Compile Data Set for Download or QSAR
maximum 50k data
Found 11 with Last Name = 'van witteloostuijn' and Initial = 'sb'
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50240819(CHEMBL4084119)
Affinity DataEC50:  0.0670nMAssay Description:Agonist activity at human GLP1 receptor expressed in HEK293 cells harboring mCerulean and mCitrine fused Epac protein assessed as increase in cAMP le...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50121394(CHEMBL3616711)
Affinity DataEC50:  0.0230nMAssay Description:Agonist activity at human GLP1 receptor expressed in HEK293 cells harboring mCerulean and mCitrine fused Epac protein assessed as increase in cAMP le...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50152769(CHEMBL410972 | GLP-1(7-36)-NH2 | GLP-17-(7-36) der...)
Affinity DataEC50:  0.0440nMAssay Description:Agonist activity at human GLP1 receptor expressed in HEK293 cells harboring mCerulean and mCitrine fused Epac protein assessed as increase in cAMP le...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50240820(CHEMBL4073765)
Affinity DataEC50:  0.0680nMAssay Description:Agonist activity at human GLP1 receptor expressed in HEK293 cells harboring mCerulean and mCitrine fused Epac protein assessed as increase in cAMP le...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50240821(CHEMBL4100575)
Affinity DataEC50:  0.221nMAssay Description:Agonist activity at human GLP1 receptor expressed in HEK293 cells harboring mCerulean and mCitrine fused Epac protein assessed as increase in cAMP le...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlbumin(Homo sapiens (Human))
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM17638(2-{1-[(4-chlorophenyl)carbonyl]-5-methoxy-2-methyl...)
Affinity DataKd:  700nMAssay Description:Binding affinity to human serum albuminMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50240823(CHEMBL4083273)
Affinity DataEC50:  0.118nMAssay Description:Binding affinity against dopamine receptor D2 by using [3H]spiperone as radioligand in caudate-putamen of monkeyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlbumin(Homo sapiens (Human))
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50240510(CHEMBL898 | DIFLUNISAL)
Affinity DataKd:  3.00E+3nMAssay Description:Binding affinity to human serum albuminMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50240824(CHEMBL4062410)
Affinity DataEC50:  0.148nMAssay Description:Agonist activity at human GLP1 receptor expressed in HEK293 cells harboring mCerulean and mCitrine fused Epac protein assessed as increase in cAMP le...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50240825(CHEMBL4103967)
Affinity DataEC50:  0.522nMAssay Description:Agonist activity at human GLP1 receptor expressed in HEK293 cells harboring mCerulean and mCitrine fused Epac protein assessed as increase in cAMP le...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50240822(CHEMBL4079706)
Affinity DataEC50:  0.547nMAssay Description:Agonist activity at human GLP1 receptor expressed in HEK293 cells harboring mCerulean and mCitrine fused Epac protein assessed as increase in cAMP le...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed