Compile Data Set for Download or QSAR
maximum 50k data
Found 53 with Last Name = 'de capua' and Initial = 'a'
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50272772(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKi:  0.570nMAssay Description:Binding affinity towards somatostatin receptor type 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50175598(CHEMBL262017 | H-D-Phe-Cys-Tyr-D-Trp-Lys-Val-Cys-T...)
Affinity DataKi:  1.70nMAssay Description:Binding affinity towards somatostatin receptor type 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50272772(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKi:  6.80nMAssay Description:Binding affinity towards somatostatin receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50175598(CHEMBL262017 | H-D-Phe-Cys-Tyr-D-Trp-Lys-Val-Cys-T...)
Affinity DataKi:  13.1nMAssay Description:Binding affinity towards somatostatin receptor type 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50272772(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKi:  26.8nMAssay Description:Binding affinity towards somatostatin receptor type 3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50272772(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKi:  875nMAssay Description:Binding affinity towards somatostatin receptor type 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50175598(CHEMBL262017 | H-D-Phe-Cys-Tyr-D-Trp-Lys-Val-Cys-T...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity towards somatostatin receptor type 3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50175598(CHEMBL262017 | H-D-Phe-Cys-Tyr-D-Trp-Lys-Val-Cys-T...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity towards somatostatin receptor type 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50175598(CHEMBL262017 | H-D-Phe-Cys-Tyr-D-Trp-Lys-Val-Cys-T...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity towards somatostatin receptor type 4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50272772(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity towards somatostatin receptor type 4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50272772(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataIC50:  0.0200nMAssay Description:Inhibitory concentration against human somatostatin receptor type 2 in CC531 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50175599((4-amino-3-iodo)-D-Phe-c[Cys-(3-iodo)-Tyr-D-Trp-Ly...)
Affinity DataIC50:  0.630nMAssay Description:Inhibitory concentration against human somatostatin receptor type 2 in CC531 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50175599((4-amino-3-iodo)-D-Phe-c[Cys-(3-iodo)-Tyr-D-Trp-Ly...)
Affinity DataIC50:  0.650nMAssay Description:Inhibitory concentration against human somatostatin receptor type 5 in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50175600((4-amino)-D-Phe-c[Cys-(3-iodo)-Tyr-D-Trp-Lys-Val-C...)
Affinity DataIC50:  1nMAssay Description:Inhibitory concentration against human somatostatin receptor type 5 in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50175590((4-amino)-D-Phe-c[Cys-Tyr-D-Trp-Lys-Val-Cys]-D-Asp...)
Affinity DataIC50:  1.10nMAssay Description:Inhibitory concentration against human somatostatin receptor type 2 in CC531 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50175594((4-amino-3-iodo)-D-Phe-c[Cys-Tyr-D-Trp-Lys-Val-Cys...)
Affinity DataIC50:  1.40nMAssay Description:Inhibitory concentration against human somatostatin receptor type 2 in CC531 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50175596((4-amino)-D-Phe-c[Cys-Tyr-D-Trp-Lys-Val-Cys]-Thr-N...)
Affinity DataIC50:  1.60nMAssay Description:Inhibitory concentration against human somatostatin receptor type 2 in CC531 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50175595((4-amino-3-iodo)-D-Phe-c[Cys-(3-iodo)-Tyr-D-Trp-Ly...)
Affinity DataIC50:  1.90nMAssay Description:Inhibitory concentration against human somatostatin receptor type 2 in CC531 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50175595((4-amino-3-iodo)-D-Phe-c[Cys-(3-iodo)-Tyr-D-Trp-Ly...)
Affinity DataIC50:  2.90nMAssay Description:Inhibitory concentration against human somatostatin receptor type 5 in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50175597((4-amino)-D-Phe-c[Cys-Tyr-D-Trp-Lys-Val-Cys]-D-Thr...)
Affinity DataIC50:  3.40nMAssay Description:Inhibitory concentration against human somatostatin receptor type 5 in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50175601(CHEMBL269532 | D-Phe-c[Cys-Tyr-D-Trp-Lys-Val-Cys]-...)
Affinity DataIC50:  5.60nMAssay Description:Inhibitory concentration against human somatostatin receptor type 5 in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50175600((4-amino)-D-Phe-c[Cys-(3-iodo)-Tyr-D-Trp-Lys-Val-C...)
Affinity DataIC50:  6.20nMAssay Description:Inhibitory concentration against human somatostatin receptor type 2 in CC531 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50175594((4-amino-3-iodo)-D-Phe-c[Cys-Tyr-D-Trp-Lys-Val-Cys...)
Affinity DataIC50:  10nMAssay Description:Inhibitory concentration against human somatostatin receptor type 5 in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50175593((4-amino)-D-Phe-c[Cys-Tyr-D-Trp-Lys-Val-Cys]-Asp-N...)
Affinity DataIC50:  11nMAssay Description:Inhibitory concentration against human somatostatin receptor type 2 in CC531 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50175591((4-amino-3-iodo)-D-Phe-c[Cys-Tyr-D-Trp-Lys-Val-Cys...)
Affinity DataIC50:  12nMAssay Description:Inhibitory concentration against human somatostatin receptor type 2 in CC531 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50175596((4-amino)-D-Phe-c[Cys-Tyr-D-Trp-Lys-Val-Cys]-Thr-N...)
Affinity DataIC50:  14nMAssay Description:Inhibitory concentration against human somatostatin receptor type 5 in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50175597((4-amino)-D-Phe-c[Cys-Tyr-D-Trp-Lys-Val-Cys]-D-Thr...)
Affinity DataIC50:  17nMAssay Description:Inhibitory concentration against human somatostatin receptor type 2 in CC531 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50175601(CHEMBL269532 | D-Phe-c[Cys-Tyr-D-Trp-Lys-Val-Cys]-...)
Affinity DataIC50:  18.6nMAssay Description:Inhibitory concentration against human somatostatin receptor type 2 in CC531 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50272772(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataIC50:  21.8nMAssay Description:Inhibitory concentration against human somatostatin receptor type 5 in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50175590((4-amino)-D-Phe-c[Cys-Tyr-D-Trp-Lys-Val-Cys]-D-Asp...)
Affinity DataIC50:  30nMAssay Description:Inhibitory concentration against human somatostatin receptor type 5 in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Istituto Di Biostrutture E Bioimmagini-Cnr

Curated by ChEMBL
LigandPNGBDBM50215386((S)-5-(2-((S)-1-((S)-1-((S)-1-((S)-1-(3-amino-1-((...)
Affinity DataIC50:  32nMAssay Description:Displacement of [111In]DTPAGlu-Gly-[Tyr27(SO3H)]CCK8 from human CCK1 receptor expressed in A431 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50175593((4-amino)-D-Phe-c[Cys-Tyr-D-Trp-Lys-Val-Cys]-Asp-N...)
Affinity DataIC50:  54nMAssay Description:Inhibitory concentration against human somatostatin receptor type 5 in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50175591((4-amino-3-iodo)-D-Phe-c[Cys-Tyr-D-Trp-Lys-Val-Cys...)
Affinity DataIC50:  74nMAssay Description:Inhibitory concentration against human somatostatin receptor type 5 in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50272772(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataIC50:  92.9nMAssay Description:Inhibitory concentration against human somatostatin receptor type 3 in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50175596((4-amino)-D-Phe-c[Cys-Tyr-D-Trp-Lys-Val-Cys]-Thr-N...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory concentration against human somatostatin receptor type 3 in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50175593((4-amino)-D-Phe-c[Cys-Tyr-D-Trp-Lys-Val-Cys]-Asp-N...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory concentration against human somatostatin receptor type 3 in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50175595((4-amino-3-iodo)-D-Phe-c[Cys-(3-iodo)-Tyr-D-Trp-Ly...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory concentration against human somatostatin receptor type 3 in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50175601(CHEMBL269532 | D-Phe-c[Cys-Tyr-D-Trp-Lys-Val-Cys]-...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory concentration against human somatostatin receptor type 3 in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50175590((4-amino)-D-Phe-c[Cys-Tyr-D-Trp-Lys-Val-Cys]-D-Asp...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory concentration against human somatostatin receptor type 3 in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50175591((4-amino-3-iodo)-D-Phe-c[Cys-Tyr-D-Trp-Lys-Val-Cys...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory concentration against human somatostatin receptor type 3 in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50175599((4-amino-3-iodo)-D-Phe-c[Cys-(3-iodo)-Tyr-D-Trp-Ly...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory concentration against human somatostatin receptor type 3 in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50175600((4-amino)-D-Phe-c[Cys-(3-iodo)-Tyr-D-Trp-Lys-Val-C...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory concentration against human somatostatin receptor type 3 in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50175594((4-amino-3-iodo)-D-Phe-c[Cys-Tyr-D-Trp-Lys-Val-Cys...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory concentration against human somatostatin receptor type 3 in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50175597((4-amino)-D-Phe-c[Cys-Tyr-D-Trp-Lys-Val-Cys]-D-Thr...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory concentration against human somatostatin receptor type 3 in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Istituto Di Biostrutture E Bioimmagini-Cnr

Curated by ChEMBL
LigandPNGBDBM50215383((3S)-3-amino-3-{[(1S)-1-{[(1S)-1-{[(5S,8S,11S)-11-...)
Affinity DataIC50:  6.45E+3nMAssay Description:Displacement of [111In]DTPAGlu-Gly-[Tyr27(SO3H)]CCK8 from human CCK1 receptor expressed in A431 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Istituto Di Biostrutture E Bioimmagini-Cnr

Curated by ChEMBL
LigandPNGBDBM50215381((3S)-3-amino-3-{[(1S)-1-{[(1S)-1-{[(2S,5S,8S)-11-[...)
Affinity DataIC50:  6.94E+3nMAssay Description:Displacement of [111In]DTPAGlu-Gly-[Tyr27(SO3H)]CCK8 from human CCK1 receptor expressed in A431 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Istituto Di Biostrutture E Bioimmagini-Cnr

Curated by ChEMBL
LigandPNGBDBM50215385((3S)-3-amino-3-{[(1S)-1-{[(1S)-1-{[(2S,5S,8S,11S)-...)
Affinity DataIC50:  7.20E+3nMAssay Description:Displacement of [111In]DTPAGlu-Gly-[Tyr27(SO3H)]CCK8 from human CCK1 receptor expressed in A431 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Istituto Di Biostrutture E Bioimmagini-Cnr

Curated by ChEMBL
LigandPNGBDBM50215388((3S)-3-amino-3-{[(1S)-1-{[(1S)-1-{[(2S,5S,8S)-11-[...)
Affinity DataIC50:  7.46E+3nMAssay Description:Displacement of [111In]DTPAGlu-Gly-[Tyr27(SO3H)]CCK8 from human CCK1 receptor expressed in A431 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Istituto Di Biostrutture E Bioimmagini-Cnr

Curated by ChEMBL
LigandPNGBDBM50215379((3S)-3-amino-3-{[(1S)-1-{[(1S)-1-{[(3S,6S,9S,12S,1...)
Affinity DataIC50:  1.50E+4nMAssay Description:Displacement of [111In]DTPAGlu-Gly-[Tyr27(SO3H)]CCK8 from human CCK1 receptor expressed in A431 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Istituto Di Biostrutture E Bioimmagini-Cnr

Curated by ChEMBL
LigandPNGBDBM50215384((3S)-3-amino-3-{[(1S)-1-{[(1S)-1-{[(2S,5S,8S,11S)-...)
Affinity DataIC50:  2.48E+4nMAssay Description:Displacement of [111In]DTPAGlu-Gly-[Tyr27(SO3H)]CCK8 from human CCK1 receptor expressed in A431 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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