Compile Data Set for Download or QSAR
maximum 50k data
Found 78 with Last Name = 'da cunha' and Initial = 'ef'
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481036(CHEMBL568589)
Affinity DataIC50:  0.302nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481029(CHEMBL569671)
Affinity DataIC50:  0.302nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481028(CHEMBL566620)
Affinity DataIC50:  0.302nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481018(CHEMBL568883)
Affinity DataIC50:  0.302nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481014(CHEMBL568951)
Affinity DataIC50:  0.339nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481023(CHEMBL566849)
Affinity DataIC50:  0.398nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481020(CHEMBL565964)
Affinity DataIC50:  0.398nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481040(CHEMBL566842)
Affinity DataIC50:  0.501nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Universidade Federal De Lavras-Ufla

Curated by ChEMBL
LigandPNGBDBM50111902(2-(2-ethoxy-5-(4-methylpiperazin-1-ylsulfonyl)phen...)
Affinity DataIC50:  0.603nMAssay Description:Inhibition of PDE5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Universidade Federal De Lavras-Ufla

Curated by ChEMBL
LigandPNGBDBM14776(2-{2-ethoxy-5-[(4-ethylpiperazine-1-)sulfonyl]phen...)
Affinity DataIC50:  0.708nMAssay Description:Inhibition of PDE5More data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481024(CHEMBL566902)
Affinity DataIC50:  0.741nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481015(CHEMBL568832)
Affinity DataIC50:  0.794nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481017(CHEMBL568840)
Affinity DataIC50:  0.794nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481025(CHEMBL567444)
Affinity DataIC50:  0.851nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481033(CHEMBL565528)
Affinity DataIC50:  0.891nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481035(CHEMBL569670)
Affinity DataIC50:  1nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481037(CHEMBL569236)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481032(CHEMBL569569)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481022(CHEMBL568365)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Universidade Federal De Lavras-Ufla

Curated by ChEMBL
LigandPNGBDBM50287550(5-(2-ethoxy-5-(4-(2-hydroxyethyl)piperazin-1-ylsul...)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of PDE5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM586099(BDBM50064200 | TL-3)
Affinity DataIC50:  2nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Universidade Federal De Lavras-Ufla

Curated by ChEMBL
LigandPNGBDBM50412319(CHEMBL457207)
Affinity DataIC50:  2.10nMAssay Description:Inhibition of PDE5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481019(CHEMBL571731)
Affinity DataIC50:  2.20nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481031(CHEMBL567043)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Universidade Federal De Lavras-Ufla

Curated by ChEMBL
LigandPNGBDBM50412324(CHEMBL509728)
Affinity DataIC50:  3nMAssay Description:Inhibition of PDE5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481041(CHEMBL569673)
Affinity DataIC50:  3.20nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Universidade Federal De Lavras-Ufla

Curated by ChEMBL
LigandPNGBDBM50412327(CHEMBL456142)
Affinity DataIC50:  4nMAssay Description:Inhibition of PDE5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481038(CHEMBL568977)
Affinity DataIC50:  4nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481016(CHEMBL568817)
Affinity DataIC50:  4nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Universidade Federal De Lavras-Ufla

Curated by ChEMBL
LigandPNGBDBM14777((2R,8R)-2-(2H-1,3-benzodioxol-5-yl)-6-methyl-3,6,1...)
Affinity DataIC50:  5nMAssay Description:Inhibition of PDE5More data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Universidade Federal De Lavras-Ufla

Curated by ChEMBL
LigandPNGBDBM50111897(2-(2-Ethoxy-phenyl)-3,5-dimethyl-7-propyl-3H-imida...)
Affinity DataIC50:  5nMAssay Description:Inhibition of PDE5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Universidade Federal De Lavras-Ufla

Curated by ChEMBL
LigandPNGBDBM50134099((3aR,10S)-2-Butyl-10-(4-methoxy-phenyl)-3a,4,9,10-...)
Affinity DataIC50:  5nMAssay Description:Inhibition of PDE5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Universidade Federal De Lavras-Ufla

Curated by ChEMBL
LigandPNGBDBM50287543(5-(2-ethoxy-5-(piperazin-1-ylsulfonyl)phenyl)-1-me...)
Affinity DataIC50:  5.80nMAssay Description:Inhibition of PDE5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Universidade Federal De Lavras-Ufla

Curated by ChEMBL
LigandPNGBDBM50412321(CHEMBL456577)
Affinity DataIC50:  6nMAssay Description:Inhibition of PDE5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Universidade Federal De Lavras-Ufla

Curated by ChEMBL
LigandPNGBDBM14390(5-[2-ethoxy-5-(4-methyl-1-piperazinylsulfonyl)phen...)
Affinity DataIC50:  6.60nMAssay Description:Inhibition of PDE5More data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Universidade Federal De Lavras-Ufla

Curated by ChEMBL
LigandPNGBDBM50412325(CHEMBL458714)
Affinity DataIC50:  7.10nMAssay Description:Inhibition of PDE5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Universidade Federal De Lavras-Ufla

Curated by ChEMBL
LigandPNGBDBM50412328(CHEMBL508321)
Affinity DataIC50:  7.10nMAssay Description:Inhibition of PDE5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Universidade Federal De Lavras-Ufla

Curated by ChEMBL
LigandPNGBDBM50134093((3aR,10R)-2-Butyl-10-(4-methoxy-phenyl)-3a,4,9,10-...)
Affinity DataIC50:  7.90nMAssay Description:Inhibition of PDE5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Universidade Federal De Lavras-Ufla

Curated by ChEMBL
LigandPNGBDBM50412329(CHEMBL515979)
Affinity DataIC50:  10nMAssay Description:Inhibition of PDE5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Universidade Federal De Lavras-Ufla

Curated by ChEMBL
LigandPNGBDBM50412330(CHEMBL456552)
Affinity DataIC50:  10nMAssay Description:Inhibition of PDE5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Universidade Federal De Lavras-Ufla

Curated by ChEMBL
LigandPNGBDBM50111901(2-(5-(4-methylpiperazin-1-ylsulfonyl)-2-propoxyphe...)
Affinity DataIC50:  10nMAssay Description:Inhibition of PDE5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Universidade Federal De Lavras-Ufla

Curated by ChEMBL
LigandPNGBDBM50111898(2-(2-Propoxy-phenyl)-9-propyl-1,9-dihydro-purin-6-...)
Affinity DataIC50:  10nMAssay Description:Inhibition of PDE5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM198((2S)-N-[(2S,3S,4S,5S)-3,4-dihydroxy-5-[(2S)-3-meth...)
Affinity DataIC50:  15nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Universidade Federal De Lavras-Ufla

Curated by ChEMBL
LigandPNGBDBM50412326(CHEMBL458713)
Affinity DataIC50:  18nMAssay Description:Inhibition of PDE5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481027(CHEMBL566839)
Affinity DataIC50:  18nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Universidade Federal De Lavras-Ufla

Curated by ChEMBL
LigandPNGBDBM50412331(CHEMBL456548)
Affinity DataIC50:  20nMAssay Description:Inhibition of PDE5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Universidade Federal De Lavras-Ufla

Curated by ChEMBL
LigandPNGBDBM50134094((3aR,10S)-2-Butyl-10-phenyl-3a,4,9,10-tetrahydro-2...)
Affinity DataIC50:  20nMAssay Description:Inhibition of PDE5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Universidade Federal De Lavras-Ufla

Curated by ChEMBL
LigandPNGBDBM50134104((3aR,10S)-2-Butyl-10-(4-chloro-phenyl)-3a,4,9,10-t...)
Affinity DataIC50:  20nMAssay Description:Inhibition of PDE5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Universidade Federal De Lavras-Ufla

Curated by ChEMBL
LigandPNGBDBM50412322(CHEMBL514402)
Affinity DataIC50:  20nMAssay Description:Inhibition of PDE5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481030(CHEMBL570827)
Affinity DataIC50:  22nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 78 total ) | Next | Last >>
Jump to: