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Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
1
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Target
NACHT, LRR and PYD domains-containing protein 3
(Human)
Shanghaitech University
Curated by
ChEMBL
Ligand
BDBM50593666
(CHEMBL5189690)
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Affinity Data
IC50: 641nM
Assay Description:
Inhibition of NLRP3 inflammasome activation in PMA differentiated LPS-primed human THP-1 cells assessed as reduction in nigericin-induced IL-1beta le...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
PubMed
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