Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 9 hits for monomerid = 50221583,50221589,50221600,50221603,50221611,50221612,50221583,50221589,50221600,50221603,50221611,50221612   

TargetSerine/threonine-protein kinase Chk1(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50221589(CHEMBL248396 | Chk1_146 | 4-(6,7-dimethoxy-2,4-dih...)
Affinity DataIC50: 5nMAssay Description:Inhibition of Chk1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50221589(CHEMBL248396 | Chk1_146 | 4-(6,7-dimethoxy-2,4-dih...)
Affinity DataIC50: 5nMAssay Description:Abbott Kinase Enzymatics_CHK1/289 CDC25c - IC50(uM) (IC50)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2012
Entry Details PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50221589(CHEMBL248396 | Chk1_146 | 4-(6,7-dimethoxy-2,4-dih...)
Affinity DataKi:  5nMAssay Description:Inhibition of Chk1More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
LigandPNGBDBM50221589(CHEMBL248396 | Chk1_146 | 4-(6,7-dimethoxy-2,4-dih...)
Affinity DataKi:  5.22nMAssay Description:33P-Radiometric_Method1More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2017
Entry Details
D3R

TargetSerine/threonine-protein kinase Chk1(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50221583(4-(6,7-dimethoxy-2,4-dihydro-indeno[1,2-c]pyrazol-...)
Affinity DataIC50: 19nMAssay Description:Inhibition of Chk1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50221603(4-(6,7-dimethoxy-2,4-dihydro-indeno[1,2-c]pyrazol-...)
Affinity DataIC50: 1.74E+3nMAssay Description:Inhibition of Chk1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50221612(3-ethynyl-6,7-dimethoxy-2,4-dihydro-indeno[1,2-c]p...)
Affinity DataIC50: 5.14E+3nMAssay Description:Inhibition of Chk1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50221611(4-(6,7-dimethoxy-2,4-dihydro-indeno[1,2-c]pyrazol-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Chk1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2012
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50221600(4-(6,7-dimethoxy-2,4-dihydro-indeno[1,2-c]pyrazol-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Chk1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2012
Entry Details Article
PubMed