Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

TargetLysine--tRNA ligase(Human)
Yunnan University

Curated by ChEMBL
LigandPNGBDBM50143600(CHEBI:29571 | Dehydroabietic Acid)
Affinity DataIC50:  28nMAssay Description:Inhibition of SYK (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Human)
Yunnan University

Curated by ChEMBL
LigandPNGBDBM50143600(CHEBI:29571 | Dehydroabietic Acid)
Affinity DataIC50: >100nMAssay Description:Inhibition of JAK3 (unknown origin) by mobility shift assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Human)
Southeast University

Curated by ChEMBL
LigandPNGBDBM50143600(CHEBI:29571 | Dehydroabietic Acid)
Affinity DataIC50:  3.63E+4nMAssay Description:Inhibition of human recombinant C-terminal His6-tagged full length human Cdk2/human recombinant N-terminal GST-tagged full-length Cyclin E using hist...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-gamma(Human)
Swiss Federal Institute of Technology (Eth)

Curated by ChEMBL
LigandPNGBDBM50143600(CHEBI:29571 | Dehydroabietic Acid)
Affinity DataEC50:  4.20E+4nMAssay Description:Transactivation of human Gal4-fused RXRgamma LBD expressed in HEK293T cells after 12 to 14 hrs by dual-glo luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Swiss Federal Institute of Technology (Eth)

Curated by ChEMBL
LigandPNGBDBM50143600(CHEBI:29571 | Dehydroabietic Acid)
Affinity DataEC50:  4.20E+4nMAssay Description:Transactivation of human Gal4-fused RXRalpha LBD expressed in HEK293T cells after 12 to 14 hrs by dual-glo luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-beta(Human)
Swiss Federal Institute of Technology (Eth)

Curated by ChEMBL
LigandPNGBDBM50143600(CHEBI:29571 | Dehydroabietic Acid)
Affinity DataEC50:  4.20E+4nMAssay Description:Transactivation of human Gal4-fused RXRbeta LBD expressed in HEK293T cells after 12 to 14 hrs by dual-glo luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed