TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.0550nMAssay Description:Displacement of [3H]vesamicol from VAChT in Torpedo californica cholinergic synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.410nMAssay Description:Displacement of [3H]vesamicol from VAChT in Torpedo californica cholinergic synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.530nMAssay Description:Displacement of [3H]vesamicol from VAChT in Torpedo californica cholinergic synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.540nMAssay Description:Displacement of [3H]vesamicol from VAChT in Torpedo californica cholinergic synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.660nMAssay Description:Displacement of [3H]vesamicol from VAChT in Torpedo californica cholinergic synaptic vesiclesMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 0.900nMAssay Description:In vitro binding affinity towards Nicotinic acetylcholine receptor alpha7 using [125I]-alpha-Bungarotoxin in rat brainMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 1.38nMAssay Description:Displacement of [3H]vesamicol from VAChT in Torpedo californica cholinergic synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 1.64nMAssay Description:Displacement of [3H]vesamicol from VAChT in Torpedo californica cholinergic synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 1.83nMAssay Description:Displacement of [3H]vesamicol from VAChT in Torpedo californica cholinergic synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Displacement of [3H]vesamicol from VAChT in Torpedo californica cholinergic synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 2.07nMAssay Description:Displacement of [3H]vesamicol from VAChT in Torpedo californica cholinergic synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 2.08nMAssay Description:Displacement of [3H]vesamicol from VAChT in Torpedo californica cholinergic synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 2.40nMAssay Description:Displacement of [3H]vesamicol from VAChT in Torpedo californica cholinergic synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 2.40nMAssay Description:Displacement of [3H]vesamicol from VAChT in Torpedo californica cholinergic synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 4.90nMAssay Description:Displacement of [3H]vesamicol from VAChT in Torpedo californica cholinergic synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Displacement of [3H]vesamicol from VAChT in Torpedo californica cholinergic synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 7.60nMAssay Description:Displacement of [3H]vesamicol from VAChT in Torpedo californica cholinergic synaptic vesiclesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 9.39nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membrane homogenates after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 15.9nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membrane homogenates after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 19.9nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membrane homogenates after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 21nMAssay Description:In vitro binding affinity towards nicotinic (alpha4-beta2) receptor using [3H]cytisine in rat brainMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 25.8nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membrane homogenates after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 29.4nMAssay Description:Displacement of [3H]vesamicol from VAChT in Torpedo californica cholinergic synaptic vesiclesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 29.5nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membrane homogenates after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 31nMAssay Description:Displacement of [3H]vesamicol from VAChT in Torpedo californica cholinergic synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 46.8nMAssay Description:Displacement of [3H]vesamicol from VAChT in Torpedo californica cholinergic synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:Displacement of [3H]vesamicol from VAChT in Torpedo californica cholinergic synaptic vesiclesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 50.2nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membrane homogenates after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 51.4nMAssay Description:Displacement of [3H]vesamicol from VAChT in Torpedo californica cholinergic synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 68.5nMAssay Description:Displacement of [3H]vesamicol from VAChT in Torpedo californica cholinergic synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 68.5nMAssay Description:Displacement of [3H]vesamicol from VAChT in Torpedo californica cholinergic synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 89.5nMAssay Description:Displacement of [3H]vesamicol from VAChT in Torpedo californica cholinergic synaptic vesiclesMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 93nMAssay Description:In vitro binding affinity towards nicotinic (alpha4-beta2) receptor using [3H]cytisine in rat brainMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 118nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membrane homogenates after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 129nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membrane homogenates after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 134nMAssay Description:Displacement of [3H]vesamicol from VAChT in Torpedo californica cholinergic synaptic vesiclesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 194nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membrane homogenates after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 281nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membrane homogenates after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 303nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membrane homogenates after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 395nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membrane homogenates after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 423nMAssay Description:Displacement of [3H]vesamicol from VAChT in Torpedo californica cholinergic synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 447nMAssay Description:Displacement of [3H]vesamicol from VAChT in Torpedo californica cholinergic synaptic vesiclesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 483nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membrane homogenates after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 497nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membrane homogenates after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 560nMAssay Description:Displacement of [3H]vesamicol from VAChT in Torpedo californica cholinergic synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 650nMAssay Description:Displacement of [3H]vesamicol from VAChT in Torpedo californica cholinergic synaptic vesiclesMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 763nMAssay Description:Displacement of [3H]vesamicol from VAChT in Torpedo californica cholinergic synaptic vesiclesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membrane homogenates after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membrane homogenates after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 receptor in guinea pig brain membrane homogenates after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair