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Found 26 with Last Name = 'von kleist' and Initial = 'l'
TargetLanosterol synthase(Rattus norvegicus)
Caprotec Bioanalytics

Curated by ChEMBL
LigandPNGBDBM50180953(CHEMBL3818719)
Affinity DataIC50:  54nMAssay Description:Inhibition of human recombinant His-tagged soluble COMT expressed in Escherichia coli BL21 using aesculetin as substrate after 60 mins by microplate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Rattus norvegicus)
Caprotec Bioanalytics

Curated by ChEMBL
LigandPNGBDBM50108877((3,4-Dihydroxy-5-nitro-phenyl)-p-tolyl-methanone |...)
Affinity DataIC50:  127nMAssay Description:Inhibition of human recombinant His-tagged soluble COMT expressed in Escherichia coli BL21 using aesculetin as substrate after 60 mins by microplate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Rattus norvegicus)
Caprotec Bioanalytics

Curated by ChEMBL
LigandPNGBDBM50180952(CHEMBL3818350)
Affinity DataIC50:  179nMAssay Description:Inhibition of human recombinant His-tagged soluble COMT expressed in Escherichia coli BL21 using aesculetin as substrate after 60 mins by microplate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Rattus norvegicus)
Caprotec Bioanalytics

Curated by ChEMBL
LigandPNGBDBM50108879((2E)-2-cyano-3-(3,4-dihydroxy-5-nitrophenyl)-N,N-d...)
Affinity DataIC50:  386nMAssay Description:Inhibition of human recombinant His-tagged soluble COMT expressed in Escherichia coli BL21 using aesculetin as substrate after 60 mins by microplate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Rattus norvegicus)
Caprotec Bioanalytics

Curated by ChEMBL
LigandPNGBDBM50180954(CHEMBL3819488)
Affinity DataIC50:  648nMAssay Description:Inhibition of human recombinant His-tagged soluble COMT expressed in Escherichia coli BL21 using aesculetin as substrate after 60 mins by microplate ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDynamin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50388829(CHEMBL2062753)
Affinity DataIC50:  5.90E+3nMAssay Description:Inhibition of dynamin1-mediated endocytosis in human U2OS cells assessed as inhibition of Texas red-Tf uptake incubated for 30 mins prior to Texas re...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetClathrin heavy chain 1(Homo sapiens (Human))
The University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM50446548(CHEMBL3110181)
Affinity DataIC50:  6.90E+3nMAssay Description:Inhibition of recombinant GST-tagged clathrin heavy chain (unknown origin) after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDynamin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50388828(CHEMBL2062743)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of dynamin1-mediated endocytosis in human U2OS cells assessed as inhibition of Texas red-Tf uptake incubated for 30 mins prior to Texas re...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetClathrin heavy chain 1(Homo sapiens (Human))
The University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM50446543(CHEMBL3110178)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of recombinant GST-tagged clathrin heavy chain (unknown origin) after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetClathrin heavy chain 1(Homo sapiens (Human))
The University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM50446549(CHEMBL3110180)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of recombinant GST-tagged clathrin heavy chain (unknown origin) after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetClathrin heavy chain 1(Homo sapiens (Human))
The University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM50446544(CHEMBL3110188)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of recombinant GST-tagged clathrin heavy chain (unknown origin) after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetClathrin heavy chain 1(Homo sapiens (Human))
The University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM50446542(CHEMBL3110179)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of recombinant GST-tagged clathrin heavy chain (unknown origin) after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetClathrin heavy chain 1(Homo sapiens (Human))
The University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM50446540(CHEMBL3110184)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of recombinant GST-tagged clathrin heavy chain (unknown origin) after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetClathrin heavy chain 1(Homo sapiens (Human))
The University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM50446546(CHEMBL3110183)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of recombinant GST-tagged clathrin heavy chain (unknown origin) after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetClathrin heavy chain 1(Homo sapiens (Human))
The University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM50446551(CHEMBL3110174)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of recombinant GST-tagged clathrin heavy chain (unknown origin) after 1 hr by ELISAMore data for this Ligand-Target Pair
TargetDynamin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50388827(CHEMBL2062731)
Affinity DataIC50:  1.81E+4nMAssay Description:Inhibition of dynamin1-mediated endocytosis in human U2OS cells assessed as inhibition of Texas red-Tf uptake incubated for 30 mins prior to Texas re...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetClathrin heavy chain 1(Homo sapiens (Human))
The University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM50446547(CHEMBL3110182)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of recombinant GST-tagged clathrin heavy chain (unknown origin) after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetClathrin heavy chain 1(Homo sapiens (Human))
The University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM50446553(CHEMBL3110161)
Affinity DataIC50:  8.00E+4nMAssay Description:Inhibition of recombinant GST-tagged clathrin heavy chain (unknown origin) after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetClathrin heavy chain 1(Homo sapiens (Human))
The University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM50446552(CHEMBL3110162)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of recombinant GST-tagged clathrin heavy chain (unknown origin) after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDynamin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50388830(CHEMBL2062756)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of dynamin1-mediated endocytosis in human U2OS cells assessed as inhibition of Texas red-Tf uptake incubated for 30 mins prior to Texas re...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetClathrin heavy chain 1(Homo sapiens (Human))
The University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM50446555(CHEMBL3110160)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of recombinant GST-tagged clathrin heavy chain (unknown origin) after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetClathrin heavy chain 1(Homo sapiens (Human))
The University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM50446545(CHEMBL3110186)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of recombinant GST-tagged clathrin heavy chain (unknown origin) after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetClathrin heavy chain 1(Homo sapiens (Human))
The University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM50446541(CHEMBL3110185)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of recombinant GST-tagged clathrin heavy chain (unknown origin) after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetClathrin heavy chain 1(Homo sapiens (Human))
The University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM50446550(CHEMBL3110177)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of recombinant GST-tagged clathrin heavy chain (unknown origin) after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetClathrin heavy chain 1(Homo sapiens (Human))
The University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM50446556(CHEMBL3110158)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of recombinant GST-tagged clathrin heavy chain (unknown origin) after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetClathrin heavy chain 1(Homo sapiens (Human))
The University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM50446554(CHEMBL3110159)
Affinity DataIC50:  1.20E+5nMAssay Description:Inhibition of recombinant GST-tagged clathrin heavy chain (unknown origin) after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed