Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

TargetNischarin(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50091345(CHEMBL2092861)
Affinity DataKi:  1.10nMAssay Description:Displacement of [125I]-p-iodoclonidin from I1-imidazoline receptor in rat PC12 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50091345(CHEMBL2092861)
Affinity DataKi:  1.10nMAssay Description:Displacement of [125I]PIC from Imidazoline-1 receptor in rat PC12 cell membrane by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(Rat)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50091345(CHEMBL2092861)
Affinity DataKi:  1.10nMAssay Description:Binding affinity to I1 imidazoline binding site in Rattus norvegicus (rat) PC12 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNischarin(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50091345(CHEMBL2092861)
Affinity DataKi:  1.10nMAssay Description:Displacement of [125I]p-iodoclonidine from imidazoline receptor I-1 in rat pheochromocytoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50091345(CHEMBL2092861)
Affinity DataKi:  145nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 of rabbit kidney membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50091345(CHEMBL2092861)
Affinity DataKi:  5.01E+3nMAssay Description:Displacement of [3H]clonidine from rat cortex membrane Alpha-2 adrenergic receptorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed