Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetAmine oxidase [flavin-containing] A/B(Homo sapiens (Human))
Universit£

Curated by ChEMBL

LigandBDBM50474215(CHEMBL2092860)Copy SMILESCopy InChI

Affinity DataKi:  100nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 of rabbit kidney membranesMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
antibodypediaantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
Universit£

Curated by ChEMBL

LigandBDBM50474215(CHEMBL2092860)Copy SMILESCopy InChI

Affinity DataKi:  1.59E+3nMAssay Description:Displacement of [3H]clonidine from rat cortex membrane Alpha-2 adrenergic receptorsMore data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetNischarin(RAT)TBA

LigandBDBM50474215(CHEMBL2092860)Copy SMILESCopy InChI

Affinity DataKi:  7.24E+3nMAssay Description:Binding affinity to I1 imidazoline binding site in Rattus norvegicus (rat) PC12 cellsMore data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails Article
Copy BDB DOI

TargetNischarin(Homo sapiens (Human))
Universit£

Curated by ChEMBL

LigandBDBM50474215(CHEMBL2092860)Copy SMILESCopy InChI

Affinity DataKi:  7.24E+3nMAssay Description:Displacement of [125I]p-iodoclonidine from imidazoline receptor I-1 in rat pheochromocytoma cellsMore data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI