Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 13 hits for monomerid = 50401993,50401998,50402001,50402004,50402005,50401993,50401998,50402001,50402004,50402005
TargetPeroxisome proliferator-activated receptor alpha(Human)
D'Annunzio University of Chieti
Curated by ChEMBL
D'Annunzio University of Chieti
Curated by ChEMBL
Affinity DataEC50: 600nMAssay Description:Transactivation of human GAL4-fused PPARalpha ligand binding domain transfected in HEK293 cells after 18 hrs by dual luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
D'Annunzio University of Chieti
Curated by ChEMBL
D'Annunzio University of Chieti
Curated by ChEMBL
Affinity DataEC50: 1.09E+3nMAssay Description:Agonist activity at Gal4-fused human PPARalpha LBD transfected in HEK293T cells assessed as transcriptional activation incubated for 14 to 16 hrs by ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Human)
D'Annunzio University of Chieti
Curated by ChEMBL
D'Annunzio University of Chieti
Curated by ChEMBL
Affinity DataEC50: 1.40E+3nMAssay Description:Transactivation of human GAL4-fused PPARgamma ligand binding domain transfected in HEK293 cells after 18 hrs by dual luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
D'Annunzio University of Chieti
Curated by ChEMBL
D'Annunzio University of Chieti
Curated by ChEMBL
Affinity DataEC50: 2.10E+3nMAssay Description:Transactivation of GAL4-tagged human PPARalpha LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Human)
Goethe-University Frankfurt
Curated by ChEMBL
Goethe-University Frankfurt
Curated by ChEMBL
Affinity DataEC50: 2.20E+3nMAssay Description:Agonist activity at Gal4-fused human PPARdelta LBD transfected in HEK293T cells assessed as transcriptional activation incubated for 14 to 16 hrs by ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Human)
D'Annunzio University of Chieti
Curated by ChEMBL
D'Annunzio University of Chieti
Curated by ChEMBL
Affinity DataEC50: 2.67E+3nMAssay Description:Agonist activity at Gal4-fused human PPARgamma LBD transfected in HEK293T cells assessed as transcriptional activation incubated for 14 to 16 hrs by ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Human)
D'Annunzio University of Chieti
Curated by ChEMBL
D'Annunzio University of Chieti
Curated by ChEMBL
Affinity DataEC50: 5.90E+3nMAssay Description:Transactivation of human GAL4-fused PPARgamma ligand binding domain transfected in HEK293 cells after 18 hrs by dual luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Human)
Goethe-University Frankfurt
Curated by ChEMBL
Goethe-University Frankfurt
Curated by ChEMBL
Affinity DataEC50: 6.40E+3nMAssay Description:Transactivation of GAL4-tagged human PPARdelta LBD expressed in human HepG2 cells at 100 nM to 100 uM incubated for 20 to 22 hrs by luciferase report...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Human)
D'Annunzio University of Chieti
Curated by ChEMBL
D'Annunzio University of Chieti
Curated by ChEMBL
Affinity DataEC50: 6.90E+3nMAssay Description:Transactivation of human GAL4-fused PPARgamma ligand binding domain transfected in HEK293 cells after 18 hrs by dual luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
D'Annunzio University of Chieti
Curated by ChEMBL
D'Annunzio University of Chieti
Curated by ChEMBL
Affinity DataEC50: 1.16E+4nMAssay Description:Transactivation of human GAL4-fused PPARalpha ligand binding domain transfected in HEK293 cells after 18 hrs by dual luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Human)
D'Annunzio University of Chieti
Curated by ChEMBL
D'Annunzio University of Chieti
Curated by ChEMBL
Affinity DataEC50: 1.26E+4nMAssay Description:Transactivation of human GAL4-fused PPARgamma ligand binding domain transfected in HEK293 cells after 18 hrs by dual luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Human)
D'Annunzio University of Chieti
Curated by ChEMBL
D'Annunzio University of Chieti
Curated by ChEMBL
Affinity DataEC50: 5.46E+4nMAssay Description:Transactivation of human GAL4-fused PPARgamma ligand binding domain transfected in HEK293 cells after 18 hrs by dual luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
D'Annunzio University of Chieti
Curated by ChEMBL
D'Annunzio University of Chieti
Curated by ChEMBL
Affinity DataEC50: 6.40E+4nMAssay Description:Transactivation of human GAL4-fused PPARalpha ligand binding domain transfected in HEK293 cells after 18 hrs by dual luciferase reporter gene assayMore data for this Ligand-Target Pair
