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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
8
hits in this display
Target
5-hydroxytryptamine receptor 3A/3B
(Rat)
Searle Research and Development
Curated by
ChEMBL
Ligand
BDBM50368604
(CHEMBL1907770)
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Affinity Data
Ki: 0.230nM
Assay Description:
Inhibition of [3H]GR-65630 binding to 5-hydroxytryptamine 3 receptor
More data for this Ligand-Target Pair
Target Info
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CHEMBL
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PC sid
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Article
PubMed
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Target
Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor
(Rat)
Searle Research and Development
Curated by
ChEMBL
Ligand
BDBM50368604
(CHEMBL1907770)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
The ability to inhibit [3H]rauwolscine binding to alpha-2 adrenergic receptor in rat cortex
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Article
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Target
Beta-1/Beta-2/Beta-3 adrenergic receptor
(Rat)
Searle Research and Development
Curated by
ChEMBL
Ligand
BDBM50368604
(CHEMBL1907770)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
The ability to inhibit [3H]dihydroalprenolol prenolol binding to Beta adrenergic receptor in rat whole brain
More data for this Ligand-Target Pair
Target Info
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Article
PubMed
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Target
Serotonin 2 (5-HT2) receptor
(Rat)
Searle Research and Development
Curated by
ChEMBL
Ligand
BDBM50368604
(CHEMBL1907770)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
The ability to inhibit [3H]ketanserin binding to 5-hydroxytryptamine 2 receptor in rat whole brain
More data for this Ligand-Target Pair
Target Info
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Article
PubMed
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Target
Alpha-1A adrenergic receptor
(Rat)
Searle Research and Development
Curated by
ChEMBL
Ligand
BDBM50368604
(CHEMBL1907770)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
The ability to inhibit [3H]prazosin binding to Alpha-1 adrenergic receptor in rat whole brain
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Target Info
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Article
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Target
D(2) dopamine receptor
(Rat)
Searle Research and Development
Curated by
ChEMBL
Ligand
BDBM50368604
(CHEMBL1907770)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
The ability to inhibit [3H]domperidone binding to dopamine receptor D2 in rat striata
More data for this Ligand-Target Pair
Target Info
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CHEMBL
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Article
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Target
5-hydroxytryptamine receptor 1A/1B/1D/1F
(Rat)
Searle Research and Development
Curated by
ChEMBL
Ligand
BDBM50368604
(CHEMBL1907770)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
The ability to inhibit [3H]5-HT binding to 5-hydroxytryptamine 1 receptor in rat cortex
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
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Ligand Info
CHEMBL
PC cid
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In Depth
Details
Article
PubMed
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Target
D(1A) dopamine receptor
(Rat)
Searle Research and Development
Curated by
ChEMBL
Ligand
BDBM50368604
(CHEMBL1907770)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
The ability to inhibit [3H]-SCH- 23390 binding to Dopamine receptor D1 in rat striata
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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