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Found 368 with Last Name = 'van der neut' and Initial = 'm'
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50316949((3R)-3-((3-((2-oxo-1,2,3,4-tetrahydroquinolin-7-yl...)
Affinity DataKi:  0.260nMAssay Description:Displacement of [3H]citalopram form human SRET by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50072775(2-((1R,2R,5R)-5-hydroxy-2-(3-hydroxypropyl)cyclohe...)
Affinity DataKi:  0.620nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50172158((S)-N-(1-(4-(4-chloro-2-(2-fluorophenylsulfonyl)ph...)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302225((1S)-1-[3-(dimethylamino)propyl]-1-(4-fluorophenyl...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]citalopram form human SRET by liquid scintillation countingMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50309538(5-Ethyl-2-methyl-1-phenyl-1H-imidazole-4-carboxyli...)
Affinity DataKi:  1.03nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50072775(2-((1R,2R,5R)-5-hydroxy-2-(3-hydroxypropyl)cyclohe...)
Affinity DataKi:  1.36nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50316948((R)-7-[8-(2-Oxo-1,2,3,4-tetrahydro-quinolin-7-ylme...)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]citalopram form human SRET by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50159929(CHEMBL3786752)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]-N-Methyl-Lysergic acid diethylamide from human 5-HT6 receptor expressed in CHO cells after 30 mins by liquid scintillation count...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50309540(2-Ethyl-5-methyl-1-phenyl-1H-imidazole-4-carboxyli...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50316947(CHEMBL1087818 | N-(3-(2-(8-((2-oxo-1,2,3,4-tetrahy...)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]citalopram form human SRET by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50159784(CHEMBL3785453)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]-N-Methyl-Lysergic acid diethylamide from human 5-HT6 receptor expressed in CHO cells after 30 mins by liquid scintillation count...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50316955((R)-3-((4-((2-oxo-1,2,3,4-tetrahydroquinolin-7-yl)...)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]citalopram form human SRET by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50312822((R)-1-(4-chlorophenyl)-N-methyl-5-phenyl-N'-(4-(tr...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]CP-55940 from human cannabinoid CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50316952((R)-3-((4-(2-oxo-1,2,3,4-tetrahydroquinolin-7-ylox...)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]spiperone form human dopamine D2 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50309534(2,5-Dimethyl-1-phenyl-1H-imidazole-4-carboxylic ac...)
Affinity DataKi:  2.70nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50354607(CHEMBL1834337)
Affinity DataKi:  2.70nMAssay Description:Displacement of [3H]-methyllysergic acid diethylamide from human 5-HT6 receptor expressed in CHO cells after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50354585(CHEMBL1834226)
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]-methyllysergic acid diethylamide from human 5-HT6 receptor expressed in CHO cells after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50354585(CHEMBL1834226)
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]-methyllysergic acid diethylamide from human 5-HT6 receptor expressed in CHO cells after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50317250(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-(methy...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]spiperone form human dopamine D2 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCannabinoid receptor 1(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50303835(3-(4-Chlorophenyl)-N'-((4-chlorophenyl)sulfonyl)-N...)
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50325599(3-Pentyl-4-phenyl-4,5-dihydro-pyrazole-1-carboxyli...)
Affinity DataKi:  3.26nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50325587(3-butyl-5,5-dimethyl-4-phenyl-N-((1R,2S,4R)-1,7,7-...)
Affinity DataKi:  3.40nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50309537(2,5-dimethyl-1-phenyl-N-(2-(trifluoromethyl)benzyl...)
Affinity DataKi:  3.5nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50354608(CHEMBL1834342)
Affinity DataKi:  4.10nMAssay Description:Displacement of [3H]-methyllysergic acid diethylamide from human 5-HT6 receptor expressed in CHO cells after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50325590(1-pentyl-5-phenyl-N-((1R,2S,4R)-1,7,7-trimethylbic...)
Affinity DataKi:  4.70nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50312833((S)-3-(4-chlorophenyl)-N-methyl-4-phenyl-N'-(4-(tr...)
Affinity DataKi:  4.70nMAssay Description:Displacement of [3H]CP-55940 from human cannabinoid CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50159769(CHEMBL3785100)
Affinity DataKi:  4.80nMAssay Description:Displacement of [3H]-N-Methyl-Lysergic acid diethylamide from human 5-HT6 receptor expressed in CHO cells after 30 mins by liquid scintillation count...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50316946(CHEMBL1087585 | N-(2-fluoro-5-(2-(8-((2-oxo-1,2,3,...)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]citalopram form human SRET by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50354609(CHEMBL1834348)
Affinity DataKi:  5.20nMAssay Description:Displacement of [3H]-methyllysergic acid diethylamide from human 5-HT6 receptor expressed in CHO cells after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50325584((+)-3-pentyl-4-phenyl-N-((1R,2S,4S)-1,7,7-trimethy...)
Affinity DataKi:  5.30nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50354610(CHEMBL1834338)
Affinity DataKi:  5.60nMAssay Description:Displacement of [3H]-methyllysergic acid diethylamide from human 5-HT6 receptor expressed in CHO cells after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50159783(CHEMBL3787201)
Affinity DataKi:  5.80nMAssay Description:Displacement of [3H]-N-Methyl-Lysergic acid diethylamide from human 5-HT6 receptor expressed in CHO cells after 30 mins by liquid scintillation count...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50159754(CHEMBL3785512)
Affinity DataKi:  6.10nMAssay Description:Displacement of [3H]-N-Methyl-Lysergic acid diethylamide from human 5-HT6 receptor expressed in CHO cells after 30 mins by liquid scintillation count...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50325591(5-(2-fluorophenyl)-1-pentyl-N-((1R,2S,4R)-1,7,7-tr...)
Affinity DataKi:  6.10nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50316948((R)-7-[8-(2-Oxo-1,2,3,4-tetrahydro-quinolin-7-ylme...)
Affinity DataKi:  6.30nMAssay Description:Displacement of [3H]spiperone form human dopamine D2 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50325597(3-Pentyl-4-phenyl-4,5-dihydro-pyraz ole-1-carboxyl...)
Affinity DataKi:  6.30nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50354611(CHEMBL1834347)
Affinity DataKi:  6.40nMAssay Description:Displacement of [3H]-methyllysergic acid diethylamide from human 5-HT6 receptor expressed in CHO cells after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50325597(3-Pentyl-4-phenyl-4,5-dihydro-pyraz ole-1-carboxyl...)
Affinity DataKi:  6.40nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Solvay Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM50004108((+-)-nicotine | (R,S)-nicotine | (RS)-nicotine | 3...)
TargetD(2) dopamine receptor(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50316946(CHEMBL1087585 | N-(2-fluoro-5-(2-(8-((2-oxo-1,2,3,...)
Affinity DataKi:  7nMAssay Description:Displacement of [3H]spiperone form human dopamine D2 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50159786(CHEMBL3786693)
Affinity DataKi:  7.10nMAssay Description:Displacement of [3H]-N-Methyl-Lysergic acid diethylamide from human 5-HT6 receptor expressed in CHO cells after 30 mins by liquid scintillation count...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50325588(1-Pentyl-5-phenyl-4,5-dihydro-1H-pyrazole-3-carbox...)
Affinity DataKi:  7.10nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50354612(CHEMBL1834350)
Affinity DataKi:  7.20nMAssay Description:Displacement of [3H]-methyllysergic acid diethylamide from human 5-HT6 receptor expressed in CHO cells after 30 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50159931(CHEMBL3785626)
Affinity DataKi:  7.20nMAssay Description:Displacement of [3H]-N-Methyl-Lysergic acid diethylamide from human 5-HT6 receptor expressed in CHO cells after 30 mins by liquid scintillation count...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50325584((+)-3-pentyl-4-phenyl-N-((1R,2S,4S)-1,7,7-trimethy...)
Affinity DataKi:  7.40nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50325584((+)-3-pentyl-4-phenyl-N-((1R,2S,4S)-1,7,7-trimethy...)
Affinity DataKi:  7.40nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50325592(3-Pentyl-4-phenyl-4,5-dihydro-pyrazole-1-carboxyli...)
Affinity DataKi:  7.40nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50312831(3-(4-chlorophenyl)-N'-(4-fluoropiperidin-1-ylsulfo...)
Affinity DataKi:  7.5nMAssay Description:Displacement of [3H]CP-55940 from human cannabinoid CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Abbott Healthcare Products

Curated by ChEMBL
LigandPNGBDBM50312821((S)-1-(4-chlorophenyl)-N-methyl-5-phenyl-N'-(4-(tr...)
Affinity DataKi:  7.60nMAssay Description:Displacement of [3H]CP-55940 from human cannabinoid CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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