Affinity DataIC50: 78.2nMAssay Description:Inhibition of peptidase activity of CPP32More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Harbor Branch Oceanographic Institution
Curated by ChEMBL
Harbor Branch Oceanographic Institution
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of Cdc2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 480nMAssay Description:Binding affinity against Purinergic receptor P2Y12 using [3H]-2-methylthio-ADP as radioligandMore data for this Ligand-Target Pair
TargetNitric oxide synthase, inducible(Mus musculus (mouse))
Harbor Branch Oceanographic Institution
Curated by ChEMBL
Harbor Branch Oceanographic Institution
Curated by ChEMBL
Affinity DataIC50: 723nMAssay Description:Inhibition of iNOS-mediated NO production in LPS-stimulated mouse RAW264.7 cells by Griess methodMore data for this Ligand-Target Pair
Affinity DataIC50: 775nMAssay Description:Inhibition of CPP32 peptidase activityMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+3nMAssay Description:Binding affinity against Purinergic receptor P2Y12 using [3H]-2-methylthio-ADP as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 2.35E+3nMAssay Description:Inhibition of peptidase activity of CPP32More data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Florida Atlantic University
Curated by ChEMBL
Florida Atlantic University
Curated by ChEMBL
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of MCL1 binding to Bak by FRET assayMore data for this Ligand-Target Pair
TargetSodium channel protein type 10 subunit alpha(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by ChEMBL
Schering-Plough Research Institute
Curated by ChEMBL
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of sodium channel NaV1.8 expressed in rat ND7/23 cells by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.09E+4nMAssay Description:Inhibition of human HDAC1 assessed as [3H]acetate release after 90 mins by scintillation countingMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Harbor Branch Oceanographic Institution
Curated by ChEMBL
Harbor Branch Oceanographic Institution
Curated by ChEMBL
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of Cdc2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+4nMAssay Description:Displacement of [125I]thrombin from thrombin receptor in human platelet membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 2.58E+4nMAssay Description:Inhibition of peptidase activity of CPP32More data for this Ligand-Target Pair
Affinity DataIC50: 3.90E+4nMAssay Description:Displacement of [125]ET1 from ETA receptor in pig thoracic aortaMore data for this Ligand-Target Pair
TargetLeukotriene B4 receptor 1(Homo sapiens (Human))
Harbor Branch Oceanographic Institution
Curated by ChEMBL
Harbor Branch Oceanographic Institution
Curated by ChEMBL
Affinity DataIC50: 4.45E+4nMAssay Description:Displacement of [3H]LTB4 from LTB4 receptor in human neutrophilsMore data for this Ligand-Target Pair