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Found 76 with Last Name = 'wu' and Initial = 'mt'
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50280908(1-[3-chlorophenyl(phenyl)carbamoyl]-4-dipentylcarb...)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of Angiotensin II receptor, type 2 in rat midbrain using [125I]-Sar1,Ile8 angiotensin II binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50000040(((2S,3S)-2-Benzhydryl-1-aza-bicyclo[2.2.2]oct-3-yl...)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of [125I]-Substance P binding to human NK1 receptors in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50280914(1-[(3-Bromo-phenyl)-phenyl-carbamoyl]-4-dipentylca...)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of Angiotensin II receptor, type 2 in rat midbrain using [125I]-Sar1,Ile8 angiotensin II binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50280913(4-Dipentylcarbamoyl-1-(phenyl-m-tolyl-carbamoyl)-p...)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of Angiotensin II receptor, type 2 in rat midbrain using [125I]-Sar1,Ile8 angiotensin II binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50280924(4-dipentylcarbamoyl-1-(2,2-diphenylacetyl)hexahydr...)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of Angiotensin II receptor, type 2 in rat midbrain using [125I]-Sar1,Ile8 angiotensin II binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50280912((S)-4-Dipentylcarbamoyl-1-diphenylcarbamoyl-pipera...)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of Angiotensin II receptor, type 2 in rat midbrain using [125I]-Sar1,Ile8 angiotensin II binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50280907((S)-1,4-Bis-diphenylcarbamoyl-piperazine-2-carboxy...)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of Angiotensin II receptor, type 2 in rat midbrain using [125I]-Sar1,Ile8 angiotensin II binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50280912((S)-4-Dipentylcarbamoyl-1-diphenylcarbamoyl-pipera...)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of Angiotensin II receptor, type 2 in rat midbrain using [125I]-Sar1,Ile8 angiotensin II binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50280910(1-[(4-Bromo-phenyl)-phenyl-carbamoyl]-4-dipentylca...)
Affinity DataIC50:  2.70nMAssay Description:Inhibition of Angiotensin II receptor, type 2 in rat midbrain using [125I]-Sar1,Ile8 angiotensin II binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50280921((R)-4-Dipentylcarbamoyl-1-diphenylcarbamoyl-pipera...)
Affinity DataIC50:  4.5nMAssay Description:Inhibition of Angiotensin II receptor, type 2 in rat midbrain using [125I]-Sar1,Ile8 angiotensin II binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50280922(4-Dipentylcarbamoyl-1-[(4-iodo-phenyl)-phenyl-carb...)
Affinity DataIC50:  7nMAssay Description:Inhibition of Angiotensin II receptor, type 2 in rat midbrain using [125I]-Sar1,Ile8 angiotensin II binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50280925(4-Dipentylcarbamoyl-1-[(3-methoxy-phenyl)-phenyl-c...)
Affinity DataIC50:  7.80nMAssay Description:Inhibition of Angiotensin II receptor, type 2 in rat midbrain using [125I]-Sar1,Ile8 angiotensin II binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281196((S)-Piperazine-1,2,4-tricarboxylic acid 4-dipentyl...)
Affinity DataIC50:  9nMAssay Description:Inhibition of [125I]-Substance P binding to human NK1 receptors in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281189((S)-Piperazine-1,2,4-tricarboxylic acid 4-dipentyl...)
Affinity DataIC50:  9nMAssay Description:Inhibition of [125I]-Substance P binding to human NK1 receptors in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50280919(2,5-Dimethyl-piperazine-1,4-dicarboxylic acid bis-...)
Affinity DataIC50:  10nMAssay Description:Inhibition of Angiotensin II receptor, type 2 in rat midbrain using [125I]-Sar1,Ile8 angiotensin II binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281194((S)-Piperazine-1,2,4-tricarboxylic acid 2-[(2-diet...)
Affinity DataIC50:  11nMAssay Description:Inhibition of [125I]-Substance P binding to human NK1 receptors in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50280927(CHEMBL292939 | methyl 4-dipentylcarbamoyl-1-diphen...)
Affinity DataIC50:  12nMAssay Description:Inhibition of Angiotensin II receptor, type 2 in rat midbrain using [125I]-Sar1,Ile8 angiotensin II binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50280911(1-diphenylcarbamoyl-4-methyl(pentyl)carbamoyl-(2S)...)
Affinity DataIC50:  15nMAssay Description:Inhibition of Angiotensin II receptor, type 2 in rat midbrain using [125I]-Sar1,Ile8 angiotensin II binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50280916(1N,1N,4N,4N-tetraphenyl-2-methylhexahydro-1,4-pyra...)
Affinity DataIC50:  15nMAssay Description:Inhibition of Angiotensin II receptor, type 2 in rat midbrain using [125I]-Sar1,Ile8 angiotensin II binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50280909(4N,4N-dipentyl-1N,1N-diphenyl-2-(2-hydroxyethyl)-(...)
Affinity DataIC50:  15nMAssay Description:Inhibition of Angiotensin II receptor, type 2 in rat midbrain using [125I]-Sar1,Ile8 angiotensin II binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281198((S)-Piperazine-1,2,4-tricarboxylic acid 4-dipentyl...)
Affinity DataIC50:  17nMAssay Description:Inhibition of [125I]-Substance P binding to human NK1 receptors in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50280918(4-diphenylcarbamoyl-1-pentyl(phenyl)carbamoyl-(2S)...)
Affinity DataIC50:  20nMAssay Description:Inhibition of Angiotensin II receptor, type 2 in rat midbrain using [125I]-Sar1,Ile8 angiotensin II binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50280928(1-dipentylcarbamoyl-4-diphenylcarbamoyl-(2S)-hexah...)
Affinity DataIC50:  23nMAssay Description:Inhibition of Angiotensin II receptor, type 2 in rat midbrain using [125I]-Sar1,Ile8 angiotensin II binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50280905((S)-2-Hydroxymethyl-piperazine-1,4-dicarboxylic ac...)
Affinity DataIC50:  30nMAssay Description:Inhibition of Angiotensin II receptor, type 2 in rat midbrain using [125I]-Sar1,Ile8 angiotensin II binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50280929(4-Dipentylcarbamoyl-1-[(4-ethoxycarbonyl-phenyl)-p...)
Affinity DataIC50:  35nMAssay Description:Inhibition of Angiotensin II receptor, type 2 in rat midbrain using [125I]-Sar1,Ile8 angiotensin II binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50280906(1N,1N,4N,4N-tetraphenylhexahydro-1,4-pyrazinedicar...)
Affinity DataIC50:  37nMAssay Description:Inhibition of Angiotensin II receptor, type 2 in rat midbrain using [125I]-Sar1,Ile8 angiotensin II binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50010359((S)-5-Diphenylacetyl-1-(4-methoxy-3-methyl-benzyl)...)
Affinity DataIC50:  38nMAssay Description:Compound was evaluated for inhibition of Angiotensin II receptor, type 2 in rat midbrain AT2 assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50280926(4-diisopropylcarbamoyl-1-diphenylcarbamoyl-(2S)-he...)
Affinity DataIC50:  40nMAssay Description:Inhibition of Angiotensin II receptor, type 2 in rat midbrain using [125I]-Sar1,Ile8 angiotensin II binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281187((S)-Piperazine-1,2,4-tricarboxylic acid 2-[(3-diet...)
Affinity DataIC50:  41nMAssay Description:Inhibition of [125I]-Substance P binding to human NK1 receptors in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281200((S)-Piperazine-1,2,4-tricarboxylic acid 2-[(2-dime...)
Affinity DataIC50:  55nMAssay Description:Inhibition of [125I]-Substance P binding to human NK1 receptors in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281201((S)-Piperazine-1,2,4-tricarboxylic acid 2-[(2-amin...)
Affinity DataIC50:  57nMAssay Description:Inhibition of [125I]-Substance P binding to human NK1 receptors in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50280915(1N,1N-dipentyl-4N,4N-diphenylhexahydro-1,4-pyrazin...)
Affinity DataIC50:  70nMAssay Description:Inhibition of Angiotensin II receptor, type 2 in rat midbrain using [125I]-Sar1,Ile8 angiotensin II binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50280920(1,4-di(dipentylcarbamoyl)-(2S)-hexahydro-2-pyrazin...)
Affinity DataIC50:  82nMAssay Description:Inhibition of Angiotensin II receptor, type 2 in rat midbrain using [125I]-Sar1,Ile8 angiotensin II binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280912((S)-4-Dipentylcarbamoyl-1-diphenylcarbamoyl-pipera...)
Affinity DataIC50:  130nMAssay Description:Inhibition of [125I]-Substance P binding to human NK1 receptors in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281192((S)-Piperazine-1,2,4-tricarboxylic acid 2-[(2-acet...)
Affinity DataIC50:  140nMAssay Description:Inhibition of [125I]-Substance P binding to human NK1 receptors in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50280917(1-diphenylcarbamoyl-4-methyl(phenyl)carbamoyl-(2S)...)
Affinity DataIC50:  170nMAssay Description:Inhibition of Angiotensin II receptor, type 2 in rat midbrain using [125I]-Sar1,Ile8 angiotensin II binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50280923(1-[(4-Carboxy-phenyl)-phenyl-carbamoyl]-4-dipentyl...)
Affinity DataIC50:  180nMAssay Description:Inhibition of Angiotensin II receptor, type 2 in rat midbrain using [125I]-Sar1,Ile8 angiotensin II binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50010361((S)-1-(4-Amino-3-methyl-benzyl)-5-diphenylacetyl-4...)
Affinity DataIC50:  190nMAssay Description:Compound was evaluated for inhibition of Angiotensin II receptor, type 2 in rat midbrain AT2 assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281193((S)-Piperazine-1,2,4-tricarboxylic acid 2-({2-[(3,...)
Affinity DataIC50:  200nMAssay Description:Inhibition of [125I]-Substance P binding to human NK1 receptors in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281191((S)-Piperazine-1,2,4-tricarboxylic acid 2-[(2-diis...)
Affinity DataIC50:  217nMAssay Description:Inhibition of [125I]-Substance P binding to human NK1 receptors in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50280930(4-Dipentylcarbamoyl-1-[(4-hydroxy-phenyl)-phenyl-c...)
Affinity DataIC50:  230nMAssay Description:Inhibition of Angiotensin II receptor, type 2 in rat midbrain using [125I]-Sar1,Ile8 angiotensin II binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281188((S)-Piperazine-1,2,4-tricarboxylic acid 4-dipentyl...)
Affinity DataIC50:  267nMAssay Description:Inhibition of [125I]-Substance P binding to human NK1 receptors in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280905((S)-2-Hydroxymethyl-piperazine-1,4-dicarboxylic ac...)
Affinity DataIC50:  280nMAssay Description:Inhibition of [125I]-Substance P binding to human NK1 receptors in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281199((S)-Piperazine-1,2,4-tricarboxylic acid 2-{[2-(ben...)
Affinity DataIC50:  290nMAssay Description:Inhibition of [125I]-Substance P binding to human NK1 receptors in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280915(1N,1N-dipentyl-4N,4N-diphenylhexahydro-1,4-pyrazin...)
Affinity DataIC50:  500nMAssay Description:Inhibition of [125I]-Substance P binding to human NK1 receptors in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281195(CHEMBL90035 | [((S)-4-Dipentylcarbamoyl-1-diphenyl...)
Affinity DataIC50:  597nMAssay Description:Inhibition of [125I]-Substance P binding to human NK1 receptors in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281190((S)-Piperazine-1,2,4-tricarboxylic acid 2-[(2-dime...)
Affinity DataIC50:  930nMAssay Description:Inhibition of [125I]-Substance P binding to human NK1 receptors in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50281197((S)-Piperazine-1,2,4-tricarboxylic acid 2-({2-[(3,...)
Affinity DataIC50:  1.08E+3nMAssay Description:Inhibition of [125I]-Substance P binding to human NK1 receptors in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50280923(1-[(4-Carboxy-phenyl)-phenyl-carbamoyl]-4-dipentyl...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of angiotensin Angiotensin II receptor, type 1 in rabbit aorta using [125I-Sar1,Ile8] angiotensin II binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280921((R)-4-Dipentylcarbamoyl-1-diphenylcarbamoyl-pipera...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of [125I]-Substance P binding to human NK1 receptors in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
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