Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 24 hits in this display   

TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479261(Altertoxin I)
Affinity DataIC50:  1.87E+3nMAssay Description:Inhibition of recombinant FLT3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Human)
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479261(Altertoxin I)
Affinity DataIC50:  2.78E+3nMAssay Description:Inhibition of recombinant Aurora BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Human)
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479261(Altertoxin I)
Affinity DataIC50:  3.97E+3nMAssay Description:Inhibition of recombinant VEGFR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK4(Human)
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479261(Altertoxin I)
Affinity DataIC50:  4.82E+3nMAssay Description:Inhibition of recombinant SAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Human)
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479261(Altertoxin I)
Affinity DataIC50:  4.82E+3nMAssay Description:Inhibition of recombinant Aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin-like growth factor 1 receptor(Human)
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479261(Altertoxin I)
Affinity DataIC50:  4.82E+3nMAssay Description:Inhibition of recombinant IGF1RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479261(Altertoxin I)
Affinity DataIC50:  5.96E+3nMAssay Description:Inhibition of recombinant SRCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNUAK family SNF1-like kinase 1(Human)
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479261(Altertoxin I)
Affinity DataIC50:  6.24E+3nMAssay Description:Inhibition of recombinant ARK5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 3(Human)
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479261(Altertoxin I)
Affinity DataIC50:  7.94E+3nMAssay Description:Inhibition of recombinant VEGFR3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Human)
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479261(Altertoxin I)
Affinity DataIC50:  9.93E+3nMAssay Description:Inhibition of recombinant EGFRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 8(Human)
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479261(Altertoxin I)
Affinity DataIC50:  1.56E+4nMAssay Description:Inhibition of recombinant COTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479261(Altertoxin I)
Affinity DataIC50:  1.81E+4nMAssay Description:Inhibition of recombinant CDK4/CycD1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Human)
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479261(Altertoxin I)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of recombinant B-RAF-V600E mutantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Human)
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479261(Altertoxin I)
Affinity DataIC50:  1.98E+4nMAssay Description:Inhibition of recombinant METMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFocal adhesion kinase 1(Human)
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479261(Altertoxin I)
Affinity DataIC50:  2.07E+4nMAssay Description:Inhibition of recombinant FAKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor beta(Human)
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479261(Altertoxin I)
Affinity DataIC50:  2.15E+4nMAssay Description:Inhibition of recombinant PDGFRbetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiopoietin-1 receptor(Human)
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479261(Altertoxin I)
Affinity DataIC50:  2.49E+4nMAssay Description:Inhibition of recombinant TIE2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Human)
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479261(Altertoxin I)
Affinity DataIC50:  2.52E+4nMAssay Description:Inhibition of recombinant EPHB4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Human)
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479261(Altertoxin I)
Affinity DataIC50:  2.66E+4nMAssay Description:Inhibition of recombinant INSRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479261(Altertoxin I)
Affinity DataIC50: >2.83E+4nMAssay Description:Inhibition of recombinant PLK1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCasein kinase II subunit alpha(Human)
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479261(Altertoxin I)
Affinity DataIC50: >2.83E+4nMAssay Description:Inhibition of recombinant CK2alpha1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479261(Altertoxin I)
Affinity DataIC50: >2.83E+4nMAssay Description:Inhibition of recombinant ERBB2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479261(Altertoxin I)
Affinity DataIC50: >2.83E+4nMAssay Description:Inhibition of recombinant AKT1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Human)
Heinrich-Heine-Universit£T

Curated by ChEMBL
LigandPNGBDBM50479261(Altertoxin I)
Affinity DataIC50: >2.83E+4nMAssay Description:Inhibition of recombinant CDK2/CycAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed