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Found 217 with Last Name = 'woodward' and Initial = 'df'
TargetProstaglandin F2-alpha receptor(Homo sapiens (Human))
Albert Einstein College of Medicine

Curated by PDSP Ki Database
LigandPNGBDBM85339(17-PHENYL TRINOR PGF2ALPHA-IPR | CAS_130209-76-6 |...)
Affinity DataKi:  18nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 2A1(Homo sapiens (Human))
Albert Einstein College of Medicine

Curated by PDSP Ki Database
LigandPNGBDBM85720(AGN 194394)
Affinity DataKi:  34nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 2A1(Homo sapiens (Human))
Albert Einstein College of Medicine

Curated by PDSP Ki Database
LigandPNGBDBM50020300((S-isomer)7-[3,5-Dihydroxy-2-(3-hydroxy-oct-1-enyl...)
Affinity DataKi:  45nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(Homo sapiens (Human))
Albert Einstein College of Medicine

Curated by PDSP Ki Database
LigandPNGBDBM50020300((S-isomer)7-[3,5-Dihydroxy-2-(3-hydroxy-oct-1-enyl...)
Affinity DataKi:  48nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 2A1(Homo sapiens (Human))
Albert Einstein College of Medicine

Curated by PDSP Ki Database
LigandPNGBDBM85718(AGN 191366)
Affinity DataKi:  71nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 2A1(Homo sapiens (Human))
Albert Einstein College of Medicine

Curated by PDSP Ki Database
LigandPNGBDBM85339(17-PHENYL TRINOR PGF2ALPHA-IPR | CAS_130209-76-6 |...)
Affinity DataKi:  168nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(Homo sapiens (Human))
Albert Einstein College of Medicine

Curated by PDSP Ki Database
LigandPNGBDBM85716(AGN 191995)
Affinity DataKi:  228nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 2A1(Homo sapiens (Human))
Albert Einstein College of Medicine

Curated by PDSP Ki Database
LigandPNGBDBM85715(AGN 191365)
Affinity DataKi:  307nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(Homo sapiens (Human))
Albert Einstein College of Medicine

Curated by PDSP Ki Database
LigandPNGBDBM85719(PGF2 Alpha, 1-isopropyl ester)
Affinity DataKi:  3.20E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 2A1(Homo sapiens (Human))
Albert Einstein College of Medicine

Curated by PDSP Ki Database
LigandPNGBDBM85719(PGF2 Alpha, 1-isopropyl ester)
Affinity DataKi:  5.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 2A1(Homo sapiens (Human))
Albert Einstein College of Medicine

Curated by PDSP Ki Database
LigandPNGBDBM85714(AGN 190911)
Affinity DataKi:  7.30E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(Homo sapiens (Human))
Albert Einstein College of Medicine

Curated by PDSP Ki Database
LigandPNGBDBM85718(AGN 191366)
Affinity DataKi:  8.13E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 2A1(Homo sapiens (Human))
Albert Einstein College of Medicine

Curated by PDSP Ki Database
LigandPNGBDBM85717(AGN 192151)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(Homo sapiens (Human))
Albert Einstein College of Medicine

Curated by PDSP Ki Database
LigandPNGBDBM85714(AGN 190911)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 2A1(Homo sapiens (Human))
Albert Einstein College of Medicine

Curated by PDSP Ki Database
LigandPNGBDBM85716(AGN 191995)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(Homo sapiens (Human))
Albert Einstein College of Medicine

Curated by PDSP Ki Database
LigandPNGBDBM85720(AGN 194394)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier organic anion transporter family member 2A1(Homo sapiens (Human))
Albert Einstein College of Medicine

Curated by PDSP Ki Database
LigandPNGBDBM85721(AGN 191088)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(Homo sapiens (Human))
Albert Einstein College of Medicine

Curated by PDSP Ki Database
LigandPNGBDBM85721(AGN 191088)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(Homo sapiens (Human))
Albert Einstein College of Medicine

Curated by PDSP Ki Database
LigandPNGBDBM85717(AGN 192151)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin F2-alpha receptor(Homo sapiens (Human))
Albert Einstein College of Medicine

Curated by PDSP Ki Database
LigandPNGBDBM85715(AGN 191365)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50133817(4-(3-Chloro-pyridin-2-yl)-piperazine-1-carboxylic ...)
Affinity DataIC50:  6.70nMAssay Description:Antagonist activity at human TRPV1 expressed in HEK293 cells assessed as decrease in intracellular calcium levelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM22999(N-[2-(5-hydroxy-1H-indol-3-yl)ethyl]-2-(3-pentylph...)
Affinity DataIC50:  240nMAssay Description:The antagonistic effects of test compounds were evaluated using HEK293 cells stably overexpressing human TRPV1. Experiments were carried out by measu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50312085(4-tert-butylphenyl 4-(3-(trifluoromethyl)pyridin-2...)
Affinity DataIC50:  260nMAssay Description:Antagonist activity at human TRPV1 expressed in HEK293 cells assessed as decrease in intracellular calcium levelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM22987((5Z,8Z,11Z,14Z)-N-[2-(5-hydroxy-1H-indol-3-yl)ethy...)
Affinity DataIC50:  270nMAssay Description:The antagonistic effects of test compounds were evaluated using HEK293 cells stably overexpressing human TRPV1. Experiments were carried out by measu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50312091(CHEMBL1081905 | biphenyl-3-yl 4-(3-(trifluoromethy...)
Affinity DataIC50:  380nMAssay Description:Inhibition of FAAH-mediated hydrolysis of [3H]AEA in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM23000(JMC506554 Compound 1m | N-[2-(5-hydroxy-1H-indol-3...)
Affinity DataIC50:  430nMAssay Description:The antagonistic effects of test compounds were evaluated using HEK293 cells stably overexpressing human TRPV1. Experiments were carried out by measu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM22989((9Z,12Z,15Z)-N-[2-(5-hydroxy-1H-indol-3-yl)ethyl]o...)
Affinity DataIC50:  470nMAssay Description:The antagonistic effects of test compounds were evaluated using HEK293 cells stably overexpressing human TRPV1. Experiments were carried out by measu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50312078(4-tert-butylphenyl 4-(3-chloropyridin-2-yl)piperaz...)
Affinity DataIC50:  480nMAssay Description:Antagonist activity at human TRPV1 expressed in HEK293 cells assessed as decrease in intracellular calcium levelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM26741(N-phenyl-4-(quinolin-2-ylmethyl)piperazine-1-carbo...)
Affinity DataIC50:  500nMAssay Description:Inhibition of FAAH-mediated hydrolysis of [3H]AEA in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM23015(3-phenylphenyl N-[2-(5-hydroxy-1H-indol-3-yl)ethyl...)
Affinity DataIC50:  500nMpH: 9.0 T: 2°CAssay Description:The effect of the test compounds on the enzymatic hydrolysis of [14C]anandamide was evaluated by using membranes prepared from rat brain. [14C]Ethano...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50312088(3-(trifluoromethyl)phenyl 4-(3-(trifluoromethyl)py...)
Affinity DataIC50:  610nMAssay Description:Inhibition of FAAH-mediated hydrolysis of [3H]AEA in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM22998(N-[2-(5-hydroxy-1H-indol-3-yl)ethyl]-9-phenylnonan...)
Affinity DataIC50:  680nMAssay Description:The antagonistic effects of test compounds were evaluated using HEK293 cells stably overexpressing human TRPV1. Experiments were carried out by measu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM23007(3-[2-(5-hydroxy-1H-indol-3-yl)ethyl]-1-(3-phenylph...)
Affinity DataIC50:  720nMAssay Description:The antagonistic effects of test compounds were evaluated using HEK293 cells stably overexpressing human TRPV1. Experiments were carried out by measu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM22995(N-[2-(5-hydroxy-1H-indol-3-yl)ethyl]dodecanamide |...)
Affinity DataIC50:  740nMAssay Description:The antagonistic effects of test compounds were evaluated using HEK293 cells stably overexpressing human TRPV1. Experiments were carried out by measu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50312090(3-chlorophenyl 4-(3-(trifluoromethyl)pyridin-2-yl)...)
Affinity DataIC50:  740nMAssay Description:Inhibition of FAAH-mediated hydrolysis of [3H]AEA in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50312084(CHEMBL1079442 | biphenyl-3-yl 4-(3-chloropyridin-2...)
Affinity DataIC50:  750nMAssay Description:Inhibition of FAAH-mediated hydrolysis of [3H]AEA in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM22994(N-[2-(5-hydroxy-1H-indol-3-yl)ethyl]undecanamide |...)
Affinity DataIC50:  760nMAssay Description:The antagonistic effects of test compounds were evaluated using HEK293 cells stably overexpressing human TRPV1. Experiments were carried out by measu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50312086(3-tert-butylphenyl 4-(3-(trifluoromethyl)pyridin-2...)
Affinity DataIC50:  770nMAssay Description:Inhibition of FAAH-mediated hydrolysis of [3H]AEA in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50312083(3-chlorophenyl 4-(3-chloropyridin-2-yl)piperazine-...)
Affinity DataIC50:  910nMAssay Description:Inhibition of FAAH-mediated hydrolysis of [3H]AEA in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM22990((6Z,9Z,12Z)-N-[2-(5-hydroxy-1H-indol-3-yl)ethyl]oc...)
Affinity DataIC50:  950nMAssay Description:The antagonistic effects of test compounds were evaluated using HEK293 cells stably overexpressing human TRPV1. Experiments were carried out by measu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50312087(4-(trifluoromethyl)phenyl 4-(3-(trifluoromethyl)py...)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity at human TRPV1 expressed in HEK293 cells assessed as decrease in intracellular calcium levelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM23026(4-(benzyloxy)phenyl N-[2-(5-hydroxy-1H-indol-3-yl)...)
Affinity DataIC50:  1.17E+3nMAssay Description:The effect of the test compounds on the enzymatic hydrolysis of [14C]anandamide was evaluated by using membranes prepared from rat brain. [14C]Ethano...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50312079(1-(4-(3-(3-tert-butylphenyl)prop-1-en-2-yl)cyclohe...)
Affinity DataIC50:  1.27E+3nMAssay Description:Inhibition of FAAH-mediated hydrolysis of [3H]AEA in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM23022(3-iodophenyl N-[2-(5-hydroxy-1H-indol-3-yl)ethyl]c...)
Affinity DataIC50:  1.80E+3nMAssay Description:The effect of the test compounds on the enzymatic hydrolysis of [14C]anandamide was evaluated by using membranes prepared from rat brain. [14C]Ethano...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM22991((9Z,12Z)-N-[2-(5-hydroxy-1H-indol-3-yl)ethyl]octad...)
Affinity DataIC50:  1.82E+3nMAssay Description:The antagonistic effects of test compounds were evaluated using HEK293 cells stably overexpressing human TRPV1. Experiments were carried out by measu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM23020(3-chlorophenyl N-[2-(5-hydroxy-1H-indol-3-yl)ethyl...)
Affinity DataIC50:  1.90E+3nMAssay Description:The effect of the test compounds on the enzymatic hydrolysis of [14C]anandamide was evaluated by using membranes prepared from rat brain. [14C]Ethano...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM22997(N-[2-(5-hydroxy-1H-indol-3-yl)ethyl]-8-phenyloctan...)
Affinity DataIC50:  2.13E+3nMAssay Description:The antagonistic effects of test compounds were evaluated using HEK293 cells stably overexpressing human TRPV1. Experiments were carried out by measu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50312089(4-chlorophenyl 4-(3-(trifluoromethyl)pyridin-2-yl)...)
Affinity DataIC50:  2.19E+3nMAssay Description:Inhibition of FAAH-mediated hydrolysis of [3H]AEA in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM23018(3-(trifluoromethyl)phenyl N-[2-(5-hydroxy-1H-indol...)
Affinity DataIC50:  2.20E+3nMAssay Description:The effect of the test compounds on the enzymatic hydrolysis of [14C]anandamide was evaluated by using membranes prepared from rat brain. [14C]Ethano...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM23014(3-pentylphenyl N-[2-(5-hydroxy-1H-indol-3-yl)ethyl...)
Affinity DataIC50:  2.40E+3nMAssay Description:The antagonistic effects of test compounds were evaluated using HEK293 cells stably overexpressing human TRPV1. Experiments were carried out by measu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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