Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetAlpha-2A adrenergic receptor(Human)
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM50473529(CHEMBL165529)
Affinity DataKi:  1.30nMAssay Description:Binding affinity for human alpha-2 adrenergic receptor expressed in CHO cellMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50473529(CHEMBL165529)
Affinity DataKi:  10nMAssay Description:In vitro binding affinity against alpha-2 adrenergic receptor of rat in presence of [3H]-RX 821002 radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rat)
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM50473529(CHEMBL165529)
Affinity DataKi:  16nMAssay Description:In vitro binding affinity was determined against serotonin reuptake site of rat in presence of [3H]paroxetine radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransporter(Rat)
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM50473529(CHEMBL165529)
Affinity DataKi:  200nMAssay Description:In vitro binding affinity was determined against NA (noradrenaline) reuptake site of rat in presence of [3H]nisoxetine radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
Institut De Recherches Servier

Curated by PDSP Ki Database
LigandPNGBDBM50473529(CHEMBL165529)
Affinity DataKi:  794nMAssay Description:In vitro binding affinity against alpha-1 adrenergic receptor of rat in presence of [3H]-prazosin radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed