Affinity DataKi: 93nMAssay Description:Affinity tested by in vitro competition assay of [125I]ASOR binding to parenchymal rat liver cellsMore data for this Ligand-Target Pair
Affinity DataKi: 93nMAssay Description:Affinity tested by in vitro competition assay of [125I]ASOR binding to parenchymal rat liver cellsMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Affinity tested by in vitro competition assay of [125I]ASOR binding to parenchymal rat liver cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inhibition of Squalene SynthaseMore data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Inhibition of [3H]FPP incorporation by Protein FarnesyltransferaseMore data for this Ligand-Target Pair
Affinity DataIC50: 350nMAssay Description:In vitro anti-thrombin activity was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 384nMAssay Description:Displacement of [125I]-echistatin from alphaIIb-beta3 integrin of human plateletsMore data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataIC50: 420nMAssay Description:Inhibition of [3H]FPP incorporation by Protein FarnesyltransferaseMore data for this Ligand-Target Pair
Affinity DataIC50: 570nMAssay Description:Antithrombin III (ATIII)-mediated anti-Xa activity was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of Squalene SynthaseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.49E+3nMAssay Description:Displacement of [125I]-echistatin from alphaV-beta3 integrin of human skin fibroblastsMore data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataIC50: 1.81E+3nMAssay Description:Inhibition of Farnesyl TransferaseMore data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of [3H]FPP incorporation by Protein FarnesyltransferaseMore data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataIC50: 3.99E+3nMAssay Description:Inhibition of Farnesyl TransferaseMore data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataIC50: 1.35E+4nMAssay Description:Inhibition of Farnesyl TransferaseMore data for this Ligand-Target Pair
TargetGeranylgeranyl transferase type-1 subunit beta/Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of [3H]GGPP incorporation by Protein Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
Affinity DataIC50: 2.33E+4nMAssay Description:Inhibition of Squalene SynthaseMore data for this Ligand-Target Pair
Affinity DataIC50: 3.22E+4nMAssay Description:Displacement of [125I]-echistatin from alphaIIb-beta3 integrin of human plateletsMore data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataIC50: 3.42E+4nMAssay Description:Inhibition of Farnesyl TransferaseMore data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataIC50: 4.20E+4nMAssay Description:Inhibition of [3H]FPP incorporation by Protein FarnesyltransferaseMore data for this Ligand-Target Pair
Affinity DataIC50: 4.64E+4nMAssay Description:Inhibition of Squalene SynthaseMore data for this Ligand-Target Pair
TargetGeranylgeranyl transferase type-1 subunit beta/Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataIC50: 4.80E+4nMAssay Description:Inhibition of [3H]GGPP incorporation by Protein Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of Squalene SynthaseMore data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataIC50: 5.62E+4nMAssay Description:Inhibition of Farnesyl TransferaseMore data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataIC50: 5.70E+4nMAssay Description:Inhibition of [3H]FPP incorporation by Protein FarnesyltransferaseMore data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataIC50: 9.10E+4nMAssay Description:Inhibition of [3H]FPP incorporation by Protein FarnesyltransferaseMore data for this Ligand-Target Pair
Affinity DataIC50: 9.81E+4nMAssay Description:Displacement of [125I]-echistatin from alphaV-beta3 integrin of human skin fibroblastsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.98E+5nMAssay Description:Displacement of [125I]-echistatin from alphaIIb-beta3 integrin of human plateletsMore data for this Ligand-Target Pair
TargetGeranylgeranyl transferase type-1 subunit beta/Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataIC50: 2.06E+5nMAssay Description:Inhibition of [3H]GGPP incorporation by Protein Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
TargetGeranylgeranyl transferase type-1 subunit beta/Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataIC50: 2.61E+5nMAssay Description:Inhibition of [3H]GGPP incorporation by Protein Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
TargetGeranylgeranyl transferase type-1 subunit beta/Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataIC50: 2.70E+5nMAssay Description:Inhibition of [3H]GGPP incorporation by Protein Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
TargetGeranylgeranyl transferase type-1 subunit beta/Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataIC50: 3.11E+5nMAssay Description:Inhibition of [3H]GGPP incorporation by Protein Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataIC50: 3.21E+5nMAssay Description:Inhibition of [3H]FPP incorporation by Protein FarnesyltransferaseMore data for this Ligand-Target Pair
TargetGeranylgeranyl transferase type-1 subunit beta/Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataIC50: 4.64E+5nMAssay Description:Inhibition of [3H]GGPP incorporation by Protein Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
TargetGeranylgeranyl transferase type-1 subunit beta/Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of [3H]GGPP incorporation by Protein Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
TargetGeranylgeranyl transferase type-1 subunit beta/Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataIC50: 5.21E+5nMAssay Description:Inhibition of [3H]GGPP incorporation by Protein Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
Affinity DataIC50: 5.97E+5nMAssay Description:Displacement of [125I]-echistatin from alphaV-beta3 integrin of human skin fibroblastsMore data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of [3H]FPP incorporation by Protein FarnesyltransferaseMore data for this Ligand-Target Pair
TargetGeranylgeranyl transferase type-1 subunit beta/Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of [3H]GGPP incorporation by Protein Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of [3H]FPP incorporation by Protein FarnesyltransferaseMore data for this Ligand-Target Pair
TargetGeranylgeranyl transferase type-1 subunit beta/Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of [3H]GGPP incorporation by Protein Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
Affinity DataEC50: 750nMAssay Description:Effective concentration against thrombin was determinedMore data for this Ligand-Target Pair