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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

LigandPNGBDBM50469634(CHEMBL433033)
Affinity DataKi:  4.60nMAssay Description:In vitro binding affinity at Alpha-2 adrenergic receptor in rat cortex by radioligand binding assay using [3H]rauwolscineMore data for this Ligand-Target Pair
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TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))TBA
LigandPNGBDBM50469634(CHEMBL433033)
Affinity DataKi:  189nMAssay Description:In vitro binding affinity at Alpha-1 adrenergic receptor by radioligand binding assay using [3H]prazosinMore data for this Ligand-Target Pair
In DepthDetails Article