Compile Data Set for Download or QSAR
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Found 923 with Last Name = 'wright' and Initial = 'sd'
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50377735(CHEMBL257779)
Affinity DataIC50:  0.980nMAssay Description:Inhibition of human 11beta-HSD1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50377747(CHEMBL258388)
Affinity DataIC50:  0.980nMAssay Description:Inhibition of human 11beta-HSD1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50377736(CHEMBL403898)
Affinity DataIC50:  0.980nMAssay Description:Inhibition of human 11beta-HSD1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50377756(CHEMBL256298)
Affinity DataIC50:  1nMAssay Description:Inhibition of human 11beta-HSD1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Merck

Curated by ChEMBL
LigandPNGBDBM50377736(CHEMBL403898)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of mouse 11beta-HSD1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Merck

Curated by ChEMBL
LigandPNGBDBM50377735(CHEMBL257779)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of mouse 11beta-HSD1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50377746(CHEMBL403811)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of human 11beta-HSD1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50377712(CHEMBL401909)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of human 11beta-HSD1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50377730(CHEMBL257601)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of human 11beta-HSD1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Merck

Curated by ChEMBL
LigandPNGBDBM50377724(CHEMBL401883)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of mouse 11beta-HSD1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50377724(CHEMBL401883)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of human 11beta-HSD1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179830((S)-2-(4-(3-(2-chloro-4-cyclohexylphenoxy)propoxy)...)
Affinity DataIC50:  2nMAssay Description:Binding affinity to human PPAR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50377750(CHEMBL401908)
Affinity DataIC50:  2nMAssay Description:Inhibition of human 11beta-HSD1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Merck

Curated by ChEMBL
LigandPNGBDBM50377730(CHEMBL257601)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of mouse 11beta-HSD1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50377725(CHEMBL401884)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of human 11beta-HSD1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Merck

Curated by ChEMBL
LigandPNGBDBM50377725(CHEMBL401884)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of mouse 11beta-HSD1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50377757(CHEMBL256986)
Affinity DataIC50:  2.60nMAssay Description:Inhibition of human 11beta-HSD1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50377728(CHEMBL401975)
Affinity DataIC50:  2.70nMAssay Description:Inhibition of human 11beta-HSD1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Merck

Curated by ChEMBL
LigandPNGBDBM50377732(CHEMBL257752)
Affinity DataIC50:  2.80nMAssay Description:Inhibition of mouse 11beta-HSD1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Merck

Curated by ChEMBL
LigandPNGBDBM50377722(CHEMBL401988)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of mouse 11beta-HSD1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50377726(CHEMBL257129)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of human 11beta-HSD1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50377749(CHEMBL258389)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of human 11beta-HSD1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179833((S)-2-(4-(3-(2-chloro-4-(trifluoromethyl)phenoxy)p...)
Affinity DataIC50:  3nMAssay Description:Binding affinity to human PPAR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179824((S)-2-(4-(3-(2-chloro-4-(trifluoromethoxy)phenoxy)...)
Affinity DataIC50:  3nMAssay Description:Binding affinity to human PPAR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50377751(CHEMBL256158)
Affinity DataIC50:  3.10nMAssay Description:Inhibition of human 11beta-HSD1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50377745(CHEMBL402737)
Affinity DataIC50:  3.60nMAssay Description:Inhibition of human 11beta-HSD1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50377737(CHEMBL257963)
Affinity DataIC50:  3.90nMAssay Description:Inhibition of human 11beta-HSD1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50377732(CHEMBL257752)
Affinity DataIC50:  4.30nMAssay Description:Inhibition of human 11beta-HSD1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Merck

Curated by ChEMBL
LigandPNGBDBM50377712(CHEMBL401909)
Affinity DataIC50:  4.5nMAssay Description:Inhibition of mouse 11beta-HSD1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50377723(CHEMBL401830)
Affinity DataIC50:  4.60nMAssay Description:Inhibition of human 11beta-HSD1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179818(2-(4-(3-(2-chloro-4-(4-fluorophenoxy)phenoxy)propo...)
Affinity DataIC50:  5nMAssay Description:Binding affinity to human PPAR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50377722(CHEMBL401988)
Affinity DataIC50:  5.20nMAssay Description:Inhibition of human 11beta-HSD1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50377755(CHEMBL404638)
Affinity DataIC50:  5.80nMAssay Description:Inhibition of human 11beta-HSD1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179826((R)-2-(4-(3-(2-chloro-4-(4-fluorophenoxy)phenoxy)p...)
Affinity DataIC50:  6nMAssay Description:Binding affinity to human PPAR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Merck

Curated by ChEMBL
LigandPNGBDBM50377716(CHEMBL404743)
Affinity DataIC50:  6.40nMAssay Description:Inhibition of mouse 11beta-HSD1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Merck

Curated by ChEMBL
LigandPNGBDBM50377737(CHEMBL257963)
Affinity DataIC50:  6.60nMAssay Description:Inhibition of mouse 11beta-HSD1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Rattus norvegicus)
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393161(CHEMBL2153439)
Affinity DataIC50:  7nMAssay Description:Antagonist activity at rat GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-induc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuccinate receptor 1(Homo sapiens (Human))
Advinus Therapeutics

Curated by ChEMBL
LigandPNGBDBM50393129(CHEMBL2153461)
Affinity DataIC50:  7nMAssay Description:Antagonist activity at human GPR91 receptor expressed in CHO-K1 cells co-expressing Galpha and Gqi5 G-protein assessed as inhibition of succinate-ind...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50168554((R)-7-{3-[2-Chloro-4-(1,1-dimethyl-propyl)-phenoxy...)
Affinity DataIC50:  7nMAssay Description:In vitro binding affinity against human PPARalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Merck

Curated by ChEMBL
LigandPNGBDBM50377747(CHEMBL258388)
Affinity DataIC50:  7.10nMAssay Description:Inhibition of mouse 11beta-HSD1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50377721(CHEMBL428951)
Affinity DataIC50:  7.70nMAssay Description:Inhibition of human 11beta-HSD1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Merck

Curated by ChEMBL
LigandPNGBDBM50377756(CHEMBL256298)
Affinity DataIC50:  8nMAssay Description:Inhibition of mouse 11beta-HSD1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Merck

Curated by ChEMBL
LigandPNGBDBM50377714(CHEMBL254993)
Affinity DataIC50:  8.40nMAssay Description:Inhibition of mouse 11beta-HSD1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Merck

Curated by ChEMBL
LigandPNGBDBM50377751(CHEMBL256158)
Affinity DataIC50:  8.60nMAssay Description:Inhibition of mouse 11beta-HSD1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50377729(CHEMBL403758)
Affinity DataIC50:  9nMAssay Description:Inhibition of human 11beta-HSD1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Merck

Curated by ChEMBL
LigandPNGBDBM50377726(CHEMBL257129)
Affinity DataIC50:  9.80nMAssay Description:Inhibition of mouse 11beta-HSD1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Merck

Curated by ChEMBL
LigandPNGBDBM50377729(CHEMBL403758)
Affinity DataIC50:  10nMAssay Description:Inhibition of mouse 11beta-HSD1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50179836((S)-2-(4-(3-(2-chloro-4-(2,2,2-trifluoroethoxy)phe...)
Affinity DataIC50:  10nMAssay Description:Binding affinity to human PPAR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Merck

Curated by ChEMBL
LigandPNGBDBM50377721(CHEMBL428951)
Affinity DataIC50:  10nMAssay Description:Inhibition of mouse 11beta-HSD1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Merck

Curated by ChEMBL
LigandPNGBDBM50377746(CHEMBL403811)
Affinity DataIC50:  11nMAssay Description:Inhibition of mouse 11beta-HSD1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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