding affinity test against Neurokinin 2 (NK2) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211605((S)-N-(1-(4-(4-chloro-2-(2-fluorophenylsulfonyl)ph...)
Affinity DataKi:  2nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211627((S)-trifluoro-N-(1-(4-(2-(2-fluorophenylsulfonyl)-...)
Affinity DataKi:  2.5nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211629((S)-trifluoro-N-(1-(4-(2-(2-fluorophenylsulfonyl)-...)
Affinity DataKi:  2.5nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211610((S)-N-(1-(4-(4-chloro-2-(pyridin-2-ylsulfonyl)phen...)
Affinity DataKi:  2.90nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50108256(CHEMBL33243 | N-{3-(3,4-Dichloro-phenyl)-5-(4-hydr...)
Affinity DataKi:  3nMAssay Description:Binding affinity test against Neurokinin 2 (NK2) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50108265(CHEMBL36462 | N-{3-(3,4-Dichloro-phenyl)-5-(4-hydr...)
Affinity DataKi:  3nMAssay Description:Binding affinity test against Neurokinin 2 (NK2) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50112009(1-(2,6-Dichloro-pyridin-4-yl)-3-[4-(1H-imidazol-4-...)
Affinity DataKi:  3nMAssay Description:Compound was evaluated for its binding affinity against Histamine H3 receptor of guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17 [215-477,S266A,N452Q](Homo sapiens (Human))
Schering-Plough Research Institute

LigandPNGBDBM23487((1S,2R)-1-N-hydroxy-2-({4-[(2-methylquinolin-4-yl)...)
Affinity DataKi:  3nM ΔG°:  -48.2kJ/molepH: 7.3 T: 2°CAssay Description:Enzyme activity was determined by a kinetic assay measuring the rate of increase in fluorescent intensity generated by the cleavage of an internally ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211604((S)-N-(1-(4-(4-chloro-2-(pyridin-2-ylsulfonyl)phen...)
Affinity DataKi:  3.60nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211628((S)-N-(1-(4-(4-chloro-2-(2-fluorophenylsulfonyl)ph...)
Affinity DataKi:  3.70nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM86188(CHEMBL366977 | SCH 79687)
Affinity DataKi:  4nMAssay Description:Compound was evaluated for its binding affinity against Histamine H3 receptor of guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50108251(CHEMBL32309 | N-{3-(3,4-Dichloro-phenyl)-5-(4-hydr...)
Affinity DataKi:  4nMAssay Description:Tested for binding affinity against neurokinin 1 (NK1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50108237(CHEMBL418224 | N-{3-(3,4-Dichloro-phenyl)-5-(4-hyd...)
Affinity DataKi:  4nMAssay Description:Binding affinity test against Neurokinin 2 (NK2) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50108238(3,5-Dichloro-N-{3-(3,4-dichloro-phenyl)-5-(4-hydro...)
Affinity DataKi:  4nMAssay Description:Binding affinity test against Neurokinin 2 (NK2) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50108248(1-(4-tert-Butyl-benzyloxy)-3-(3,4-dichloro-phenyl)...)
Affinity DataKi:  4nMAssay Description:Binding affinity test against Neurokinin 2 (NK2) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50108245(5-Bromo-N-{3-(3,4-dichloro-phenyl)-5-(4-hydroxy-4-...)
Affinity DataKi:  4nMAssay Description:Binding affinity test against Neurokinin 2 (NK2) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211609((S)-N-(1-(4-(2-(2-amino-6-fluorophenylsulfonyl)-4-...)
Affinity DataKi:  4.10nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211616((S)-N-(1-(4-(4-(cyclopropylamino)-2-(2-fluoropheny...)
Affinity DataKi:  4.90nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211620((S)-trifluoro-N-(1-(4-(2-(2-fluorophenylsulfonyl)-...)
Affinity DataKi:  5nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50108262(4-Bromo-N-{3-(3,4-dichloro-phenyl)-5-(4-hydroxy-4-...)
Affinity DataKi:  5nMAssay Description:Tested for binding affinity against neurokinin 1 (NK1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50108267(CHEMBL32537 | N-{3-(3,4-Dichloro-phenyl)-5-(4-hydr...)
Affinity DataKi:  5nMAssay Description:Tested for binding affinity against neurokinin 1 (NK1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50108249(3-(3,5-Bis-trifluoromethyl-phenyl)-1-{3-(3,4-dichl...)
Affinity DataKi:  5nMAssay Description:Tested for binding affinity against neurokinin 1 (NK1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50112024(1-(3-Cyano-phenyl)-3-[4-(1H-imidazol-4-ylmethyl)-b...)
Affinity DataKi:  5nMAssay Description:Compound was evaluated for its binding affinity against Histamine H3 receptor of guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50112025((3,5-Dichloro-phenyl)-carbamic acid 4-(1H-imidazol...)
Affinity DataKi:  5nMAssay Description:Compound was evaluated for its binding affinity against Histamine H3 receptor of guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50211623((S)-N-(1-(4-(4-chloro-2-(2,6-difluorophenylsulfony...)
Affinity DataKi:  5.80nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
The Schering Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50112012(1-(3-Chloro-phenyl)-3-[4-(1H-imidazol-4-ylmethyl)-...)
Affinity DataKi:  6nMAssay Description:Compound was evaluated for its binding affinity against Histamine H3 receptor of guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50108270(3-(3,4-Dichloro-phenyl)-5-(4-hydroxy-4-phenyl-pipe...)
Affinity DataKi:  6nMAssay Description:Tested for binding affinity against neurokinin 1 (NK1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50108242(CHEMBL286646 | N-{3-(3,4-Dichloro-phenyl)-5-(4-hyd...)
Affinity DataKi:  6nMAssay Description:Binding affinity test against Neurokinin 2 (NK2) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50108278(1-(3,5-Dichloro-benzyloxy)-3-(3,4-dichloro-phenyl)...)
Affinity DataKi:  6nMAssay Description:Binding affinity test against Neurokinin 2 (NK2) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50108258(CHEMBL285986 | {3-(3,4-Dichloro-phenyl)-5-(4-hydro...)
Affinity DataKi:  6nMAssay Description:Tested for binding affinity against neurokinin 1 (NK1) receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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