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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
8
hits in this display
Target
F-box/LRR-repeat protein 19
(Homo sapiens)
University Of Virginia
Curated by
ChEMBL
Ligand
BDBM50594531
(CHEMBL5198555)
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Affinity Data
IC50: 2.17E+4nM
Assay Description:
Inhibition of GST-tagged human FBXL19 (31 to 86 residues) expressed in Escherichia coli BL21 cells incubated for 30 mins by fluorescence polarization...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
PubMed
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Target
CXXC-type zinc finger protein 4
(Homo sapiens)
University Of Virginia
Curated by
ChEMBL
Ligand
BDBM50594531
(CHEMBL5198555)
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Affinity Data
IC50: 2.30E+4nM
Assay Description:
Inhibition of GST-tagged human IDAX (130 to 181 residues) expressed in Escherichia coli BL21 cells incubated for 30 mins by fluorescence polarization...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
PubMed
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Target
Lysine-specific demethylase 2A
(Homo sapiens (Human))
University Of Virginia
Curated by
ChEMBL
Ligand
BDBM50594531
(CHEMBL5198555)
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Affinity Data
IC50: 3.00E+4nM
Assay Description:
Inhibition of GST-tagged human KDM2A (562 to 618 residues) expressed in Escherichia coli BL21 cells incubated for 30 mins by fluorescence polarizatio...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
PubMed
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Target
Methylcytosine dioxygenase TET3
(Homo sapiens)
University Of Virginia
Curated by
ChEMBL
Ligand
BDBM50594531
(CHEMBL5198555)
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Affinity Data
IC50: 3.30E+4nM
Assay Description:
Inhibition of GST-tagged human TET3 (49 to 68 residues) expressed in Escherichia coli BL21 cell incubated for 30 mins by fluorescence polarization as...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
PubMed
Copy BDB DOI
Target
Lysine-specific demethylase 2B
(Homo sapiens (Human))
University Of Virginia
Curated by
ChEMBL
Ligand
BDBM50594531
(CHEMBL5198555)
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Affinity Data
IC50: 3.50E+4nM
Assay Description:
Inhibition of GST-tagged human KDM2B (604 to 660 residues) expressed in Escherichia coli BL21 cells incubated for 30 mins by fluorescence polarizatio...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
PubMed
Copy BDB DOI
Target
Histone-lysine N-methyltransferase 2A
(Homo sapiens (Human))
University Of Virginia
Curated by
ChEMBL
Ligand
BDBM50594531
(CHEMBL5198555)
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Affinity Data
IC50: 4.60E+4nM
Assay Description:
Inhibition of GST-tagged human MLL1 (1147 to 1203 residues) expressed in Escherichia coli BL21 cells incubated for 30 mins by fluorescence polarizati...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
PubMed
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Target
CXXC-type zinc finger protein 5
(Homo sapiens)
University Of Virginia
Curated by
ChEMBL
Ligand
BDBM50594531
(CHEMBL5198555)
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Affinity Data
IC50: 5.30E+4nM
Assay Description:
Inhibition of GST-tagged human CXXC5 (255 to 305 residues) expressed in Escherichia coli BL21 cells incubated for 30 mins by fluorescence polarizatio...
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
PubMed
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Target
Methylcytosine dioxygenase TET1
(Homo sapiens)
University Of Virginia
Curated by
ChEMBL
Ligand
BDBM50594531
(CHEMBL5198555)
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Affinity Data
IC50: 1.07E+5nM
Assay Description:
Inhibition of GST-tagged human TET1 (583 to 633 residues) expressed in Escherichia coli BL21 cells incubated for 30 mins by fluorescence polarization...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
PubMed
Copy BDB DOI