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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetD(1A) dopamine receptor(Rat)
University of Crete

Curated by ChEMBL
LigandPNGBDBM50098073(1-Benzyl-1,2,3,4,4a,5,10,10a-octahydro-benzo[g]qui...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibitition of binding of [3H]-SCH-23,390 to Dopamine receptor D1 in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50098073(1-Benzyl-1,2,3,4,4a,5,10,10a-octahydro-benzo[g]qui...)
Affinity DataIC50:  5.90E+3nMAssay Description:Inhibition of binding of [3H]rauwolscine to Alpha-2 adrenergic receptor in rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50098073(1-Benzyl-1,2,3,4,4a,5,10,10a-octahydro-benzo[g]qui...)
Affinity DataIC50:  5.90E+3nMAssay Description:Inhibition of binding of [3H]rauwolscine to Alpha-2 adrenergic receptor in rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
University of Crete

Curated by ChEMBL
LigandPNGBDBM50098073(1-Benzyl-1,2,3,4,4a,5,10,10a-octahydro-benzo[g]qui...)
Affinity DataIC50:  2.18E+5nMAssay Description:Inhibition of binding of [3H]prazosin to Alpha-1 adrenergic receptor in rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rat)
University of Crete

Curated by ChEMBL
LigandPNGBDBM50098073(1-Benzyl-1,2,3,4,4a,5,10,10a-octahydro-benzo[g]qui...)
Affinity DataIC50:  2.18E+5nMAssay Description:Inhibition of binding of [3H]prazosin to Alpha-1 adrenergic receptor in rat cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed